BR0210464A - Composto, composição farmacêutica, processo para preparar um composto, e, uso de um composto - Google Patents

Composto, composição farmacêutica, processo para preparar um composto, e, uso de um composto

Info

Publication number
BR0210464A
BR0210464A BR0210464-4A BR0210464A BR0210464A BR 0210464 A BR0210464 A BR 0210464A BR 0210464 A BR0210464 A BR 0210464A BR 0210464 A BR0210464 A BR 0210464A
Authority
BR
Brazil
Prior art keywords
compound
preparing
pharmaceutical composition
pharmaceutical
variables
Prior art date
Application number
BR0210464-4A
Other languages
English (en)
Inventor
Kristjan Gudmundsson
Brian A Johns
Original Assignee
Smithkline Beecham Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beecham Corp filed Critical Smithkline Beecham Corp
Publication of BR0210464A publication Critical patent/BR0210464A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A61P31/22—Antivirals for DNA viruses for herpes viruses

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"COMPOSTO, COMPOSIçãO FARMACêUTICA, PROCESSO PARA PREPARAR UM COMPOSTO, E, USO DE UM COMPOSTO". A presente invenção fornece compostos da fórmula (1) em que todas as variáveis são como definidas aqui, composições farmacêuticas contendo os mesmos, processos para preparar os mesmos e seu uso como agentes farmacêuticos.
BR0210464-4A 2001-06-21 2002-06-10 Composto, composição farmacêutica, processo para preparar um composto, e, uso de um composto BR0210464A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US30000901P 2001-06-21 2001-06-21
PCT/US2002/018520 WO2003000689A1 (en) 2001-06-21 2002-06-10 Imidazo`1,2-a!pyridine derivatives for the prophylaxis and treatment of herpes viral infections

Publications (1)

Publication Number Publication Date
BR0210464A true BR0210464A (pt) 2004-07-20

Family

ID=23157269

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0210464-4A BR0210464A (pt) 2001-06-21 2002-06-10 Composto, composição farmacêutica, processo para preparar um composto, e, uso de um composto

Country Status (19)

Country Link
US (3) US7186714B2 (pt)
EP (1) EP1401836B1 (pt)
JP (1) JP2005500315A (pt)
KR (1) KR20040018281A (pt)
CN (1) CN1518550A (pt)
AT (1) ATE337316T1 (pt)
BR (1) BR0210464A (pt)
CA (1) CA2451008A1 (pt)
CO (1) CO5540312A2 (pt)
CZ (1) CZ20033518A3 (pt)
DE (1) DE60214179T2 (pt)
ES (1) ES2271273T3 (pt)
HU (1) HUP0400266A2 (pt)
IL (1) IL158667A0 (pt)
MX (1) MXPA03011906A (pt)
NO (1) NO20035583D0 (pt)
PL (1) PL366827A1 (pt)
WO (1) WO2003000689A1 (pt)
ZA (1) ZA200308726B (pt)

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US20100249418A1 (en) * 2007-10-24 2010-09-30 Nihon Medi-Physics Co., Ltd. Novel compound having affinity for amyloid
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UA103319C2 (en) 2008-05-06 2013-10-10 Глаксосмитклайн Ллк Thiazole- and oxazole-benzene sulfonamide compounds
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WO2014195333A1 (de) * 2013-06-04 2014-12-11 Bayer Pharma Aktiengesellschaft 3-aryl-substituierte imidazo[1,2-a]pyridine und ihre verwendung
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US11071745B2 (en) * 2014-07-07 2021-07-27 Elian Llc Viral prophylaxis treatment methods and pre-exposure prophylaxis kits
CN107001361A (zh) 2014-12-02 2017-08-01 拜耳医药股份有限公司 杂芳基取代的咪唑并[1，2‑a]吡啶及其用途
SG11201907095UA (en) * 2017-02-01 2019-08-27 Aucentra Therapeutics Pty Ltd DERIVATIVES OF N-CYCLOALKYL/HETEROCYCLOALKYL-4-(IMIDAZO [1,2-a]PYRIDINE)PYRIMIDIN-2-AMINE AS THERAPEUTIC AGENTS
CN110483504B (zh) * 2019-08-02 2022-04-26 桂林理工大学 以DMF为甲酰化试剂构建2-(2-萘基)咪唑[1,2-a]吡啶-3-醛的新方法
CN110483506B (zh) * 2019-08-02 2022-04-19 桂林理工大学 以DMF为甲酰化试剂构建2-(2-噻吩基)咪唑[1,2-a]吡啶-3-醛的新方法

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Also Published As

Publication number Publication date
ES2271273T3 (es) 2007-04-16
CN1518550A (zh) 2004-08-04
DE60214179D1 (de) 2006-10-05
US7186714B2 (en) 2007-03-06
US20070135451A1 (en) 2007-06-14
EP1401836A1 (en) 2004-03-31
IL158667A0 (en) 2004-05-12
CZ20033518A3 (en) 2004-05-12
PL366827A1 (en) 2005-02-07
KR20040018281A (ko) 2004-03-02
CA2451008A1 (en) 2003-01-03
MXPA03011906A (es) 2004-03-26
HUP0400266A2 (hu) 2004-08-30
EP1401836B1 (en) 2006-08-23
JP2005500315A (ja) 2005-01-06
ZA200308726B (en) 2005-02-10
ATE337316T1 (de) 2006-09-15
NO20035583D0 (no) 2003-12-15
US20050228004A1 (en) 2005-10-13
CO5540312A2 (es) 2005-07-29
US20060167252A1 (en) 2006-07-27
DE60214179T2 (de) 2007-01-04
WO2003000689A1 (en) 2003-01-03

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Legal Events

Date Code Title Description
B11A Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]