SE7409946L - - Google Patents

Info

Publication number: SE7409946L
Authority: SE; Sweden
Prior art keywords: gentamicin; antibiotic; mutamicin; diaminocyclitols; aminoglycosyl
Prior art date: 1973-08-06

Application number

SE7409946A

Other languages

English (en)

Other versions

SE424994B (sv

Inventor

M J Weinstein

P J L Daniels

G H Wagman

R Testa

A K Mallams

J J Wright

T L Nagabhushan

Original Assignee

Scherico Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-08-06

Filing date

1974-08-01

Publication date

1975-02-07

1974-03-19 Priority claimed from US05/452,586 external-priority patent/US4029882A/en

1974-08-01 Application filed by Scherico Ltd filed Critical Scherico Ltd

1975-02-07 Publication of SE7409946L publication Critical patent/SE7409946L/xx

1982-08-23 Publication of SE424994B publication Critical patent/SE424994B/xx

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Polysaccharides And Polysaccharide Derivatives (AREA)

SE7409946A 1973-08-06 1974-08-01 Forfarande for framstellning av nya pseudotrisackarider SE424994B (sv)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US38575173A	1973-08-06	1973-08-06
US45260074A	1974-03-19	1974-03-19
US05/452,586 US4029882A (en)	1974-03-19	1974-03-19	Selective acylation of the C-1 amino group of aminoglycoside antibiotics

Publications (2)

Publication Number	Publication Date
SE7409946L true SE7409946L (de)	1975-02-07
SE424994B SE424994B (sv)	1982-08-23

Family

ID=27409729

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7409946A SE424994B (sv)	1973-08-06	1974-08-01	Forfarande for framstellning av nya pseudotrisackarider

Country Status (20)

Country	Link
AR (1)	AR215834A1 (de)
BE (1)	BE818431A (de)
BG (1)	BG25804A3 (de)
CH (1)	CH606076A5 (de)
CY (1)	CY1018A (de)
DD (1)	DD119037A5 (de)
DE (2)	DE2437160C3 (de)
DK (1)	DK146298C (de)
FI (1)	FI62100C (de)
FR (1)	FR2240015B1 (de)
GB (1)	GB1473733A (de)
HK (1)	HK55179A (de)
IE (1)	IE40437B1 (de)
IL (1)	IL45385A (de)
KE (1)	KE2981A (de)
LU (1)	LU70661A1 (de)
MY (1)	MY8000090A (de)
NL (1)	NL171587C (de)
NO (1)	NO139483C (de)
SE (1)	SE424994B (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4217446A (en)	1974-10-26	1980-08-12	Pfizer Inc.	ωAmino-2-hydroxyalkyl derivatives of aminoglycoside antibiotics
GB1464401A (en) *	1974-10-26	1977-02-16	Pfizer Ltd	Aminoglycosides
FR2405266A1 (fr) *	1975-09-08	1979-05-04	Scherico Ltd	Nouveaux pseudotrisaccharides, et applications pharmaceutiques de ceux-ci
EP0000057B1 (de) *	1977-06-10	1982-07-14	Bayer Ag	Selektiv geschützte 4,6-Di-O-(aminoglycosyl)-1,3-diaminocyclitole
US4282350A (en) *	1977-08-05	1981-08-04	Schering Corporation	Selective 3"-N-acylation of 1,3"-di-N-unprotected-poly-N-protected-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols
JPS5492951A (en) *	1977-12-29	1979-07-23	Shionogi & Co Ltd	Novel aminoglycoside derivative
JPS5538345A (en) *	1978-09-11	1980-03-17	Shionogi & Co Ltd	Novel aminoglycoside derivative
DE2840907A1 (de) *	1978-09-20	1980-04-03	Bayer Ag	Selektiv geschuetzte 4,6-di-o-(aminoglykosyl)-1,3-diaminocyclitole
DE2928183A1 (de) *	1979-07-12	1981-01-29	Bayer Ag	1-n-alkylsisomicin-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
CN1040177C (zh) *	1993-04-23	1998-10-14	江苏省微生物研究所	一种含1-N-乙基庆大霉素C1a或其盐的药用制剂及制备方法
CN101868472B (zh)	2007-11-21	2013-05-29	尔察祯有限公司	抗菌性氨基糖苷类似物
WO2010132768A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of sisomicin
WO2010132760A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of tobramycin
WO2010132765A2 (en) *	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132759A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of dibekacin
WO2010132757A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
CN101575311B (zh) *	2009-06-19	2011-05-04	无锡好芳德药业有限公司	一种制备褪黑素的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1235311B (de) *	1963-03-25	1967-03-02	Roussel Uclaf	Verfahren zur Herstellung von N-Monophenylaethylneomycin B bzw. seinen therapeutisch vertraeglichen Salzen

1974
- 1974-07-31 CH CH1060274A patent/CH606076A5/xx not_active IP Right Cessation
- 1974-08-01 DE DE2437160A patent/DE2437160C3/de not_active Expired
- 1974-08-01 FR FR7426815A patent/FR2240015B1/fr not_active Expired
- 1974-08-01 AR AR255007A patent/AR215834A1/es active
- 1974-08-01 NL NLAANVRAGE7410363,A patent/NL171587C/xx not_active IP Right Cessation
- 1974-08-01 DK DK412474A patent/DK146298C/da not_active IP Right Cessation
- 1974-08-01 NO NO742787A patent/NO139483C/no unknown
- 1974-08-01 CY CY1018A patent/CY1018A/xx unknown
- 1974-08-01 SE SE7409946A patent/SE424994B/xx not_active IP Right Cessation
- 1974-08-01 GB GB3396874A patent/GB1473733A/en not_active Expired
- 1974-08-01 FI FI2304/74A patent/FI62100C/sv active
- 1974-08-01 IE IE1638/74A patent/IE40437B1/en not_active IP Right Cessation
- 1974-08-01 DE DE2462485A patent/DE2462485C2/de not_active Expired
- 1974-08-02 IL IL45385A patent/IL45385A/xx unknown
- 1974-08-02 BE BE147234A patent/BE818431A/xx not_active IP Right Cessation
- 1974-08-02 LU LU70661A patent/LU70661A1/xx unknown
- 1974-08-05 DD DD180344A patent/DD119037A5/xx unknown
- 1974-08-06 BG BG027440A patent/BG25804A3/xx unknown
1979
- 1979-07-09 KE KE2981A patent/KE2981A/xx unknown
- 1979-08-09 HK HK551/79A patent/HK55179A/xx unknown
1980
- 1980-12-30 MY MY90/80A patent/MY8000090A/xx unknown

Also Published As

Publication number	Publication date
SE424994B (sv)	1982-08-23
DK146298C (da)	1984-02-06
NL171587C (nl)	1983-04-18
FI62100C (fi)	1982-11-10
DE2437160C3 (de)	1979-08-30
NO139483C (no)	1979-03-21
NO139483B (no)	1978-12-11
IL45385A (en)	1978-10-31
AU7194274A (en)	1976-02-05
DE2462485A1 (de)	1977-04-21
IE40437L (en)	1975-02-06
BE818431A (fr)	1975-02-03
CH606076A5 (de)	1978-10-13
FR2240015B1 (de)	1978-08-18
LU70661A1 (de)	1975-05-21
FR2240015A1 (de)	1975-03-07
NO742787L (de)	1975-03-03
BG25804A3 (en)	1978-12-12
DD119037A5 (de)	1976-04-05
DE2437160B2 (de)	1979-01-04
FI230474A (de)	1975-02-07
DE2437160A1 (de)	1975-02-20
IL45385A0 (en)	1974-11-29
DK146298B (da)	1983-08-29
AR215834A1 (es)	1979-11-15
HK55179A (en)	1979-08-17
DK412474A (de)	1975-04-01
DE2462485C2 (de)	1987-04-09
MY8000090A (en)	1980-12-31
KE2981A (en)	1979-07-20
GB1473733A (en)	1977-05-18
IE40437B1 (en)	1979-06-06
NL7410363A (nl)	1975-02-10
FI62100B (fi)	1982-07-30
NL171587B (nl)	1982-11-16
CY1018A (en)	1979-11-23

Legal Events

Date

Code

Title

Description

1995-01-31

NUG

Patent has lapsed

Ref document number: 7409946-6

Effective date: 19940910

Format of ref document f/p: F

Publication	Publication Date	Title
SE7409946L (de)	1975-02-07
AU529263B2 (en)	1983-06-02	Pyrid(1,2,3-de)(1,4)benzoxazine derivatives
MY111077A (en)	1999-08-30	Agricultural chemical composition
RU95122661A (ru)	1998-03-10	Производные 1-n-этилгентамицина и способы их получения
BR8801690A (pt)	1988-11-16	Processo para preparar(2,2)-paraciclofano e seus derivados
MX7096E (es)	1987-06-19	Metodo para preparacion de derivados de 2-oxoazetidina
KR860008210A (ko)	1986-11-14	글리코펩타이드 유도체의 제조 방법
KR850002971A (ko)	1985-05-28	시클로헥세논 유도체의 제조방법
ES428892A1 (es)	1977-02-16	Procedimiento para la preparacion de nuevos pseudotrisacari-dos.
MX165561B (es)	1992-11-23	Control de microorganismos en sistemas acuosos con 1-hidroximetilpirazoles
DE68927554D1 (de)	1997-01-30	Cephalosporinverbindungen und Verfahren zu ihrer Herstellung
ES468658A1 (es)	1979-09-16	Un procedimiento para preparar 4-alcohiltio-2-trifluorome- tilalcanosulfonanilidas y sus derivados
CA2135850A1 (en)	1995-05-16	Esculetin Derivatives, and Method for Manufacture Thereof, Use Thereof, and Pharmaceutical Composition
IE35379L (en)	1971-10-13	Erythromycylamine compounds
SE8004621L (sv)	1980-12-26	Bensimidazolderivat
ES433990A1 (es)	1977-03-01	Procedimiento para la preparacion de derivados de diaminoci-clitoles.
US3681496A (en)	1972-08-01	Bacteriostat and fungistat compositions containing n,s-heterocyclic compounds
ES449457A1 (es)	1977-08-16	Procedimiento para la preparacion de nuevos pseudotrisacari-dos.
KR850007428A (ko)	1985-12-04	세파로스포린 화합물의 제조방법
EP0144441A4 (de)	1986-12-01	Blutdruck regulierendes agenz.
GB1003645A (en)	1965-09-08	Indolo-indolizine compounds
ES8303327A1 (es)	1983-02-01	Un metodo para preparar derivados de 1-sulfo-2-oxoazetidina .
DE68911095D1 (de)	1994-01-13	Antitumor-Substanz, Verfahren zu deren Herstellung und diese enthaltende Antikrebsmittel.
KR830010120A (ko)	1983-12-26	세펨 화합물의 제조방법
GEP19981036B (en)	1998-10-27	Manufacturing method of aminothioazolyl derivatives of cephalosporin and of sodium and potassium salts thereof