PT84561B - Processo aperfeicoado para a preparacao de derivados macrolidos - Google Patents

Processo aperfeicoado para a preparacao de derivados macrolidos

Info

Publication number
PT84561B
PT84561B PT84561A PT8456187A PT84561B PT 84561 B PT84561 B PT 84561B PT 84561 A PT84561 A PT 84561A PT 8456187 A PT8456187 A PT 8456187A PT 84561 B PT84561 B PT 84561B
Authority
PT
Portugal
Prior art keywords
macrolidary
derivatives
preparation
appropriate process
appropriate
Prior art date
Application number
PT84561A
Other languages
English (en)
Other versions
PT84561A (en
Inventor
Eddie Vi-Ping Tao
Jeffrey Thomas Vicenzi
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT84561A publication Critical patent/PT84561A/pt
Publication of PT84561B publication Critical patent/PT84561B/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H5/00—Compounds containing saccharide radicals in which the hetero bonds to oxygen have been replaced by the same number of hetero bonds to halogen, nitrogen, sulfur, selenium, or tellurium
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
PT84561A 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos PT84561B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/846,446 US4921947A (en) 1986-03-31 1986-03-31 Process for preparing macrolide derivatives

Publications (2)

Publication Number Publication Date
PT84561A PT84561A (en) 1987-04-01
PT84561B true PT84561B (pt) 1989-11-10

Family

ID=25297965

Family Applications (1)

Application Number Title Priority Date Filing Date
PT84561A PT84561B (pt) 1986-03-31 1987-03-26 Processo aperfeicoado para a preparacao de derivados macrolidos

Country Status (21)

Country Link
US (1) US4921947A (pt)
EP (1) EP0240264B1 (pt)
JP (1) JPH0710876B2 (pt)
KR (1) KR900001166B1 (pt)
CN (1) CN1018647B (pt)
AR (1) AR247402A1 (pt)
AT (1) ATE66678T1 (pt)
AU (1) AU593894B2 (pt)
CA (1) CA1292737C (pt)
DE (1) DE3772423D1 (pt)
DK (1) DK172935B1 (pt)
EG (1) EG18550A (pt)
ES (1) ES2028865T3 (pt)
GR (1) GR3002764T3 (pt)
HK (1) HK82492A (pt)
HU (1) HU199864B (pt)
IE (1) IE61018B1 (pt)
IL (1) IL82005A (pt)
NZ (1) NZ219784A (pt)
PT (1) PT84561B (pt)
ZA (1) ZA872201B (pt)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2638458A1 (fr) * 1988-10-27 1990-05-04 Adir Nouveaux derives de la tylosine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
US5354708A (en) * 1992-06-04 1994-10-11 Taskar Nikhil R Method of nitrogen doping of II-VI semiconductor compounds during epitaxial growth using an amine
TW226373B (pt) * 1992-07-15 1994-07-11 Pfizer
US5677287A (en) * 1993-03-18 1997-10-14 Pfizer Inc. Antibacterial 16-membered ring macrolides containing olefins at C-20
WO1995002594A1 (en) * 1993-07-15 1995-01-26 Pfizer Inc. Amide derivatives of 16-membered ring antibiotic macrolides
ES2076107B1 (es) * 1993-09-20 1996-04-01 Pfizer Derivados de antibioticos macrolidos de anillos de 16 miembros.
EP0778283A3 (en) * 1995-12-05 1998-01-28 Pfizer Inc. Antibiotic macrolides
DE102004027417A1 (de) * 2004-06-04 2005-12-22 Basf Ag Verbundelement
EA019504B1 (ru) 2005-12-13 2014-04-30 Инсайт Корпорейшн ГЕТЕРОАРИЛЗАМЕЩЕННЫЕ ПИРРОЛО[2,3-b]ПИРИДИНЫ И ПИРРОЛО[2,3-b]ПИРИМИДИНЫ В КАЧЕСТВЕ ИНГИБИТОРОВ ЯНУС-КИНАЗЫ
CN103193840A (zh) * 2006-05-01 2013-07-10 大正制药株式会社 大环内酯衍生物
CN102875622B (zh) * 2006-07-28 2016-12-07 英特威国际有限公司 大环内酯合成方法
EP2019112A1 (en) * 2007-07-26 2009-01-28 Intervet International BV Macrolide solid-state forms
KR101538599B1 (ko) * 2006-07-28 2015-07-21 인터벳 인터내셔널 비.브이. 마크롤라이드 합성 방법
WO2012068440A1 (en) 2010-11-19 2012-05-24 Incyte Corporation Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
JP5917545B2 (ja) 2010-11-19 2016-05-18 インサイト・ホールディングス・コーポレイションＩｎｃｙｔｅ Ｈｏｌｄｉｎｇｓ Ｃｏｒｐｏｒａｔｉｏｎ Ｊａｋ阻害剤としてのシクロブチル置換ピロロピリジンおよびピロロピリミジン誘導体
US8691807B2 (en) 2011-06-20 2014-04-08 Incyte Corporation Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
BR112014012585B1 (pt) 2011-11-25 2021-05-25 Bayer Intellectual Property Gmbh composto compreendendo derivados de tilosina, método de preparo do mesmo e composição farmacêutica ou veterinária
CN102382159B (zh) * 2011-12-07 2013-11-13 齐鲁动物保健品有限公司 一种替米考星的制备方法
KR102366356B1 (ko) 2013-03-06 2022-02-23 인사이트 홀딩스 코포레이션 Jak 저해제를 제조하기 위한 방법 및 중간생성물
BR112015029260A2 (pt) * 2013-05-23 2017-07-25 Bayer Animal Health Gmbh derivados de tilosina e seu método de preparação
CN105837648B (zh) * 2015-11-02 2018-07-06 湖北龙翔药业科技股份有限公司 一种磷酸替米考星的制备方法
CN108299531B (zh) * 2018-01-23 2021-02-05 郑州大学 甲哌泰万菌素可药用盐及其制备方法
CN111269275A (zh) * 2020-03-09 2020-06-12 浙江康牧药业有限公司 一种替米考星的制备方法
CN117304241B (zh) * 2023-11-30 2024-03-01 中国农业科学院饲料研究所 一种大环内酯类化合物及其制备方法与应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU43006B (en) * 1981-03-06 1989-02-28 Pliva Pharm & Chem Works Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
JPS58146595A (ja) * 1982-02-25 1983-09-01 Satoshi Omura マクロライド系抗生物質
US4454314A (en) * 1982-08-02 1984-06-12 Pfizer Inc. Antibacterial mycaminosyl tylonolide and related macrolide derivatives
IL69666A (en) * 1982-09-13 1987-10-20 Lilly Co Eli 20-amino-20-deoxo-5-o-mycaminosyl-23-o-mycinosyltylonolide derivatives,their preparation and veterinary antibiotic use
US4443436A (en) * 1982-09-13 1984-04-17 Eli Lilly And Company C-20-Modified macrolide derivatives of the macrolide antibiotics tylosin, desmycosin, macrocin, and lactenocin
US4468511A (en) * 1983-02-28 1984-08-28 Eli Lilly And Company C-20- And C-23-Modified macrolide derivatives

Also Published As

Publication number Publication date
CA1292737C (en) 1991-12-03
DK154087A (da) 1987-10-01
CN1018647B (zh) 1992-10-14
IE61018B1 (en) 1994-09-07
IL82005A0 (en) 1987-10-20
JPS62240681A (ja) 1987-10-21
HK82492A (en) 1992-10-30
IE870796L (en) 1987-09-30
KR870008906A (ko) 1987-10-21
US4921947A (en) 1990-05-01
DK154087D0 (da) 1987-03-26
AR247402A1 (es) 1994-12-29
EP0240264A2 (en) 1987-10-07
IL82005A (en) 1991-08-16
DK172935B1 (da) 1999-10-11
AU7067087A (en) 1987-10-08
HU199864B (en) 1990-03-28
PT84561A (en) 1987-04-01
ATE66678T1 (de) 1991-09-15
AU593894B2 (en) 1990-02-22
EP0240264B1 (en) 1991-08-28
ES2028865T3 (es) 1992-07-16
CN87102397A (zh) 1987-10-07
HUT43087A (en) 1987-09-28
ZA872201B (en) 1988-10-26
DE3772423D1 (de) 1991-10-02
EG18550A (en) 1993-10-30
GR3002764T3 (en) 1993-01-25
EP0240264A3 (en) 1987-11-19
KR900001166B1 (ko) 1990-02-27
NZ219784A (en) 1989-01-27
JPH0710876B2 (ja) 1995-02-08

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