HK1082743A1 - Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof - Google Patents

Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof

Info

Publication number
HK1082743A1
HK1082743A1 HK06102572A HK06102572A HK1082743A1 HK 1082743 A1 HK1082743 A1 HK 1082743A1 HK 06102572 A HK06102572 A HK 06102572A HK 06102572 A HK06102572 A HK 06102572A HK 1082743 A1 HK1082743 A1 HK 1082743A1
Authority
HK
Hong Kong
Prior art keywords
optionally substituted
group etc
alkyl group
chem
general formula
Prior art date
Application number
HK06102572A
Other languages
English (en)
Inventor
Teranishi Hirotaka
Fuschimi Nobuhico
Yonekubo Shigeru
Shimizu Kazuo
Shibazaki Toshihide
Isaji Masayuki
Original Assignee
Kissei Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical filed Critical Kissei Pharmaceutical
Publication of HK1082743A1 publication Critical patent/HK1082743A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK06102572A 2002-08-08 2006-02-27 Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof HK1082743A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2002232074 2002-08-08
JP2002321729 2002-11-05
PCT/JP2003/010048 WO2004014932A1 (ja) 2002-08-08 2003-08-07 ピラゾール誘導体、それを含有する医薬組成物、その医薬用途及びその製造中間体

Publications (1)

Publication Number Publication Date
HK1082743A1 true HK1082743A1 (en) 2006-06-16

Family

ID=31719857

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06102572A HK1082743A1 (en) 2002-08-08 2006-02-27 Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof

Country Status (19)

Country Link
US (2) US7375087B2 (xx)
EP (1) EP1544208B1 (xx)
JP (1) JP4540475B2 (xx)
KR (1) KR100985502B1 (xx)
AT (1) ATE469161T1 (xx)
AU (1) AU2003254847B2 (xx)
BR (1) BRPI0313290B1 (xx)
CA (1) CA2494179C (xx)
DE (1) DE60332743D1 (xx)
ES (1) ES2345250T3 (xx)
HK (1) HK1082743A1 (xx)
IL (1) IL166748A0 (xx)
MX (1) MXPA05001549A (xx)
NO (1) NO330456B1 (xx)
NZ (1) NZ538117A (xx)
PL (1) PL213095B1 (xx)
RU (1) RU2356906C2 (xx)
TW (1) TW200413401A (xx)
WO (1) WO2004014932A1 (xx)

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Also Published As

Publication number Publication date
DE60332743D1 (de) 2010-07-08
PL213095B1 (pl) 2013-01-31
NO330456B1 (no) 2011-04-18
BR0313290A (pt) 2005-07-05
CA2494179A1 (en) 2004-02-19
BRPI0313290B1 (pt) 2016-12-06
TWI341843B (xx) 2011-05-11
KR20050059067A (ko) 2005-06-17
MXPA05001549A (es) 2005-05-05
PL375473A1 (en) 2005-11-28
JP4540475B2 (ja) 2010-09-08
EP1544208A1 (en) 2005-06-22
ATE469161T1 (de) 2010-06-15
EP1544208B1 (en) 2010-05-26
US7375087B2 (en) 2008-05-20
RU2005106259A (ru) 2005-08-27
US7655632B2 (en) 2010-02-02
KR100985502B1 (ko) 2010-10-05
AU2003254847B2 (en) 2009-06-04
NO20051209L (no) 2005-04-15
CA2494179C (en) 2012-04-24
IL166748A0 (en) 2006-01-15
AU2003254847A1 (en) 2004-02-25
EP1544208A4 (en) 2007-05-02
US20060166899A1 (en) 2006-07-27
RU2356906C2 (ru) 2009-05-27
TW200413401A (en) 2004-08-01
ES2345250T3 (es) 2010-09-20
NZ538117A (en) 2007-01-26
WO2004014932A1 (ja) 2004-02-19
JPWO2004014932A1 (ja) 2005-12-02
US20080312153A1 (en) 2008-12-18

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