ES418996A1 - Un procedimiento para la preparacion de derivados de piri- midina biologicamente activos. - Google Patents
Un procedimiento para la preparacion de derivados de piri- midina biologicamente activos.Info
- Publication number
- ES418996A1 ES418996A1 ES418996A ES418996A ES418996A1 ES 418996 A1 ES418996 A1 ES 418996A1 ES 418996 A ES418996 A ES 418996A ES 418996 A ES418996 A ES 418996A ES 418996 A1 ES418996 A1 ES 418996A1
- Authority
- ES
- Spain
- Prior art keywords
- pyrimidino
- thiazepine
- oxazepine
- azepine
- dibenzo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 125000002576 diazepinyl group Chemical class N1N=C(C=CC=C1)* 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NLAANVRAGE7212915,A NL176458C (nl) | 1972-09-23 | 1972-09-23 | Werkwijze ter bereiding van een farmaceutisch preparaat en werkwijze voor de bereiding van daartoe geschikte actieve stoffen. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES418996A1 true ES418996A1 (es) | 1976-07-01 |
Family
ID=19816997
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES418996A Expired ES418996A1 (es) | 1972-09-23 | 1973-09-22 | Un procedimiento para la preparacion de derivados de piri- midina biologicamente activos. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US3892695A (es) |
| JP (1) | JPS5912678B2 (es) |
| AR (1) | AR203090A1 (es) |
| AU (1) | AU472312B2 (es) |
| BE (1) | BE805178A (es) |
| CA (1) | CA1019733A (es) |
| CH (1) | CH592094A5 (es) |
| DE (1) | DE2347727C2 (es) |
| DK (1) | DK140668B (es) |
| ES (1) | ES418996A1 (es) |
| FI (1) | FI54311C (es) |
| FR (1) | FR2199996B1 (es) |
| GB (1) | GB1445765A (es) |
| HU (1) | HU167206B (es) |
| IE (1) | IE38221B1 (es) |
| NL (1) | NL176458C (es) |
| SE (1) | SE407686B (es) |
| ZA (1) | ZA737131B (es) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4217452A (en) * | 1974-02-09 | 1980-08-12 | Akzona Incorporated | Synthesis for the preparation of tetracyclic compounds |
| NL179906C (nl) * | 1974-02-09 | 1986-12-01 | Akzo Nv | Werkwijze voor het bereiden van 1,2,3,4,10,14b-hexahydrodibenzo(c,f)pyrazino (1,2-a)azepine derivaten. |
| NL7414038A (nl) * | 1974-10-28 | 1976-05-03 | Akzo Nv | Nieuwe tetracyclische pyrrolidino derivaten. |
| GB1472382A (en) * | 1975-01-16 | 1977-05-04 | Wyeth John & Brother Ltd | Dibenzopyrimidoazepines |
| NL7610942A (nl) * | 1976-10-02 | 1978-04-04 | Akzo Nv | Werkwijze voor het bereiden van 1,4-diazepine derivaten. |
| NL7809726A (nl) * | 1978-09-26 | 1980-03-28 | Akzo Nv | Nieuwe tetracyclische verbindingen. |
| HU195491B (en) * | 1985-12-20 | 1988-05-30 | Egyt Gyogyszervegyeszeti Gyar | Process for production of optically active 2-chlor-12-/3-/dimethil-amin/-2-methil-prophil/-12h-dibenzol /d,g/ /1,3,6/-diaxazocine and medical compositions containing such compounds |
| CH678623A5 (en) * | 1989-05-17 | 1991-10-15 | Sochinaz Societe Chimique De V | Prepn. of di:benzo pyrazino azepine(s) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL154511B (nl) * | 1967-07-07 | 1977-09-15 | Organon Nv | Werkwijze ter bereiding van piperazinederivaten, werkwijze ter bereiding van een farmaceutisch preparaat, dat een dergelijke verbinding bevat en vormstukken bereid volgens deze werkwijze. |
| US3470181A (en) * | 1967-10-23 | 1969-09-30 | American Home Prod | Fused 2-pyrimidinepropionic acid compounds,related compounds,and the process for their preparation |
-
1972
- 1972-09-23 NL NLAANVRAGE7212915,A patent/NL176458C/xx not_active IP Right Cessation
-
1973
- 1973-09-06 ZA ZA737131*A patent/ZA737131B/xx unknown
- 1973-09-06 IE IE1587/73A patent/IE38221B1/xx unknown
- 1973-09-07 US US396251A patent/US3892695A/en not_active Expired - Lifetime
- 1973-09-11 AU AU60197/73A patent/AU472312B2/en not_active Expired
- 1973-09-14 GB GB4331873A patent/GB1445765A/en not_active Expired
- 1973-09-17 DK DK507673AA patent/DK140668B/da not_active IP Right Cessation
- 1973-09-18 CA CA181,312A patent/CA1019733A/en not_active Expired
- 1973-09-20 AR AR250175A patent/AR203090A1/es active
- 1973-09-20 FR FR7333768A patent/FR2199996B1/fr not_active Expired
- 1973-09-21 SE SE7312873A patent/SE407686B/sv unknown
- 1973-09-21 FI FI2963/73A patent/FI54311C/fi active
- 1973-09-21 HU HUAO373A patent/HU167206B/hu unknown
- 1973-09-21 JP JP48106809A patent/JPS5912678B2/ja not_active Expired
- 1973-09-21 BE BE135926A patent/BE805178A/xx not_active IP Right Cessation
- 1973-09-21 CH CH1358173A patent/CH592094A5/xx not_active IP Right Cessation
- 1973-09-21 DE DE2347727A patent/DE2347727C2/de not_active Expired
- 1973-09-22 ES ES418996A patent/ES418996A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| BE805178A (fr) | 1974-03-21 |
| CH592094A5 (es) | 1977-10-14 |
| IE38221B1 (en) | 1978-01-18 |
| NL7212915A (es) | 1974-03-26 |
| DE2347727A1 (de) | 1974-04-04 |
| DE2347727C2 (de) | 1986-12-11 |
| ZA737131B (en) | 1974-08-28 |
| NL176458B (nl) | 1984-11-16 |
| FR2199996A1 (es) | 1974-04-19 |
| FI54311C (fi) | 1978-11-10 |
| FR2199996B1 (es) | 1977-09-09 |
| JPS4985098A (es) | 1974-08-15 |
| AR203090A1 (es) | 1975-08-14 |
| AU472312B2 (en) | 1976-05-20 |
| HU167206B (es) | 1975-09-27 |
| NL176458C (nl) | 1985-04-16 |
| SE407686B (sv) | 1979-04-09 |
| JPS5912678B2 (ja) | 1984-03-24 |
| GB1445765A (en) | 1976-08-11 |
| DK140668C (es) | 1980-03-24 |
| US3892695A (en) | 1975-07-01 |
| DK140668B (da) | 1979-10-22 |
| AU6019773A (en) | 1975-03-13 |
| FI54311B (fi) | 1978-07-31 |
| IE38221L (en) | 1974-03-23 |
| CA1019733A (en) | 1977-10-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19880218 |