TR200000837A2 - Anti-kanser bileşimleri hazırlamak için işlem ve ara maddeler. - Google Patents

Anti-kanser bileşimleri hazırlamak için işlem ve ara maddeler.

Info

Publication number
TR200000837A2
TR200000837A2 TR2000/00837A TR200000837A TR200000837A2 TR 200000837 A2 TR200000837 A2 TR 200000837A2 TR 2000/00837 A TR2000/00837 A TR 2000/00837A TR 200000837 A TR200000837 A TR 200000837A TR 200000837 A2 TR200000837 A2 TR 200000837A2
Authority
TR
Turkey
Prior art keywords
intermediates
prepare anti
cancer compositions
cancer
compositions
Prior art date
Application number
TR2000/00837A
Other languages
English (en)
Inventor
Shelton Lehner Richard
Norris Timothy
Paul Santafianos Dinos
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of TR200000837A2 publication Critical patent/TR200000837A2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/94—Nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C22—METALLURGY; FERROUS OR NON-FERROUS ALLOYS; TREATMENT OF ALLOYS OR NON-FERROUS METALS
    • C22B—PRODUCTION AND REFINING OF METALS; PRETREATMENT OF RAW MATERIALS
    • C22B15/00—Obtaining copper
    • C22B15/0002—Preliminary treatment
    • C22B15/0004—Preliminary treatment without modification of the copper constituent
    • C—CHEMISTRY; METALLURGY
    • C22—METALLURGY; FERROUS OR NON-FERROUS ALLOYS; TREATMENT OF ALLOYS OR NON-FERROUS METALS
    • C22B—PRODUCTION AND REFINING OF METALS; PRETREATMENT OF RAW MATERIALS
    • C22B15/00—Obtaining copper
    • C22B15/0063—Hydrometallurgy
    • C22B15/0065—Leaching or slurrying
    • C22B15/0067—Leaching or slurrying with acids or salts thereof
    • C22B15/0071—Leaching or slurrying with acids or salts thereof containing sulfur
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P10/00—Technologies related to metal processing
    • Y02P10/20—Recycling

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Health & Medical Sciences (AREA)
  • Mechanical Engineering (AREA)
  • Manufacturing & Machinery (AREA)
  • Metallurgy (AREA)
  • Materials Engineering (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Mevcut bulus, formül 1'in bilesimleri; ve onun farmasötik olarak uygun tuzlari ve çözeltileri ile birlikte ilgili bilesimlerin hazirlanmasi için metodlar ve ara maddelerle ilgilidir, burada R1, R2 ve R15 burada tanimlandigi gibidir. Yukaridaki bilesimler memelilerde kanser gibi hiperproliferatif bozukluklarin tedavisinde yararlidir.
TR2000/00837A 1999-03-31 2000-03-30 Anti-kanser bileşimleri hazırlamak için işlem ve ara maddeler. TR200000837A2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12707299P 1999-03-31 1999-03-31

Publications (1)

Publication Number Publication Date
TR200000837A2 true TR200000837A2 (tr) 2000-11-21

Family

ID=22428179

Family Applications (1)

Application Number Title Priority Date Filing Date
TR2000/00837A TR200000837A2 (tr) 1999-03-31 2000-03-30 Anti-kanser bileşimleri hazırlamak için işlem ve ara maddeler.

Country Status (50)

Country Link
US (1) US6476040B1 (tr)
EP (1) EP1044969B1 (tr)
JP (2) JP3420549B2 (tr)
KR (2) KR100430210B1 (tr)
CN (2) CN100351242C (tr)
AP (2) AP1655A (tr)
AR (1) AR018705A1 (tr)
AT (1) ATE348098T1 (tr)
AU (2) AU781402B2 (tr)
BG (1) BG65194B1 (tr)
BR (1) BRPI0001486B8 (tr)
CA (2) CA2302965C (tr)
CO (1) CO5160273A1 (tr)
CR (1) CR6165A (tr)
CZ (1) CZ299426B6 (tr)
DE (1) DE60032275T2 (tr)
DK (1) DK1044969T3 (tr)
DZ (1) DZ3030A1 (tr)
EA (3) EA005892B1 (tr)
EE (1) EE04589B1 (tr)
EG (1) EG22506A (tr)
ES (1) ES2278578T3 (tr)
GE (1) GEP20022653B (tr)
GT (1) GT200000037A (tr)
HK (1) HK1029790A1 (tr)
HR (1) HRP20000182B1 (tr)
HU (1) HU227698B1 (tr)
ID (1) ID25427A (tr)
IL (2) IL135245A0 (tr)
IS (1) IS2468B (tr)
MA (1) MA25087A1 (tr)
MY (1) MY136270A (tr)
NO (2) NO321952B1 (tr)
NZ (2) NZ503683A (tr)
OA (1) OA11335A (tr)
PA (1) PA8491901A1 (tr)
PE (1) PE20001599A1 (tr)
PL (1) PL339330A1 (tr)
PT (1) PT1044969E (tr)
RS (1) RS49836B (tr)
SG (2) SG121687A1 (tr)
SK (1) SK287339B6 (tr)
SV (1) SV2002000047A (tr)
TN (1) TNSN00064A1 (tr)
TR (1) TR200000837A2 (tr)
TW (1) TW553939B (tr)
UA (2) UA70928C2 (tr)
UY (1) UY26086A1 (tr)
YU (1) YU13200A (tr)
ZA (1) ZA200001586B (tr)

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IS2468B (is) 2008-12-15
HK1029790A1 (en) 2001-04-12
PE20001599A1 (es) 2001-01-18
HRP20000182B1 (en) 2007-10-31
IL168036A (en) 2006-12-10
HU0001353D0 (en) 2000-06-28
HUP0001353A3 (en) 2002-01-28
EP1044969B1 (en) 2006-12-13
GT200000037A (es) 2001-09-21
NO321952B1 (no) 2006-07-24
SG115536A1 (en) 2005-10-28
GEP20022653B (en) 2002-03-25
EA200000274A2 (ru) 2000-10-30
HRP20000182A2 (en) 2001-04-30
DZ3030A1 (fr) 2004-03-27
SK287339B6 (sk) 2010-07-07
AP2000001778A0 (en) 2000-03-31
AU2262000A (en) 2000-10-05
ATE348098T1 (de) 2007-01-15
BR0001486A (pt) 2001-05-02
NO20054715L (no) 2000-10-02
EA200201245A1 (ru) 2003-04-24
NZ512818A (en) 2003-01-31
EA004654B1 (ru) 2004-06-24
YU13200A (sh) 2002-10-18
JP4074509B2 (ja) 2008-04-09
CO5160273A1 (es) 2002-05-30
CA2302965C (en) 2004-02-17
AU2005201494A1 (en) 2005-05-05
AU781402B2 (en) 2005-05-19
DE60032275D1 (de) 2007-01-25
ZA200001586B (en) 2001-10-01
JP3420549B2 (ja) 2003-06-23
NO20001648D0 (no) 2000-03-30
EG22506A (en) 2003-03-31
EP1044969A2 (en) 2000-10-18
CZ299426B6 (cs) 2008-07-23
ID25427A (id) 2000-10-05
PL339330A1 (en) 2000-10-09
NZ503683A (en) 2001-09-28
CN1699350A (zh) 2005-11-23
CN1276370A (zh) 2000-12-13
BRPI0001486B1 (pt) 2019-01-29
BG104278A (en) 2001-08-31
EA005561B1 (ru) 2005-04-28
OA11335A (en) 2003-12-10
EA200201244A1 (ru) 2003-04-24
PT1044969E (pt) 2007-05-31
CA2427221C (en) 2008-09-16
IS5411A (is) 2000-10-02
PA8491901A1 (es) 2001-12-14
CZ20001155A3 (cs) 2001-03-14
KR100430209B1 (ko) 2004-05-03
NO20001648L (no) 2000-10-02
EA005892B1 (ru) 2005-06-30
SV2002000047A (es) 2002-01-23
SG121687A1 (en) 2006-05-26
SK4442000A3 (en) 2000-10-09
BRPI0001486B8 (pt) 2021-05-25
CR6165A (es) 2008-10-10
JP2003176274A (ja) 2003-06-24
KR100430210B1 (ko) 2004-05-03
CA2302965A1 (en) 2000-09-30
MY136270A (en) 2008-09-30
UA70928C2 (uk) 2004-11-15
CN100351242C (zh) 2007-11-28
TW553939B (en) 2003-09-21
EE200000255A (et) 2000-12-15
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EA200000274A3 (ru) 2003-02-27
HU227698B1 (en) 2011-12-28
CN1215061C (zh) 2005-08-17
DK1044969T3 (da) 2007-04-23
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BG65194B1 (bg) 2007-06-29
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NO324745B1 (no) 2007-12-03
TNSN00064A1 (fr) 2005-11-10
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RS49836B (sr) 2008-08-07
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