DK1163250T3 - Forbedret syntese af [2.2.1]bicyclonukleosider - Google Patents

Forbedret syntese af [2.2.1]bicyclonukleosider

Info

Publication number
DK1163250T3
DK1163250T3 DK00912410T DK00912410T DK1163250T3 DK 1163250 T3 DK1163250 T3 DK 1163250T3 DK 00912410 T DK00912410 T DK 00912410T DK 00912410 T DK00912410 T DK 00912410T DK 1163250 T3 DK1163250 T3 DK 1163250T3
Authority
DK
Denmark
Prior art keywords
general formula
synthesis
instance
formula iii
bicyclo
Prior art date
Application number
DK00912410T
Other languages
English (en)
Inventor
Alexei Kochkine
Jef Fensholdt
Henrik M Pfundheller
Original Assignee
Exiqon As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Exiqon As filed Critical Exiqon As
Application granted granted Critical
Publication of DK1163250T3 publication Critical patent/DK1163250T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06Pyrimidine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16Purine radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK00912410T 1999-03-24 2000-03-24 Forbedret syntese af [2.2.1]bicyclonukleosider DK1163250T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DKPA199900407 1999-03-24
DKPA200000099 2000-01-21
EP00912410A EP1163250B1 (en) 1999-03-24 2000-03-24 Improved synthesis of ¬2.2.1|bicyclo nucleosides

Publications (1)

Publication Number Publication Date
DK1163250T3 true DK1163250T3 (da) 2006-11-13

Family

ID=26063935

Family Applications (1)

Application Number Title Priority Date Filing Date
DK00912410T DK1163250T3 (da) 1999-03-24 2000-03-24 Forbedret syntese af [2.2.1]bicyclonukleosider

Country Status (10)

Country Link
US (1) US6639059B1 (da)
EP (1) EP1163250B1 (da)
JP (1) JP4768132B2 (da)
AT (1) ATE332909T1 (da)
AU (1) AU3418800A (da)
DE (1) DE60029314T2 (da)
DK (1) DK1163250T3 (da)
ES (1) ES2269113T3 (da)
IL (1) IL145496A0 (da)
WO (1) WO2000056746A2 (da)

Families Citing this family (201)

* Cited by examiner, † Cited by third party
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