UY29838A1 - Derivados sustituidos de 4,5,6,7-tetrahidropirrolo(3,2,c)piridin-4-ona y de 4,5-tetrahidropirrolo(3,2,c)piridin-4-ona, composiciones farmacéuticas conteniéndolos, procesos de preparación y aplicaciones - Google Patents

Derivados sustituidos de 4,5,6,7-tetrahidropirrolo(3,2,c)piridin-4-ona y de 4,5-tetrahidropirrolo(3,2,c)piridin-4-ona, composiciones farmacéuticas conteniéndolos, procesos de preparación y aplicaciones

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Publication number
UY29838A1
UY29838A1 UY29838A UY29838A UY29838A1 UY 29838 A1 UY29838 A1 UY 29838A1 UY 29838 A UY29838 A UY 29838A UY 29838 A UY29838 A UY 29838A UY 29838 A1 UY29838 A1 UY 29838A1
Authority
UY
Uruguay
Prior art keywords
tetrahidropirrolo
piridin
ona
processes
pharmaceutical compositions
Prior art date
Application number
UY29838A
Other languages
English (en)
Inventor
Leifeng Cheng
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37781800&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29838(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY29838A1 publication Critical patent/UY29838A1/es

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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  • Orthopedic Medicine & Surgery (AREA)

Abstract

La presente invención se refiere a compuestos 4,5,6,7-tetrahidropirrolo(3,2-c)piridin-4-ona y 4,5-dihidropirrolo(3,2-c)piridin-4-ona de fórmula I y a procesos para preparar dichos compuestos, a su uso en el tratamiento de obesidad, trastornos psiquiátricos y neurológicos, a métodos para su uso terapéutico y a composiciones farmacéuticas que los contienen.
UY29838A 2005-10-06 2006-10-04 Derivados sustituidos de 4,5,6,7-tetrahidropirrolo(3,2,c)piridin-4-ona y de 4,5-tetrahidropirrolo(3,2,c)piridin-4-ona, composiciones farmacéuticas conteniéndolos, procesos de preparación y aplicaciones UY29838A1 (es)

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KR20080058456A (ko) 2008-06-25
US20080312269A1 (en) 2008-12-18
ZA200802946B (en) 2009-03-25
EP1937679B1 (en) 2009-08-19
WO2007039740A3 (en) 2007-05-31
EP1937679A2 (en) 2008-07-02
JP4277062B2 (ja) 2009-06-10
ECSP088413A (es) 2008-05-30
BRPI0616653A2 (pt) 2011-06-28
US20080009513A1 (en) 2008-01-10
WO2007039740A2 (en) 2007-04-12
RU2415856C2 (ru) 2011-04-10
US7875626B2 (en) 2011-01-25
AR056560A1 (es) 2007-10-10
ATE440099T1 (de) 2009-09-15
RU2008109185A (ru) 2009-11-20
IL190025A0 (en) 2008-08-07
CA2624495A1 (en) 2007-04-12
CN101277957A (zh) 2008-10-01
JP2009504722A (ja) 2009-02-05
ES2329616T3 (es) 2009-11-27
US7576095B2 (en) 2009-08-18
HK1122808A1 (en) 2009-05-29
AU2006298530A1 (en) 2007-04-12
AU2006298530B2 (en) 2009-10-29
NO20081523L (no) 2008-07-02
TW200730525A (en) 2007-08-16

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