DK171891B1 - Pyrrolylindolderivater, fremgangsmåde til fremstilling deraf, anvendelse deraf som terapeutisk virksomme substanser og som lægemidler samt lægemidler indeholdende de substituerede pyrrolindolderivater - Google Patents

Pyrrolylindolderivater, fremgangsmåde til fremstilling deraf, anvendelse deraf som terapeutisk virksomme substanser og som lægemidler samt lægemidler indeholdende de substituerede pyrrolindolderivater Download PDF

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Publication number
DK171891B1
DK171891B1 DK055889A DK55889A DK171891B1 DK 171891 B1 DK171891 B1 DK 171891B1 DK 055889 A DK055889 A DK 055889A DK 55889 A DK55889 A DK 55889A DK 171891 B1 DK171891 B1 DK 171891B1
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Prior art keywords
indolyl
methyl
dione
formula
pyrrole
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DK055889A
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Danish (da)
English (en)
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DK55889D0 (da
DK55889A (da
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Peter David Davis
Christopher Huw Hill
Geoffrey Lawton
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Hoffmann La Roche
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Priority claimed from GB888803048A external-priority patent/GB8803048D0/en
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK55889D0 publication Critical patent/DK55889D0/da
Publication of DK55889A publication Critical patent/DK55889A/da
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/044—Pyrrole radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Pyrrole Compounds (AREA)
DK055889A 1988-02-10 1989-02-07 Pyrrolylindolderivater, fremgangsmåde til fremstilling deraf, anvendelse deraf som terapeutisk virksomme substanser og som lægemidler samt lægemidler indeholdende de substituerede pyrrolindolderivater DK171891B1 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB8803048 1988-02-10
GB888803048A GB8803048D0 (en) 1988-02-10 1988-02-10 Substituted pyrroles
GB8827565 1988-11-25
GB888827565A GB8827565D0 (en) 1988-02-10 1988-11-25 Substituted pyrroles

Publications (3)

Publication Number Publication Date
DK55889D0 DK55889D0 (da) 1989-02-07
DK55889A DK55889A (da) 1989-08-11
DK171891B1 true DK171891B1 (da) 1997-08-04

Family

ID=26293462

Family Applications (1)

Application Number Title Priority Date Filing Date
DK055889A DK171891B1 (da) 1988-02-10 1989-02-07 Pyrrolylindolderivater, fremgangsmåde til fremstilling deraf, anvendelse deraf som terapeutisk virksomme substanser og som lægemidler samt lægemidler indeholdende de substituerede pyrrolindolderivater

Country Status (22)

Country Link
US (1) US5057614A (cs)
EP (1) EP0328026B1 (cs)
JP (1) JPH0730071B2 (cs)
AU (1) AU623630B2 (cs)
CA (1) CA1320194C (cs)
CZ (1) CZ280738B6 (cs)
DE (1) DE58904168D1 (cs)
DK (1) DK171891B1 (cs)
DZ (1) DZ1323A1 (cs)
ES (1) ES2054890T3 (cs)
FI (1) FI96861C (cs)
HU (1) HU201054B (cs)
IE (1) IE63489B1 (cs)
IL (1) IL89167A (cs)
IS (1) IS1941B (cs)
MC (1) MC2010A1 (cs)
NO (1) NO172540C (cs)
NZ (1) NZ227850A (cs)
PH (1) PH25185A (cs)
PT (1) PT89661B (cs)
SK (1) SK75289A3 (cs)
YU (1) YU47101B (cs)

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FI890652A0 (fi) 1989-02-10
EP0328026A1 (de) 1989-08-16
CA1320194C (en) 1993-07-13
PT89661A (pt) 1989-10-04
IE63489B1 (en) 1995-05-03
NO890568L (no) 1989-08-11
DZ1323A1 (fr) 2004-09-13
AU623630B2 (en) 1992-05-21
YU28489A (en) 1991-06-30
PH25185A (en) 1991-03-27
DE58904168D1 (de) 1993-06-03
HU201054B (en) 1990-09-28
DK55889D0 (da) 1989-02-07
IS3433A7 (is) 1989-08-11
DK55889A (da) 1989-08-11
FI890652A (fi) 1989-08-11
CZ280738B6 (cs) 1996-04-17
NO890568D0 (no) 1989-02-09
SK278989B6 (sk) 1998-05-06
ES2054890T3 (es) 1994-08-16
MC2010A1 (fr) 1990-02-16
SK75289A3 (en) 1998-05-06
JPH0730071B2 (ja) 1995-04-05
IE890416L (en) 1989-08-10
IL89167A (en) 1994-02-27
HUT49348A (en) 1989-09-28
US5057614A (en) 1991-10-15
JPH01233281A (ja) 1989-09-19
AU2965889A (en) 1989-08-10
IL89167A0 (en) 1989-09-10
FI96861C (fi) 1996-09-10
PT89661B (pt) 1994-02-28
NZ227850A (en) 1991-11-26
YU47101B (sh) 1994-12-28
EP0328026B1 (de) 1993-04-28
IS1941B (is) 2004-07-30
CZ75289A3 (en) 1995-12-13
NO172540B (no) 1993-04-26
NO172540C (no) 1993-08-04
FI96861B (fi) 1996-05-31

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