NO317181B1 - Faste orale doseringsformer av valsartan - Google Patents

Faste orale doseringsformer av valsartan Download PDF

Info

Publication number: NO317181B1
Authority: NO; Norway
Prior art keywords: present; weight; solid oral; active agent; oral dosage
Prior art date: 1996-06-27

Application number

NO19986056A

Other languages

English (en)

Norwegian (no)

Other versions

NO986056L (no

NO986056D0 (no

Inventor

Robert Frank Wagner

Yoshimitsu Katakuse

Takashi Taike

Fujiki Yamato

Manfred Kohlmeyer

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-06-27

Filing date

1998-12-22

Publication date

2004-09-06

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10795969&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO317181(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1998-12-22 Application filed by Novartis Ag filed Critical Novartis Ag

1998-12-22 Publication of NO986056L publication Critical patent/NO986056L/no

1998-12-22 Publication of NO986056D0 publication Critical patent/NO986056D0/no

2004-09-06 Publication of NO317181B1 publication Critical patent/NO317181B1/no

Links

239000007787 solid Substances 0.000 title claims description 53
239000006186 oral dosage form Substances 0.000 title claims description 51
239000004072 C09CA03 - Valsartan Substances 0.000 title claims description 32
SJSNUMAYCRRIOM-QFIPXVFZSA-N valsartan Chemical compound C1=CC(CN(C(=O)CCCC)[C@@H](C(C)C)C(O)=O)=CC=C1C1=CC=CC=C1C1=NN=N[N]1 SJSNUMAYCRRIOM-QFIPXVFZSA-N 0.000 title claims description 32
229960004699 valsartan Drugs 0.000 title claims description 32
238000000034 method Methods 0.000 claims description 71
239000013543 active substance Substances 0.000 claims description 44
239000000654 additive Substances 0.000 claims description 33
239000000203 mixture Substances 0.000 claims description 25
JZUFKLXOESDKRF-UHFFFAOYSA-N Chlorothiazide Chemical compound C1=C(Cl)C(S(=O)(=O)N)=CC2=C1NCNS2(=O)=O JZUFKLXOESDKRF-UHFFFAOYSA-N 0.000 claims description 24
229960002003 hydrochlorothiazide Drugs 0.000 claims description 24
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WQZGKKKJIJFFOK-VFUOTHLCSA-N beta-D-glucose Chemical compound OC[C@H]1O[C@@H](O)[C@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-VFUOTHLCSA-N 0.000 claims description 2
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GXGAKHNRMVGRPK-UHFFFAOYSA-N dimagnesium;dioxido-bis[[oxido(oxo)silyl]oxy]silane Chemical compound [Mg+2].[Mg+2].[O-][Si](=O)O[Si]([O-])([O-])O[Si]([O-])=O GXGAKHNRMVGRPK-UHFFFAOYSA-N 0.000 claims description 2
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Classifications

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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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NO19986056A 1996-06-27 1998-12-22 Faste orale doseringsformer av valsartan NO317181B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GBGB9613470.5A GB9613470D0 (en)	1996-06-27	1996-06-27	Small solid oral dosage form
PCT/EP1997/003172 WO1997049394A2 (en)	1996-06-27	1997-06-18	Sold oral dosage forms of valsartan

Publications (3)

Publication Number	Publication Date
NO986056L NO986056L (no)	1998-12-22
NO986056D0 NO986056D0 (no)	1998-12-22
NO317181B1 true NO317181B1 (no)	2004-09-06

Family

ID=10795969

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
NO19986056A NO317181B1 (no)	1996-06-27	1998-12-22	Faste orale doseringsformer av valsartan
NO20041287A NO331739B1 (no)	1996-06-27	2004-03-26	Komprimerte, faste orale doseringsformer av valsartan og hydroklortiazid

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
NO20041287A NO331739B1 (no)	1996-06-27	2004-03-26	Komprimerte, faste orale doseringsformer av valsartan og hydroklortiazid

Country Status (33)

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US (3)	US6294197B1 (xx)
EP (7)	EP1774967A1 (xx)
JP (5)	JP2000506540A (xx)
KR (6)	KR20060079260A (xx)
CN (3)	CN1475207B (xx)
AR (2)	AR008618A1 (xx)
AT (3)	ATE446749T1 (xx)
BR (1)	BR9709956A (xx)
CA (2)	CA2259148C (xx)
CO (1)	CO4870755A1 (xx)
CY (1)	CY2553B1 (xx)
CZ (1)	CZ296850B6 (xx)
DE (3)	DE69738089T2 (xx)
DK (3)	DK1410797T3 (xx)
ES (3)	ES2335683T3 (xx)
GB (1)	GB9613470D0 (xx)
HK (2)	HK1019858A1 (xx)
HU (1)	HU229134B1 (xx)
ID (1)	ID17553A (xx)
IL (2)	IL127564A0 (xx)
MY (3)	MY156312A (xx)
NO (2)	NO317181B1 (xx)
NZ (2)	NZ333385A (xx)
PE (1)	PE87498A1 (xx)
PL (2)	PL188233B1 (xx)
PT (3)	PT1410797E (xx)
RU (5)	RU2203054C2 (xx)
SI (2)	SI1410797T1 (xx)
SK (1)	SK285902B6 (xx)
TR (1)	TR199802698T2 (xx)
TW (1)	TW473394B (xx)
WO (1)	WO1997049394A2 (xx)
ZA (1)	ZA975673B (xx)

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JP3534130B2 (ja) *	1994-03-01	2004-06-07	旭化成ケミカルズ株式会社	医薬品組成物
GB9404010D0 (en) *	1994-03-02	1994-04-20	Opt Tel Services Limited	Telephone dialling monitoring and route selecting apparatus
HUT76542A (en)	1994-03-17	1997-09-29	Ciba Geigy Ag	Use of valsartan for the preparation of pharmaceutical composition serving for the treatment of diabetic nephropathy
GB9408117D0 (en)	1994-04-23	1994-06-15	Smithkline Beecham Corp	Pharmaceutical formulations
DE19502065C2 (de) *	1995-01-14	1996-05-02	Prophyta Biolog Pflanzenschutz	Pilzisolat mit fungizider Wirkung
US5994348A (en) *	1995-06-07	1999-11-30	Sanofi	Pharmaceutical compositions containing irbesartan
FR2735365B1 (fr) *	1995-06-14	1997-09-05	Sanofi Sa	Utilisation d'un antagoniste de l'angiotensine ii et d'un derive du benzofurane pour la preparation d'un medicament utile dans le traitement des affections cardiovasculaires
GB9613470D0 (en) *	1996-06-27	1996-08-28	Ciba Geigy Ag	Small solid oral dosage form
JP2011123241A (ja) *	2009-12-10	2011-06-23	Canon Inc	撮影システム

1996
- 1996-06-27 GB GBGB9613470.5A patent/GB9613470D0/en active Pending
1997
- 1997-06-14 MY MYPI20093392A patent/MY156312A/en unknown
- 1997-06-14 MY MYPI20041863A patent/MY146868A/en unknown
- 1997-06-14 MY MYPI97002679A patent/MY123149A/en unknown
- 1997-06-18 CN CN031466788A patent/CN1475207B/zh not_active Expired - Lifetime
- 1997-06-18 EP EP06126829A patent/EP1774967A1/en not_active Withdrawn
- 1997-06-18 KR KR1020067011260A patent/KR20060079260A/ko not_active Application Discontinuation
- 1997-06-18 CN CNB971958912A patent/CN1133427C/zh not_active Expired - Lifetime
- 1997-06-18 KR KR1020097017936A patent/KR101161283B1/ko not_active IP Right Cessation
- 1997-06-18 IL IL12756497A patent/IL127564A0/xx unknown
- 1997-06-18 DK DK03027840T patent/DK1410797T3/da active
- 1997-06-18 DK DK06126819.9T patent/DK1767206T3/da active
- 1997-06-18 HU HU0203374A patent/HU229134B1/hu not_active IP Right Cessation
- 1997-06-18 SI SI9730773T patent/SI1410797T1/sl unknown
- 1997-06-18 DE DE69738089T patent/DE69738089T2/de not_active Expired - Lifetime
- 1997-06-18 SK SK1784-98A patent/SK285902B6/sk not_active IP Right Cessation
- 1997-06-18 SI SI9730686T patent/SI0914119T1/xx unknown
- 1997-06-18 ES ES06126819T patent/ES2335683T3/es not_active Expired - Lifetime
- 1997-06-18 PT PT03027840T patent/PT1410797E/pt unknown
- 1997-06-18 KR KR1020117011286A patent/KR101208430B1/ko not_active IP Right Cessation
- 1997-06-18 KR KR1020057015071A patent/KR100792389B1/ko not_active IP Right Cessation
- 1997-06-18 CA CA002259148A patent/CA2259148C/en not_active Expired - Fee Related
- 1997-06-18 PL PL97330709A patent/PL188233B1/pl not_active IP Right Cessation
- 1997-06-18 AT AT06126819T patent/ATE446749T1/de active
- 1997-06-18 CA CA2673462A patent/CA2673462C/en not_active Expired - Fee Related
- 1997-06-18 PL PL97363524A patent/PL188271B1/pl unknown
- 1997-06-18 AT AT97929209T patent/ATE276750T1/de active
- 1997-06-18 NZ NZ333385A patent/NZ333385A/xx not_active IP Right Cessation
- 1997-06-18 EP EP03027840A patent/EP1410797B1/en not_active Revoked
- 1997-06-18 BR BR9709956A patent/BR9709956A/pt not_active Application Discontinuation
- 1997-06-18 KR KR1020087000538A patent/KR20080014149A/ko active Search and Examination
- 1997-06-18 EP EP97929209A patent/EP0914119B1/en not_active Expired - Lifetime
- 1997-06-18 EP EP06126819A patent/EP1767206B1/en not_active Revoked
- 1997-06-18 JP JP10502269A patent/JP2000506540A/ja active Pending
- 1997-06-18 DE DE69730834T patent/DE69730834T2/de not_active Expired - Lifetime
- 1997-06-18 RU RU99101056/14A patent/RU2203054C2/ru active IP Right Maintenance
- 1997-06-18 KR KR1019980710521A patent/KR100618038B1/ko not_active IP Right Cessation
- 1997-06-18 EP EP06126834A patent/EP1776953A1/en not_active Withdrawn
- 1997-06-18 EP EP09001681A patent/EP2055301A1/en not_active Withdrawn
- 1997-06-18 WO PCT/EP1997/003172 patent/WO1997049394A2/en active Search and Examination
- 1997-06-18 DK DK97929209T patent/DK0914119T3/da active
- 1997-06-18 TR TR1998/02698T patent/TR199802698T2/xx unknown
- 1997-06-18 US US09/202,805 patent/US6294197B1/en not_active Expired - Lifetime
- 1997-06-18 PT PT97929209T patent/PT914119E/pt unknown
- 1997-06-18 ES ES97929209T patent/ES2231873T3/es not_active Expired - Lifetime
- 1997-06-18 PT PT06126819T patent/PT1767206E/pt unknown
- 1997-06-18 EP EP06126838A patent/EP1767207A3/en not_active Withdrawn
- 1997-06-18 ES ES03027840T patent/ES2290400T3/es not_active Expired - Lifetime
- 1997-06-18 RU RU99101056/63D patent/RU2294743C2/ru not_active IP Right Cessation
- 1997-06-18 CN CN2006100999105A patent/CN1951372B/zh not_active Expired - Lifetime
- 1997-06-18 AT AT03027840T patent/ATE371449T1/de active
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- 1997-06-18 CZ CZ0426998A patent/CZ296850B6/cs not_active IP Right Cessation
- 1997-06-23 CO CO97034775A patent/CO4870755A1/es unknown
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- 1997-06-25 AR ARP970102790A patent/AR008618A1/es active IP Right Grant
- 1997-06-26 ID IDP972207A patent/ID17553A/id unknown
- 1997-06-26 ZA ZA9705673A patent/ZA975673B/xx unknown
- 1997-09-09 TW TW086113018A patent/TW473394B/zh not_active IP Right Cessation
1998
- 1998-12-22 NO NO19986056A patent/NO317181B1/no not_active IP Right Cessation
1999
- 1999-11-09 HK HK99105148A patent/HK1019858A1/xx not_active IP Right Cessation
2001
- 2001-08-01 US US09/920,159 patent/US6485745B1/en not_active Expired - Fee Related
2002
- 2002-09-20 US US10/251,009 patent/US6858228B2/en not_active Expired - Fee Related
2003
- 2003-01-23 JP JP2003014987A patent/JP2003231634A/ja not_active Withdrawn
- 2003-02-21 NZ NZ524346A patent/NZ524346A/en not_active IP Right Cessation
2004
- 2004-03-26 NO NO20041287A patent/NO331739B1/no not_active IP Right Cessation
- 2004-05-25 HK HK04103718.1A patent/HK1060700A1/xx not_active IP Right Cessation
2006
- 2006-03-21 CY CY0600007A patent/CY2553B1/xx unknown
2007
- 2007-01-10 RU RU2007100200/15A patent/RU2453306C2/ru not_active IP Right Cessation
- 2007-02-06 AR ARP070100474A patent/AR059324A2/es not_active Application Discontinuation
- 2007-06-28 JP JP2007170267A patent/JP4969338B2/ja not_active Expired - Lifetime
2008
- 2008-11-17 IL IL195339A patent/IL195339A0/en unknown
2009
- 2009-04-27 RU RU2009115778/15A patent/RU2009115778A/ru unknown
2011
- 2011-12-09 JP JP2011270429A patent/JP2012051948A/ja not_active Withdrawn
2013
- 2013-03-26 RU RU2013113610/15A patent/RU2013113610A/ru not_active Application Discontinuation
- 2013-10-25 JP JP2013221985A patent/JP2014012747A/ja active Pending

Also Published As

Publication number	Publication date
EP2055301A1 (en)	2009-05-06
DK1767206T3 (da)	2010-01-25
HUP0203374A3 (en)	2004-06-28
SK285902B6 (sk)	2007-10-04
DE69730834T2 (de)	2005-10-06
EP1767207A2 (en)	2007-03-28
CA2259148A1 (en)	1997-12-31
DK0914119T3 (da)	2005-01-31
JP2012051948A (ja)	2012-03-15
EP1767206A2 (en)	2007-03-28
IL195339A0 (en)	2009-08-03
CN1951372B (zh)	2011-03-23
IL127564A0 (en)	1999-10-28
HK1019858A1 (en)	2000-06-09
DE69739642D1 (de)	2009-12-10
SK178498A3 (en)	1999-06-11
JP2000506540A (ja)	2000-05-30
ATE446749T1 (de)	2009-11-15
KR20110063587A (ko)	2011-06-10
ATE371449T1 (de)	2007-09-15
PL188233B1 (pl)	2004-12-31
HK1060700A1 (en)	2004-08-20
EP1410797B1 (en)	2007-08-29
TW473394B (en)	2002-01-21
KR20000022111A (ko)	2000-04-25
KR20090099020A (ko)	2009-09-18
EP0914119B1 (en)	2004-09-22
MY156312A (en)	2016-01-29
SI1410797T1 (sl)	2008-08-31
DE69738089T2 (de)	2008-05-21
KR100618038B1 (ko)	2006-11-30
PL188271B1 (pl)	2005-01-31
KR20060079260A (ko)	2006-07-05
CO4870755A1 (es)	1999-12-27
KR100792389B1 (ko)	2008-01-08
MY123149A (en)	2006-05-31
ATE276750T1 (de)	2004-10-15
PE87498A1 (es)	1998-12-21
KR20080014149A (ko)	2008-02-13
RU2203054C2 (ru)	2003-04-27
CZ296850B6 (cs)	2006-07-12
CN1475207B (zh)	2010-09-29
CZ426998A3 (cs)	1999-03-17
WO1997049394A3 (en)	2001-12-20
RU2013113610A (ru)	2014-10-10
EP1776953A1 (en)	2007-04-25
CY2553B1 (en)	2008-07-02
EP1410797A1 (en)	2004-04-21
MY146868A (en)	2012-09-28
US20030035832A1 (en)	2003-02-20
US6485745B1 (en)	2002-11-26
DE69738089D1 (de)	2007-10-11
CA2673462A1 (en)	1997-12-31
ID17553A (id)	1998-01-08
US6858228B2 (en)	2005-02-22
WO1997049394A2 (en)	1997-12-31
EP1767206B1 (en)	2009-10-28
EP1767206A3 (en)	2007-04-18
ES2335683T3 (es)	2010-03-31
KR20050092054A (ko)	2005-09-16
AU3340297A (en)	1998-01-14
GB9613470D0 (en)	1996-08-28
CN1232394A (zh)	1999-10-20
RU2453306C2 (ru)	2012-06-20
NO20041287L (no)	2004-03-26
NO986056L (no)	1998-12-22
EP1767207A3 (en)	2007-04-18
NZ524346A (en)	2004-09-24
RU2294743C2 (ru)	2007-03-10
NO331739B1 (no)	2012-03-12
JP2014012747A (ja)	2014-01-23
SI0914119T1 (en)	2005-04-30
CN1133427C (zh)	2004-01-07
PL330709A1 (en)	1999-05-24
JP2003231634A (ja)	2003-08-19
PT914119E (pt)	2005-02-28
KR101161283B1 (ko)	2012-07-02
EP1774967A1 (en)	2007-04-18
CN1951372A (zh)	2007-04-25
JP4969338B2 (ja)	2012-07-04
ES2290400T3 (es)	2008-02-16
KR101208430B1 (ko)	2012-12-05
JP2007238637A (ja)	2007-09-20
CN1475207A (zh)	2004-02-18
RU2009115778A (ru)	2010-11-10
US6294197B1 (en)	2001-09-25
DE69730834D1 (de)	2004-10-28
BR9709956A (pt)	1999-08-10
HUP0203374A2 (hu)	2004-05-28
AR008618A1 (es)	2000-02-09
PT1767206E (pt)	2010-01-27
AR059324A2 (es)	2008-03-26
ZA975673B (en)	1997-12-29
TR199802698T2 (xx)	1999-04-21
RU2007100200A (ru)	2008-07-20
ES2231873T3 (es)	2005-05-16
NO986056D0 (no)	1998-12-22
HU229134B1 (en)	2013-08-28
NZ333385A (en)	2000-09-29
CA2259148C (en)	2009-09-29
AU724998B2 (en)	2000-10-05
CA2673462C (en)	2011-10-04
EP0914119A3 (en)	2002-03-06
PT1410797E (pt)	2007-12-03
EP0914119A2 (en)	1999-05-12
DK1410797T3 (da)	2007-10-15

Legal Events

Date	Code	Title	Description
2015-01-26	MM1K	Lapsed by not paying the annual fees

Publication	Publication Date	Title
NO317181B1 (no)	2004-09-06	Faste orale doseringsformer av valsartan
RU2333757C2 (ru)	2008-09-20	Фармацевтические композиции
AU2001240092A1 (en)	2001-11-29	Sustained release ranolazine formulations
EP1263439A2 (en)	2002-12-11	Sustained release ranolazine formulations