SE393376B - Forfarande for framstellning av pyrimidinonderivat - Google Patents

Forfarande for framstellning av pyrimidinonderivat

Info

Publication number: SE393376B
Authority: SE; Sweden
Prior art keywords: pyrimidinon; derivatives; preparing; procedure; pyrimidinon derivatives
Prior art date: 1971-10-29

Application number

SE7212358A

Other languages

English (en)

Swedish (sv)

Inventor

C A Lipinski

J G Stam

G G Deangelis

H-J E Hess

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1971-10-29

Filing date

1972-09-25

Publication date

1977-05-09

1972-09-25 Application filed by Pfizer filed Critical Pfizer

1977-05-09 Publication of SE393376B publication Critical patent/SE393376B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/56—One oxygen atom and one sulfur atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/52—Two oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/60—Three or more oxygen or sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Epidemiology (AREA)
Pulmonology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

SE7212358A 1971-10-29 1972-09-25 Forfarande for framstellning av pyrimidinonderivat SE393376B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US19400671A	1971-10-29	1971-10-29

Publications (1)

Publication Number	Publication Date
SE393376B true SE393376B (sv)	1977-05-09

Family

ID=22715935

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
SE7212358A SE393376B (sv)	1971-10-29	1972-09-25	Forfarande for framstellning av pyrimidinonderivat
SE7505279A SE397090B (sv)	1971-10-29	1975-05-06	Forfarande for framstellning av hydroxipyrimidiner

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
SE7505279A SE397090B (sv)	1971-10-29	1975-05-06	Forfarande for framstellning av hydroxipyrimidiner

Country Status (25)

Country	Link
JP (2)	JPS5337870B2 (de)
AR (2)	AR198798A1 (de)
AT (2)	AT321308B (de)
AU (1)	AU467600B2 (de)
BE (1)	BE790125A (de)
CA (1)	CA980778A (de)
CH (2)	CH555832A (de)
DE (3)	DE2248741C3 (de)
DK (1)	DK131465B (de)
EG (1)	EG11013A (de)
ES (2)	ES407730A1 (de)
FI (1)	FI55503C (de)
FR (1)	FR2157865B1 (de)
GB (2)	GB1377308A (de)
IE (1)	IE37043B1 (de)
IL (2)	IL40458A (de)
LU (1)	LU66304A1 (de)
NL (1)	NL166470C (de)
NO (1)	NO136574C (de)
PH (2)	PH10129A (de)
PL (2)	PL84634B1 (de)
SE (2)	SE393376B (de)
SU (2)	SU498908A3 (de)
YU (2)	YU35125B (de)
ZA (1)	ZA727362B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS55151912U (de) *	1979-04-17	1980-11-01
JPS5752409Y2 (de) *	1979-11-05	1982-11-15
DE3222914A1 (de) *	1982-06-18	1983-12-22	Beiersdorf Ag, 2000 Hamburg	Substituierte 5-phenylthio-6-amino-pyrimidinone, verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen
JPH0655686B2 (ja) *	1988-08-30	1994-07-27	宇部興産株式会社	ｐ−ブロモフェノキシアセトアルデヒドジアルキルアセタール類の製造方法
ATE533488T1 (de)	2005-08-22	2011-12-15	Melior Pharmaceuticals I Inc	Verfahren und formulierungen zur modulierung von lyn-kinaseaktivität und behandlung assoziierter erkrankungen
US8552184B2 (en)	2008-07-03	2013-10-08	Melior Pharmaceuticals I, Inc.	Compounds and methods for treating disorders related to glucose metabolism
US20130158055A1 (en)	2010-05-28	2013-06-20	Andrew G. Reaume	Prevention Of Pancreatic Beta Cell Degeneration
EP3609500B1 (de)	2017-04-10	2024-11-13	Melior Pharmaceuticals I, Inc.	Behandlung von adipozyten

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US2913462A (en) *		1959-11-17		Eahl h
GB951432A (en) *	1959-03-17	1964-03-04	Wellcome Found	Pyrimidine derivatives and the manufacture thereof

0
- BE BE790125D patent/BE790125A/xx not_active IP Right Cessation
1972
- 1972-02-18 GB GB774872A patent/GB1377308A/en not_active Expired
- 1972-02-18 GB GB5005373A patent/GB1377720A/en not_active Expired
- 1972-09-25 SE SE7212358A patent/SE393376B/xx unknown
- 1972-09-28 IL IL40458A patent/IL40458A/en unknown
- 1972-09-28 AU AU47228/72A patent/AU467600B2/en not_active Expired
- 1972-10-02 PH PH13959A patent/PH10129A/en unknown
- 1972-10-05 DE DE2248741A patent/DE2248741C3/de not_active Expired
- 1972-10-05 DE DE2264374A patent/DE2264374C3/de not_active Expired
- 1972-10-05 DE DE2264657A patent/DE2264657C2/de not_active Expired
- 1972-10-06 AT AT858972A patent/AT321308B/de not_active IP Right Cessation
- 1972-10-06 AT AT00933/74A patent/AT320656B/de not_active IP Right Cessation
- 1972-10-12 FI FI2825/72A patent/FI55503C/fi active
- 1972-10-12 YU YU2551/72A patent/YU35125B/xx unknown
- 1972-10-13 SU SU1839308A patent/SU498908A3/ru active
- 1972-10-13 NO NO3686/72A patent/NO136574C/no unknown
- 1972-10-16 NL NL7213959.A patent/NL166470C/xx not_active IP Right Cessation
- 1972-10-16 ZA ZA727362A patent/ZA727362B/xx unknown
- 1972-10-16 CA CA153,956A patent/CA980778A/en not_active Expired
- 1972-10-16 JP JP10279972A patent/JPS5337870B2/ja not_active Expired
- 1972-10-16 DK DK510072AA patent/DK131465B/da not_active IP Right Cessation
- 1972-10-16 IE IE1398/72A patent/IE37043B1/xx unknown
- 1972-10-16 FR FR7236560A patent/FR2157865B1/fr not_active Expired
- 1972-10-16 CH CH1507872A patent/CH555832A/fr not_active IP Right Cessation
- 1972-10-16 PL PL1972158297A patent/PL84634B1/pl unknown
- 1972-10-16 CH CH165674A patent/CH549579A/fr not_active IP Right Cessation
- 1972-10-16 PL PL1972174103A patent/PL89852B1/pl unknown
- 1972-10-16 LU LU66304A patent/LU66304A1/xx unknown
- 1972-10-18 ES ES407730A patent/ES407730A1/es not_active Expired
- 1972-10-19 EG EG431/72A patent/EG11013A/xx active
- 1972-10-23 AR AR244763A patent/AR198798A1/es active
1973
- 1973-07-12 AR AR249053A patent/AR196263A1/es active
1974
- 1974-03-26 SU SU2008490A patent/SU505362A3/ru active
1975
- 1975-04-15 ES ES436624A patent/ES436624A1/es not_active Expired
- 1975-05-06 SE SE7505279A patent/SE397090B/xx unknown
- 1975-11-21 PH PH17784A patent/PH11594A/en unknown
1976
- 1976-01-05 IL IL48790A patent/IL48790A/en unknown
1978
- 1978-02-08 JP JP1336078A patent/JPS53116386A/ja active Granted
1979
- 1979-04-25 YU YU991/79A patent/YU36295B/xx unknown

Also Published As

Publication number	Publication date
DE2264374A1 (de)	1973-05-24
PH10129A (en)	1976-09-02
NL166470C (nl)	1981-08-17
YU36295B (en)	1982-06-18
YU255172A (en)	1980-03-15
FR2157865B1 (de)	1975-10-31
PH11594A (en)	1978-03-31
DE2264374C3 (de)	1981-07-23
GB1377308A (en)	1974-12-11
JPS4852780A (de)	1973-07-24
AU467600B2 (en)	1975-12-04
IE37043B1 (en)	1977-04-27
NL166470B (nl)	1981-03-16
AU4722872A (en)	1974-04-04
DE2264657C2 (de)	1982-09-16
EG11013A (en)	1976-11-30
AR198798A1 (es)	1974-07-24
CH555832A (fr)	1974-11-15
CH549579A (fr)	1974-05-31
DK131465C (de)	1975-12-08
YU99179A (en)	1981-08-31
DE2248741A1 (de)	1973-05-03
SU505362A3 (ru)	1976-02-28
JPS5422995B2 (de)	1979-08-10
AT321308B (de)	1975-03-25
IL40458A0 (en)	1972-11-28
BE790125A (fr)	1973-04-16
SE7505279L (sv)	1975-05-06
SE397090B (sv)	1977-10-17
IL40458A (en)	1976-05-31
GB1377720A (en)	1974-12-18
DE2248741B2 (de)	1974-11-14
FI55503B (fi)	1979-04-30
ZA727362B (en)	1973-11-28
YU35125B (en)	1980-09-25
PL89852B1 (de)	1976-12-31
DE2264657A1 (de)	1974-06-20
DK131465B (da)	1975-07-21
DE2248741C3 (de)	1975-06-26
JPS53116386A (en)	1978-10-11
FR2157865A1 (de)	1973-06-08
ES436624A1 (es)	1977-02-01
CA980778A (en)	1975-12-30
JPS5337870B2 (de)	1978-10-12
IE37043L (en)	1973-04-29
NL7213959A (de)	1973-05-02
ES407730A1 (es)	1976-01-16
NO136574B (de)	1977-06-20
IL48790A0 (en)	1976-03-31
NO136574C (no)	1977-09-28
IL48790A (en)	1976-05-31
AT320656B (de)	1975-02-25
SU498908A3 (ru)	1976-01-05
PL84634B1 (de)	1976-04-30
FI55503C (fi)	1979-08-10
AR196263A1 (es)	1973-12-10
DE2264374B2 (de)	1980-08-07
LU66304A1 (de)	1973-05-03

Publication	Publication Date	Title
SE422325B (sv)	1982-03-01	Forfarande for framstellning av vissa angivna 1,2,4-triazolderivat
SE432102B (sv)	1984-03-19	Forfarande for framstellning av estrar av penicilliner
SE398877B (sv)	1978-01-23	Forfarande for framstellning av 14-hydroxi-morfinanderivat
SE400771B (sv)	1978-04-10	Forfarande for framstellning av 3alfa-hydroxi- och 3alfa-hydroxi-19-norpregnaner
SE413246B (sv)	1980-05-12	Forfarande for framstellning av kolesteroloxidas
SE383358B (sv)	1976-03-08	Forfarande for framstellning av pullulan
SE399268B (sv)	1978-02-06	Forfarande for framstellning av nya purinnukleosidderivat
NO145918C (no)	1982-06-23	Fremgangsmaate for fremstilling av 7-acylamido-3-cefem-4-karboksylsyrer
SE419339B (sv)	1981-07-27	Forfarande for framstellning av substituerade sulfonylacetamidocefalosporiner
SE397530B (sv)	1977-11-07	Forfarande for framstellning av 1-pyrazolylalkyl-4-arylpiperazinderivat
NO139124C (no)	1979-01-10	Fremgangsmaate for fremstilling av estere
SE382809B (sv)	1976-02-16	Forfarande for framstellning av fenoxiettiksyraderivat
AR200387A1 (es)	1974-11-08	Procedimiento para preparar derivados de trifluorometilfenilpiperazina
SE423092B (sv)	1982-04-13	Forfarande for framstellning av vissa 13-tiaprostaglandiner
SE417711B (sv)	1981-04-06	Forfarande for framstellning av 5-iminometyl-2-nitroimidazolderivat
SE393376B (sv)	1977-05-09	Forfarande for framstellning av pyrimidinonderivat
SE395455B (sv)	1977-08-15	Forfarande for framstellning av 3-(fenyl-piperazinyl) etylindoliner
SE384686B (sv)	1976-05-17	Forfarande for framstellning av linkomycinderivat
SE387344B (sv)	1976-09-06	Forfarande for framstellning av pyrazin-4-oxidderivat
SE408177B (sv)	1979-05-21	Forfarande for framstellning av 4-hydroximetyl-1-ftalazonderivat
SE409858B (sv)	1979-09-10	Forfarande for framstallning av vissa angivna aminoalkylfenylacetonitrilderivat
SE380528B (sv)	1975-11-10	Forfarande for framstellning av 2-klor-7-hydroxi-11-piperazinyldibensoxazepmderivat
SE373572B (sv)	1975-02-10	Forfarande for framstellning av pyroglutamyl-histidyl-prolinamid
SE402454B (sv)	1978-07-03	Forfarande for framstellning av 2-alkoxi-5-alkylsulfonyl-toluen
IT966747B (it)	1974-02-20	Procedimento per preparare dinitroantrachinoni