DK2498756T3 - Tabletformuleringer af neratinibmaleat - Google Patents

Tabletformuleringer af neratinibmaleat Download PDF

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Publication number
DK2498756T3
DK2498756T3 DK10779339T DK10779339T DK2498756T3 DK 2498756 T3 DK2498756 T3 DK 2498756T3 DK 10779339 T DK10779339 T DK 10779339T DK 10779339 T DK10779339 T DK 10779339T DK 2498756 T3 DK2498756 T3 DK 2498756T3
Authority
DK
Denmark
Prior art keywords
neratinibmaleate
tablet formulations
formulations
tablet
Prior art date
Application number
DK10779339T
Other languages
English (en)
Other versions
DK2498756T4 (da
Inventor
Muhammad Ashraf
Krishnendu Ghosh
Chimanlall Goolcharran
Mainuddin Mahmud
Arwinder Singh Nagi
Original Assignee
Wyeth Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43478191&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2498756(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wyeth Llc filed Critical Wyeth Llc
Publication of DK2498756T3 publication Critical patent/DK2498756T3/da
Application granted granted Critical
Publication of DK2498756T4 publication Critical patent/DK2498756T4/da

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4709Non-condensed quinolines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Plural Heterocyclic Compounds (AREA)
DK10779339.0T 2009-11-09 2010-11-02 Tabletformuleringer af neratinibmaleat DK2498756T4 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25940309P 2009-11-09 2009-11-09
PCT/IB2010/054964 WO2011055303A1 (en) 2009-11-09 2010-11-02 Tablet formulations of neratinib maleate

Publications (2)

Publication Number Publication Date
DK2498756T3 true DK2498756T3 (da) 2019-11-25
DK2498756T4 DK2498756T4 (da) 2023-03-20

Family

ID=43478191

Family Applications (1)

Application Number Title Priority Date Filing Date
DK10779339.0T DK2498756T4 (da) 2009-11-09 2010-11-02 Tabletformuleringer af neratinibmaleat

Country Status (21)

Country Link
US (2) US8518446B2 (da)
EP (3) EP2498756B2 (da)
JP (3) JP5835883B2 (da)
CN (2) CN102724970B (da)
AR (2) AR078952A1 (da)
AU (1) AU2010316683B2 (da)
CA (1) CA2780428C (da)
CY (1) CY1122330T1 (da)
DK (1) DK2498756T4 (da)
ES (1) ES2757882T5 (da)
FI (1) FI2498756T4 (da)
HR (1) HRP20192026T4 (da)
HU (1) HUE046606T2 (da)
LT (1) LT2498756T (da)
NZ (1) NZ599763A (da)
PL (1) PL2498756T5 (da)
PT (1) PT2498756T (da)
RS (1) RS59599B2 (da)
SI (1) SI2498756T2 (da)
TW (1) TWI466690B (da)
WO (1) WO2011055303A1 (da)

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Also Published As

Publication number Publication date
CN102724970A (zh) 2012-10-10
AR114143A2 (es) 2020-07-29
SI2498756T1 (sl) 2020-01-31
CN102724970B (zh) 2014-06-25
US8790708B2 (en) 2014-07-29
FI2498756T4 (fi) 2023-03-22
JP2011098964A (ja) 2011-05-19
CN103893140A (zh) 2014-07-02
SI2498756T2 (sl) 2023-04-28
AR078952A1 (es) 2011-12-14
AU2010316683B2 (en) 2015-10-08
JP5835883B2 (ja) 2015-12-24
US8518446B2 (en) 2013-08-27
CA2780428C (en) 2018-02-13
EP3566697B1 (en) 2024-09-11
JP2017075192A (ja) 2017-04-20
ES2757882T3 (es) 2020-04-30
EP2498756A1 (en) 2012-09-19
EP3566697A1 (en) 2019-11-13
CY1122330T1 (el) 2021-01-27
HRP20192026T4 (hr) 2023-03-31
TW201138774A (en) 2011-11-16
AU2010316683A1 (en) 2012-05-24
RS59599B2 (sr) 2023-03-31
DK2498756T4 (da) 2023-03-20
PL2498756T5 (pl) 2023-04-17
EP2498756B2 (en) 2023-02-15
WO2011055303A1 (en) 2011-05-12
CN103893140B (zh) 2016-06-01
ES2757882T5 (es) 2023-05-10
HRP20192026T1 (hr) 2020-02-07
LT2498756T (lt) 2019-12-10
PL2498756T3 (pl) 2020-03-31
TWI466690B (zh) 2015-01-01
HUE046606T2 (hu) 2020-03-30
CA2780428A1 (en) 2011-05-12
EP4066821A1 (en) 2022-10-05
US20110111018A1 (en) 2011-05-12
EP2498756B1 (en) 2019-09-04
NZ599763A (en) 2014-06-27
PT2498756T (pt) 2019-11-26
RS59599B1 (sr) 2020-01-31
JP2015091882A (ja) 2015-05-14
US20140004184A1 (en) 2014-01-02

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