DK148036C - Analogifremgangsmaade til fremstilling af epimere 4''-amino-erythromycin-forbindelser eller syreadditionssalte deraf - Google Patents

Analogifremgangsmaade til fremstilling af epimere 4''-amino-erythromycin-forbindelser eller syreadditionssalte deraf

Info

Publication number: DK148036C
Authority: DK; Denmark
Prior art keywords: epimere; analogue; amino; preparation; acid addition
Prior art date: 1977-02-04

Application number

DK51878A

Other languages

English (en)

Other versions

DK51878A (da

DK148036B (da

Inventor

Frank Christian Sciavolino

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-02-04

Filing date

1978-02-03

Publication date

1985-07-15

1977-12-01 Priority claimed from US05/856,479 external-priority patent/US4150220A/en

1978-02-03 Application filed by Pfizer filed Critical Pfizer

1978-08-05 Publication of DK51878A publication Critical patent/DK51878A/da

1985-02-11 Publication of DK148036B publication Critical patent/DK148036B/da

1985-07-15 Application granted granted Critical

1985-07-15 Publication of DK148036C publication Critical patent/DK148036C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK51878A 1977-02-04 1978-02-03 Analogifremgangsmaade til fremstilling af epimere 4''-amino-erythromycin-forbindelser eller syreadditionssalte deraf DK148036C (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US76548077A	1977-02-04	1977-02-04
US76548077		1977-02-04
US05/856,479 US4150220A (en)	1977-02-04	1977-12-01	Semi-synthetic 4"-erythromycin A derivatives
US85647977		1977-12-01

Publications (3)

Publication Number	Publication Date
DK51878A DK51878A (da)	1978-08-05
DK148036B DK148036B (da)	1985-02-11
DK148036C true DK148036C (da)	1985-07-15

Family

ID=27117613

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK51878A DK148036C (da)	1977-02-04	1978-02-03	Analogifremgangsmaade til fremstilling af epimere 4''-amino-erythromycin-forbindelser eller syreadditionssalte deraf

Country Status (30)

Country	Link
JP (1)	JPS5827798B2 (da)
AR (1)	AR222147A1 (da)
AU (1)	AU501298B1 (da)
BG (2)	BG33159A3 (da)
CA (1)	CA1106367A (da)
CH (1)	CH628906A5 (da)
CS (1)	CS221801B2 (da)
DD (1)	DD140048A5 (da)
DE (1)	DE2804507C2 (da)
DK (1)	DK148036C (da)
ES (2)	ES466057A1 (da)
FI (1)	FI780354A (da)
FR (2)	FR2379550A1 (da)
GB (2)	GB1585316A (da)
GR (1)	GR68691B (da)
HU (1)	HU182559B (da)
IE (1)	IE46661B1 (da)
IL (2)	IL53968A0 (da)
IT (1)	IT1094209B (da)
LU (1)	LU79004A1 (da)
NL (1)	NL176174C (da)
NO (2)	NO146472C (da)
NZ (1)	NZ186385A (da)
PH (2)	PH14421A (da)
PL (1)	PL116228B1 (da)
PT (1)	PT67568B (da)
RO (4)	RO79686A7 (da)
SE (2)	SE445223B (da)
SU (1)	SU927122A3 (da)
YU (3)	YU40913B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4124755A (en) *	1978-01-03	1978-11-07	Pfizer Inc.	11-Alkanoyl-4"-deoxy-4"-isonitrilo-oleandomycin derivatives
US4133950A (en) *	1978-01-03	1979-01-09	Pfizer Inc.	4"-Deoxy-4"-carbamate and dithiocarbamate derivatives of oleandomycin and its esters
US4382085A (en) *	1982-03-01	1983-05-03	Pfizer Inc.	4"-Epi erythromycin A and derivatives thereof as useful antibacterial agents
US4518590A (en) *	1984-04-13	1985-05-21	Pfizer Inc.	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
US6407074B1 (en)	1997-06-11	2002-06-18	Pfizer Inc	C-4″-substituted macrolide derivatives
HN1998000074A (es) *	1997-06-11	1999-01-08	Pfizer Prod Inc	Derivados de macrolidos c-4 sustituidos

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3836519A (en) *	1973-05-04	1974-09-17	Abbott Lab	Sulfonyl derivatives of erythromycin
US3884903A (en) *	1973-06-21	1975-05-20	Abbott Lab	4{41 -Deoxy-4{41 -oxoerythromycin B derivatives

1978
- 1978-01-10 SE SE7800270A patent/SE445223B/sv not_active IP Right Cessation
- 1978-01-13 PH PH20662A patent/PH14421A/en unknown
- 1978-01-17 ES ES466057A patent/ES466057A1/es not_active Expired
- 1978-01-18 AR AR270752A patent/AR222147A1/es active
- 1978-01-18 YU YU73/78A patent/YU40913B/xx unknown
- 1978-01-23 PT PT67568A patent/PT67568B/pt unknown
- 1978-01-31 CH CH106178A patent/CH628906A5/fr not_active IP Right Cessation
- 1978-02-02 GB GB34309/79A patent/GB1585316A/en not_active Expired
- 1978-02-02 CA CA296,037A patent/CA1106367A/en not_active Expired
- 1978-02-02 DE DE2804507A patent/DE2804507C2/de not_active Expired
- 1978-02-02 GB GB4165/78A patent/GB1585315A/en not_active Expired
- 1978-02-02 RO RO78101650A patent/RO79686A7/ro unknown
- 1978-02-02 RO RO78101651A patent/RO79687A7/ro unknown
- 1978-02-02 RO RO105255A patent/RO81622B/ro unknown
- 1978-02-02 CS CS78703A patent/CS221801B2/cs unknown
- 1978-02-02 RO RO7893080A patent/RO77345A/ro unknown
- 1978-02-02 GR GR55330A patent/GR68691B/el unknown
- 1978-02-03 AU AU32990/78A patent/AU501298B1/en not_active Expired
- 1978-02-03 DD DD78203547A patent/DD140048A5/de unknown
- 1978-02-03 SU SU782573754A patent/SU927122A3/ru active
- 1978-02-03 NL NLAANVRAGE7801262,A patent/NL176174C/xx not_active IP Right Cessation
- 1978-02-03 BG BG040069A patent/BG33159A3/xx unknown
- 1978-02-03 HU HU78PI611A patent/HU182559B/hu not_active IP Right Cessation
- 1978-02-03 JP JP53011352A patent/JPS5827798B2/ja not_active Expired
- 1978-02-03 LU LU79004A patent/LU79004A1/xx unknown
- 1978-02-03 PL PL1978204428A patent/PL116228B1/pl unknown
- 1978-02-03 IT IT20005/78A patent/IT1094209B/it active
- 1978-02-03 NO NO780389A patent/NO146472C/no unknown
- 1978-02-03 BG BG038579A patent/BG32718A3/xx unknown
- 1978-02-03 IL IL53968A patent/IL53968A0/xx not_active IP Right Cessation
- 1978-02-03 NZ NZ186385A patent/NZ186385A/xx unknown
- 1978-02-03 FI FI780354A patent/FI780354A/fi not_active Application Discontinuation
- 1978-02-03 FR FR7803066A patent/FR2379550A1/fr active Granted
- 1978-02-03 IE IE239/78A patent/IE46661B1/en not_active IP Right Cessation
- 1978-02-03 DK DK51878A patent/DK148036C/da not_active IP Right Cessation
- 1978-07-07 FR FR7820334A patent/FR2385735A1/fr active Granted
- 1978-08-08 ES ES472429A patent/ES472429A1/es not_active Expired
- 1978-09-01 PH PH21555A patent/PH16675A/en unknown
1981
- 1981-01-27 IL IL61997A patent/IL61997A0/xx unknown
- 1981-06-05 NO NO811913A patent/NO150484C/no unknown
1983
- 1983-02-07 YU YU265/83A patent/YU40798B/xx unknown
- 1983-02-16 SE SE8300870A patent/SE457086B/xx not_active IP Right Cessation
- 1983-11-21 YU YU2279/83A patent/YU40799B/xx unknown

Also Published As

Publication number	Publication date
YU40798B (en)	1986-06-30
RO81622A (ro)	1983-04-29
NO811913L (no)	1978-08-07
YU227983A (en)	1984-04-30
PL204428A1 (pl)	1979-06-04
IL61997A0 (en)	1981-02-27
DK51878A (da)	1978-08-05
IL53968A0 (en)	1978-04-30
DD140048A5 (de)	1980-02-06
NO150484C (no)	1984-10-24
FI780354A (fi)	1978-08-05
YU40913B (en)	1986-08-31
GB1585315A (en)	1981-02-25
RO79687A7 (ro)	1982-08-17
YU40799B (en)	1986-06-30
SE457086B (sv)	1988-11-28
NL7801262A (nl)	1978-08-08
BG33159A3 (en)	1982-12-15
PT67568B (en)	1979-06-18
ES466057A1 (es)	1978-10-01
SE8300870D0 (sv)	1983-02-16
RO79686A7 (ro)	1982-08-17
YU26583A (en)	1984-02-29
IE780239L (en)	1978-08-04
BG32718A3 (en)	1982-09-15
RO81622B (ro)	1983-04-30
CA1106367A (en)	1981-08-04
AU501298B1 (en)	1979-06-14
FR2379550A1 (fr)	1978-09-01
SE7800270L (sv)	1978-08-05
FR2379550B1 (da)	1980-07-04
NO150484B (no)	1984-07-16
IE46661B1 (en)	1983-08-24
NZ186385A (en)	1980-10-08
NL176174C (nl)	1985-03-01
PT67568A (en)	1978-02-01
NO146472B (no)	1982-06-28
SU927122A3 (ru)	1982-05-07
LU79004A1 (fr)	1979-09-06
ES472429A1 (es)	1979-04-01
PH16675A (en)	1983-12-13
GR68691B (da)	1982-02-01
HU182559B (en)	1984-02-28
SE8300870L (sv)	1983-02-16
GB1585316A (en)	1981-02-25
PL116228B1 (en)	1981-05-30
AR222147A1 (es)	1981-04-30
CS221801B2 (en)	1983-04-29
RO77345A (ro)	1981-08-17
FR2385735B1 (da)	1980-10-24
CH628906A5 (en)	1982-03-31
PH14421A (en)	1981-07-10
JPS53101337A (en)	1978-09-04
DE2804507A1 (de)	1978-08-10
IT1094209B (it)	1985-07-26
IT7820005A0 (it)	1978-02-03
YU7378A (en)	1983-04-30
SE445223B (sv)	1986-06-09
NL176174B (nl)	1984-10-01
DK148036B (da)	1985-02-11
FR2385735A1 (fr)	1978-10-27
NO780389L (no)	1978-08-07
DE2804507C2 (de)	1982-11-04
JPS5827798B2 (ja)	1983-06-11
NO146472C (no)	1982-10-06

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Legal Events

Date	Code	Title	Description
1994-10-24	PBP	Patent lapsed