NO20090738L - Tilveiebringelse av EP2 agonister, fremgangsmate for fremstilling derav, farmasoytiske sammensetninger inneholdende disse forbindelser og fremgangsmater for anvendelse av forbindelsene og sammensetningene for a senke intraokkulaert trykk og behandle glaukom - Google Patents
Tilveiebringelse av EP2 agonister, fremgangsmate for fremstilling derav, farmasoytiske sammensetninger inneholdende disse forbindelser og fremgangsmater for anvendelse av forbindelsene og sammensetningene for a senke intraokkulaert trykk og behandle glaukomInfo
- Publication number
- NO20090738L NO20090738L NO20090738A NO20090738A NO20090738L NO 20090738 L NO20090738 L NO 20090738L NO 20090738 A NO20090738 A NO 20090738A NO 20090738 A NO20090738 A NO 20090738A NO 20090738 L NO20090738 L NO 20090738L
- Authority
- NO
- Norway
- Prior art keywords
- compounds
- methods
- agonists
- preparation
- intraocular pressure
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 208000010412 Glaucoma Diseases 0.000 title abstract 2
- 239000000556 agonist Substances 0.000 title abstract 2
- 230000004410 intraocular pressure Effects 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C311/04—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US83390706P | 2006-07-28 | 2006-07-28 | |
| US94192307P | 2007-06-04 | 2007-06-04 | |
| PCT/IB2007/002044 WO2008015517A2 (en) | 2006-07-28 | 2007-07-16 | Ep2 agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20090738L true NO20090738L (no) | 2009-04-27 |
Family
ID=38896126
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20090738A NO20090738L (no) | 2006-07-28 | 2009-02-16 | Tilveiebringelse av EP2 agonister, fremgangsmate for fremstilling derav, farmasoytiske sammensetninger inneholdende disse forbindelser og fremgangsmater for anvendelse av forbindelsene og sammensetningene for a senke intraokkulaert trykk og behandle glaukom |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US7622475B2 (ja) |
| EP (1) | EP2059507B1 (ja) |
| JP (1) | JP4583500B2 (ja) |
| KR (1) | KR101088942B1 (ja) |
| AP (1) | AP2009004754A0 (ja) |
| AR (1) | AR062122A1 (ja) |
| AU (1) | AU2007280130B2 (ja) |
| BR (1) | BRPI0714683A2 (ja) |
| CA (1) | CA2659184C (ja) |
| CL (1) | CL2007002207A1 (ja) |
| CR (1) | CR10554A (ja) |
| EA (1) | EA200970067A1 (ja) |
| EC (1) | ECSP099071A (ja) |
| GT (1) | GT200700064A (ja) |
| HK (1) | HK1133876A1 (ja) |
| IL (1) | IL196355A0 (ja) |
| MA (1) | MA30604B1 (ja) |
| MX (1) | MX2009001062A (ja) |
| NO (1) | NO20090738L (ja) |
| NZ (1) | NZ573964A (ja) |
| PE (1) | PE20080408A1 (ja) |
| RS (1) | RS20090002A (ja) |
| TN (1) | TN2009000028A1 (ja) |
| TW (1) | TWI372757B (ja) |
| UY (1) | UY30511A1 (ja) |
| WO (1) | WO2008015517A2 (ja) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR201904655T4 (tr) * | 2008-03-12 | 2019-06-21 | Ube Industries | Piridilaminoasetik asit bileşiği. |
| EP2415763B1 (en) | 2009-03-30 | 2016-01-27 | Ube Industries, Ltd. | Pharmaceutical composition for treating or preventing glaucoma |
| WO2011030865A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | 置換ベンジル化合物 |
| CA2773997A1 (en) * | 2009-09-11 | 2011-03-17 | Ube Industries, Ltd. | Aniline compound |
| CA2773998A1 (en) * | 2009-09-11 | 2011-03-17 | Ube Industries, Ltd. | Substituted carbonyl compound |
| WO2011030872A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | スルホンアミド化合物 |
| WO2011030873A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | ベンジル化合物 |
| WO2011030871A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | Ｎ－置換ヘテロアリール化合物 |
| KR20120101722A (ko) * | 2009-12-25 | 2012-09-14 | 우베 고산 가부시키가이샤 | 아미노피리딘 화합물 |
| KR20140003395A (ko) * | 2010-08-17 | 2014-01-09 | 알러간, 인코포레이티드 | 각막 혼탁 치료용 ep2 또는 ep4 항진제들 |
| SG11201400555SA (en) | 2011-09-16 | 2014-04-28 | Fovea Pharmaceuticals | Aniline derivatives,their preparation and their therapeutic application |
| WO2013109991A1 (en) * | 2012-01-20 | 2013-07-25 | Acucela Inc. | Substituted heterocyclic compounds for disease treatment |
| CN104507906B (zh) | 2012-05-03 | 2017-04-12 | 塔科达有限责任公司 | 新的ep2受体激动剂 |
| US9339496B2 (en) | 2012-07-13 | 2016-05-17 | Santen Pharmaceutical Co., Ltd. | Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist |
| US9676720B2 (en) * | 2013-03-28 | 2017-06-13 | Ube Industries, Ltd. | Substituted biaryl compound |
| JP2017206445A (ja) * | 2014-09-26 | 2017-11-24 | 宇部興産株式会社 | 呼吸器疾患の治療及び／又は予防のための医薬組成物 |
| JP2017206443A (ja) * | 2014-09-26 | 2017-11-24 | 宇部興産株式会社 | 置換ビアリール化合物及び他の医薬の組み合わせ |
| AR105215A1 (es) * | 2015-07-01 | 2017-09-13 | Santen Pharmaceutical Co Ltd | Formulación de depósito que contiene ésteres de ácido cítrico |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4599353A (en) * | 1982-05-03 | 1986-07-08 | The Trustees Of Columbia University In The City Of New York | Use of eicosanoids and their derivatives for treatment of ocular hypertension and glaucoma |
| US5296504A (en) * | 1988-09-06 | 1994-03-22 | Kabi Pharmacia | Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension |
| UA59384C2 (uk) * | 1996-12-20 | 2003-09-15 | Пфайзер, Інк. | Похідні сульфонамідів та амідів як агоністи простагландину, фармацевтична композиція та способи лікування на їх основі |
| UA67754C2 (uk) * | 1997-10-10 | 2004-07-15 | Пфайзер, Інк. | Агоністи простагландину, фармацевтична композиція на їх основі (варіанти), спосіб нарощення та збереження кісткової маси у хребетних та спосіб лікування (варіанти) |
| EP1000619A3 (en) * | 1998-06-23 | 2002-07-24 | Pfizer Products Inc. | Method for treating glaucoma |
| IL139941A0 (en) | 1999-12-02 | 2002-02-10 | Pfizer Prod Inc | Use of prostaglandin agonists to treat erectile dysfunction or impotence |
| US20020115695A1 (en) * | 2000-11-07 | 2002-08-22 | Paralkar Vishwas M. | Combination therapies for the stimulation of bone growth |
| JP2005513030A (ja) | 2001-11-30 | 2005-05-12 | ファイザー・プロダクツ・インク | 医薬組成物及びｅｐ２受容体選択的アゴニストの投与方法 |
| KR20040077884A (ko) * | 2002-01-31 | 2004-09-07 | 화이자 프로덕츠 인코포레이티드 | （3-｛〔（4-3급-뷰틸-벤질）-（피리딘-3-설폰일）-아미노〕-메틸｝-페녹시）-아세트산의 대사산물 |
| KR20050105511A (ko) | 2003-03-04 | 2005-11-04 | 화이자 프로덕츠 인크. | 의학적 치료에서 ｅｐ2 선택적 수용체 효능제의 용도 |
| US20050203086A1 (en) * | 2004-03-04 | 2005-09-15 | Pfizer Inc. | Methods of treatment using an EP2 selective receptor agonist |
| US7915316B2 (en) * | 2005-08-22 | 2011-03-29 | Allergan, Inc | Sulfonamides |
| US7696235B2 (en) * | 2005-08-29 | 2010-04-13 | Allergan, Inc. | EP2 receptor agonists for treating glaucoma |
-
2007
- 2007-07-16 BR BRPI0714683-3A patent/BRPI0714683A2/pt not_active IP Right Cessation
- 2007-07-16 KR KR1020097001522A patent/KR101088942B1/ko not_active IP Right Cessation
- 2007-07-16 MX MX2009001062A patent/MX2009001062A/es active IP Right Grant
- 2007-07-16 JP JP2009522350A patent/JP4583500B2/ja not_active Expired - Fee Related
- 2007-07-16 WO PCT/IB2007/002044 patent/WO2008015517A2/en active Application Filing
- 2007-07-16 RS RSP-2009/0002A patent/RS20090002A/sr unknown
- 2007-07-16 EP EP07766635A patent/EP2059507B1/en not_active Not-in-force
- 2007-07-16 AU AU2007280130A patent/AU2007280130B2/en not_active Ceased
- 2007-07-16 CA CA2659184A patent/CA2659184C/en not_active Expired - Fee Related
- 2007-07-16 AP AP2009004754A patent/AP2009004754A0/xx unknown
- 2007-07-16 EA EA200970067A patent/EA200970067A1/ru unknown
- 2007-07-16 NZ NZ573964A patent/NZ573964A/en not_active IP Right Cessation
- 2007-07-26 PE PE2007000967A patent/PE20080408A1/es not_active Application Discontinuation
- 2007-07-26 AR ARP070103330A patent/AR062122A1/es unknown
- 2007-07-27 UY UY30511A patent/UY30511A1/es not_active Application Discontinuation
- 2007-07-27 CL CL200702207A patent/CL2007002207A1/es unknown
- 2007-07-27 US US11/829,176 patent/US7622475B2/en not_active Expired - Fee Related
- 2007-07-27 TW TW096127590A patent/TWI372757B/zh not_active IP Right Cessation
- 2007-07-27 GT GT200700064A patent/GT200700064A/es unknown
-
2009
- 2009-01-05 IL IL196355A patent/IL196355A0/en unknown
- 2009-01-13 CR CR10554A patent/CR10554A/es not_active Application Discontinuation
- 2009-01-14 EC EC2009009071A patent/ECSP099071A/es unknown
- 2009-01-26 TN TN2009000028A patent/TN2009000028A1/fr unknown
- 2009-01-28 MA MA31593A patent/MA30604B1/fr unknown
- 2009-02-16 NO NO20090738A patent/NO20090738L/no not_active Application Discontinuation
- 2009-10-07 US US12/575,373 patent/US20100105905A1/en not_active Abandoned
- 2009-11-10 HK HK09110479.0A patent/HK1133876A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20090738L (no) | Tilveiebringelse av EP2 agonister, fremgangsmate for fremstilling derav, farmasoytiske sammensetninger inneholdende disse forbindelser og fremgangsmater for anvendelse av forbindelsene og sammensetningene for a senke intraokkulaert trykk og behandle glaukom | |
| PL1899329T3 (pl) | Pirymidyno-podstawione pochodne benzimidazolu jako inhibitory kinaz białkowych | |
| UA103319C2 (en) | Thiazole- and oxazole-benzene sulfonamide compounds | |
| NO20090295L (no) | Substituerte heteroarylderivater | |
| NO20092711L (no) | Metoder for anvendelse av cyclopaminanaloger | |
| NO20092138L (no) | Forbindelser og sammensetninger som proteinkinase inhibitorer | |
| NO20080675L (no) | P38-Map kinaseinhibitorer og metoder for deres anvendelse | |
| MX2009000884A (es) | Derivados de piridizinona. | |
| NO20084850L (no) | MGLUR5 modulatorer I | |
| EA200971051A1 (ru) | Ингибиторы p70 s6 киназы | |
| WO2008051942A3 (en) | Farnesoid x receptor agonists | |
| NO20093009L (no) | Kondensert ring heterocykel kinase modulatorer | |
| EA200900135A1 (ru) | Производные пиразола в качестве ингибиторов цитохрома р450 | |
| ATE526318T1 (de) | Farnesoid-x-rezeptor-agonisten | |
| WO2008131000A3 (en) | 7-substituted indole mcl-1 inhibitors | |
| WO2008017932A3 (en) | Heterocycles useful as inhibitors of carbonic anhydrase | |
| NO20081554L (no) | Isoindollmidforbindelser og sammensetninger omfattende samme, og anvendelse derav | |
| NO20083923L (no) | Pyrazolkinoloner er potente parp-inhibitorer | |
| NO20081160L (no) | Benzimidazoltiofen forbindelser | |
| NO341679B1 (no) | Substituerte pyridylamidforbindelser, fremstilling av slike og farmasøytiske sammensetninger inneholdende slike, samt anvendelse som modulatorer av histamin H3-reseptoren | |
| NI200900052A (es) | Heterocíclicos derivados de los inhibidores de metaloproteasa | |
| GB2466912A (en) | Compositions and methods for treating lysosomal disorders | |
| NO20064344L (no) | Caspaseinhibitorer og anvendelser derav | |
| TN2011000207A1 (en) | Akt and p70 s6 kinase inhibitors | |
| CL2007000595A1 (es) | Compuestos derivados de piperidina; composicion farmaceutica y uso para el tratamiento y/o profilaxis de enfermedades seleccionadas entre hipertension, insuficiencia cardiaca congestiva e insuficiencia renal entre otras. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |