HK1069382A1 - A process for preparing a phenylalanine derivative and intermediates thereof - Google Patents

A process for preparing a phenylalanine derivative and intermediates thereof

Info

Publication number
HK1069382A1
HK1069382A1 HK05102898.4A HK05102898A HK1069382A1 HK 1069382 A1 HK1069382 A1 HK 1069382A1 HK 05102898 A HK05102898 A HK 05102898A HK 1069382 A1 HK1069382 A1 HK 1069382A1
Authority
HK
Hong Kong
Prior art keywords
intermediates
preparing
phenylalanine derivative
phenylalanine
derivative
Prior art date
Application number
HK05102898.4A
Other languages
English (en)
Inventor
Isao Inoue
Toru Kuroda
Ryuzo Yoshioka
Original Assignee
Mitsubishi Tanabe Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Publication of HK1069382A1 publication Critical patent/HK1069382A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C233/00—Carboxylic acid amides
    • C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
    • C07C233/81—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
    • C07C233/82—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
    • C07C233/87—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom of a carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK05102898.4A 2002-02-28 2005-04-07 A process for preparing a phenylalanine derivative and intermediates thereof HK1069382A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2002052605 2002-02-28
PCT/JP2003/002181 WO2003072536A1 (en) 2002-02-28 2003-02-27 A process for preparing a phenylalanine derivative and intermediates thereof

Publications (1)

Publication Number Publication Date
HK1069382A1 true HK1069382A1 (en) 2005-05-20

Family

ID=27764341

Family Applications (1)

Application Number Title Priority Date Filing Date
HK05102898.4A HK1069382A1 (en) 2002-02-28 2005-04-07 A process for preparing a phenylalanine derivative and intermediates thereof

Country Status (22)

Country Link
US (1) US7476758B2 (xx)
EP (1) EP1478619B1 (xx)
KR (1) KR100681224B1 (xx)
CN (2) CN100480233C (xx)
AR (1) AR038624A1 (xx)
AT (1) ATE495147T1 (xx)
AU (1) AU2003208618B2 (xx)
BR (1) BR0308027A (xx)
CA (1) CA2476022C (xx)
DE (1) DE60335704D1 (xx)
ES (1) ES2359302T3 (xx)
HK (1) HK1069382A1 (xx)
IL (1) IL163429A (xx)
MX (1) MXPA04008359A (xx)
MY (1) MY140707A (xx)
NO (1) NO331001B1 (xx)
NZ (1) NZ534957A (xx)
PL (1) PL211046B1 (xx)
RU (1) RU2280641C2 (xx)
TW (1) TWI327996B (xx)
WO (1) WO2003072536A1 (xx)
ZA (1) ZA200406747B (xx)

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CR20210213A (es) 2018-10-30 2021-06-24 Gilead Sciences Inc Derivados de quinolina como inhibidores de la integrina alfa4beta7
WO2020092401A1 (en) 2018-10-30 2020-05-07 Gilead Sciences, Inc. COMPOUNDS FOR INHIBITION OF ALPHA 4β7 INTEGRIN
EP3873897B1 (en) 2018-10-30 2024-08-14 Gilead Sciences, Inc. N-benzoyl-phenylalanine derivatives as alpha4beta7 integrin inhibitors for treating inflammatory diseases
CN114222730B (zh) 2019-08-14 2024-09-10 吉利德科学公司 用于抑制α4β7整合素的化合物

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Also Published As

Publication number Publication date
MY140707A (en) 2010-01-15
IL163429A (en) 2012-07-31
BR0308027A (pt) 2004-12-28
CN1817853A (zh) 2006-08-16
RU2280641C2 (ru) 2006-07-27
AU2003208618A1 (en) 2003-09-09
TW200303854A (en) 2003-09-16
ES2359302T3 (es) 2011-05-20
PL371386A1 (en) 2005-06-13
WO2003072536A1 (en) 2003-09-04
KR20040091665A (ko) 2004-10-28
AU2003208618B2 (en) 2008-06-19
AR038624A1 (es) 2005-01-19
DE60335704D1 (de) 2011-02-24
EP1478619A1 (en) 2004-11-24
EP1478619B1 (en) 2011-01-12
NZ534957A (en) 2006-11-30
CA2476022C (en) 2008-07-15
NO20044087L (no) 2004-09-27
PL211046B1 (pl) 2012-04-30
US7476758B2 (en) 2009-01-13
CN1646482A (zh) 2005-07-27
TWI327996B (en) 2010-08-01
KR100681224B1 (ko) 2007-02-09
ZA200406747B (en) 2005-08-31
CA2476022A1 (en) 2003-09-04
MXPA04008359A (es) 2004-11-26
CN100522930C (zh) 2009-08-05
NO331001B1 (no) 2011-09-05
CN100480233C (zh) 2009-04-22
RU2004128935A (ru) 2006-02-20
US20050165107A1 (en) 2005-07-28
ATE495147T1 (de) 2011-01-15

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20150227