ECSP088413A - Preparación y uso de derivados de tetrahidropirrolo[3,2-c]piridin-4-ona para el tratamiento de la obesidad, trastornos psiquiátricos y neurológicos - Google Patents

Preparación y uso de derivados de tetrahidropirrolo[3,2-c]piridin-4-ona para el tratamiento de la obesidad, trastornos psiquiátricos y neurológicos

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Publication number
ECSP088413A
ECSP088413A EC2008008413A ECSP088413A ECSP088413A EC SP088413 A ECSP088413 A EC SP088413A EC 2008008413 A EC2008008413 A EC 2008008413A EC SP088413 A ECSP088413 A EC SP088413A EC SP088413 A ECSP088413 A EC SP088413A
Authority
EC
Ecuador
Prior art keywords
psychiatric
obesity
treatment
neurological disorders
tetrahydropirrolo
Prior art date
Application number
EC2008008413A
Other languages
English (en)
Inventor
Leifeng Cheng
Original Assignee
Astrazeneca Ab
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37781800&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP088413(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of ECSP088413A publication Critical patent/ECSP088413A/es

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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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Abstract

La presente invención se refiere a compuestos de 4, 5, 6, 7 -tetrahidropirrolo[3,2-c]piridin-4-ona y 4, 5-dihidropirrolo[3,2-c]piridin-4-ona de la fórmula (I) y a procesos para preparar dichos compuestos, a su uso en el tratamiento de la obesidad, trastornos psiquiátricos y neurológicos, a métodos para su uso terapéutico y a composiciones farmacéuticas que los contienen.
EC2008008413A 2005-10-06 2008-04-30 Preparación y uso de derivados de tetrahidropirrolo[3,2-c]piridin-4-ona para el tratamiento de la obesidad, trastornos psiquiátricos y neurológicos ECSP088413A (es)

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KR20080058456A (ko) 2008-06-25
US20080312269A1 (en) 2008-12-18
ZA200802946B (en) 2009-03-25
EP1937679B1 (en) 2009-08-19
WO2007039740A3 (en) 2007-05-31
EP1937679A2 (en) 2008-07-02
JP4277062B2 (ja) 2009-06-10
BRPI0616653A2 (pt) 2011-06-28
US20080009513A1 (en) 2008-01-10
WO2007039740A2 (en) 2007-04-12
RU2415856C2 (ru) 2011-04-10
US7875626B2 (en) 2011-01-25
AR056560A1 (es) 2007-10-10
ATE440099T1 (de) 2009-09-15
RU2008109185A (ru) 2009-11-20
IL190025A0 (en) 2008-08-07
CA2624495A1 (en) 2007-04-12
CN101277957A (zh) 2008-10-01
JP2009504722A (ja) 2009-02-05
ES2329616T3 (es) 2009-11-27
US7576095B2 (en) 2009-08-18
HK1122808A1 (en) 2009-05-29
AU2006298530A1 (en) 2007-04-12
AU2006298530B2 (en) 2009-10-29
UY29838A1 (es) 2007-05-31
NO20081523L (no) 2008-07-02
TW200730525A (en) 2007-08-16

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