DD204257A5 - Verfahren zur herstellung von cephalosporinen, die in position 3 substituiert sind - Google Patents

Verfahren zur herstellung von cephalosporinen, die in position 3 substituiert sind Download PDF

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Publication number
DD204257A5
DD204257A5 DD82245454A DD24545482A DD204257A5 DD 204257 A5 DD204257 A5 DD 204257A5 DD 82245454 A DD82245454 A DD 82245454A DD 24545482 A DD24545482 A DD 24545482A DD 204257 A5 DD204257 A5 DD 204257A5
Authority
DD
German Democratic Republic
Prior art keywords
ppm
acid
reaction
group
formula
Prior art date
Application number
DD82245454A
Other languages
German (de)
English (en)
Inventor
Bernard Labeeuw
Ali Salhi
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of DD204257A5 publication Critical patent/DD204257A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36—Methylene radicals, substituted by sulfur atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Tunnel Furnaces (AREA)
  • Noodles (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
  • Polyesters Or Polycarbonates (AREA)
  • Peptides Or Proteins (AREA)
DD82245454A 1981-12-01 1982-12-01 Verfahren zur herstellung von cephalosporinen, die in position 3 substituiert sind DD204257A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8122506A FR2517309A1 (fr) 1981-12-01 1981-12-01 Nouveaux derives de cephalosporines substitues en position 3 par un groupe heterocycle thiomethyl; procede de preparation desdits composes et compositions pharmaceutiques en contenant

Publications (1)

Publication Number Publication Date
DD204257A5 true DD204257A5 (de) 1983-11-23

Family

ID=9264556

Family Applications (1)

Application Number Title Priority Date Filing Date
DD82245454A DD204257A5 (de) 1981-12-01 1982-12-01 Verfahren zur herstellung von cephalosporinen, die in position 3 substituiert sind

Country Status (30)

Country Link
US (1) US4609654A (es)
EP (1) EP0080944B1 (es)
JP (1) JPS58103392A (es)
KR (1) KR880001775B1 (es)
AT (1) ATE15199T1 (es)
AU (1) AU564235B2 (es)
CA (1) CA1189854A (es)
CS (1) CS232743B2 (es)
DD (1) DD204257A5 (es)
DE (1) DE3265901D1 (es)
DK (1) DK532282A (es)
EG (1) EG15644A (es)
ES (1) ES8308331A1 (es)
FI (1) FI73221C (es)
FR (1) FR2517309A1 (es)
GR (1) GR76739B (es)
HU (2) HU186999B (es)
IE (1) IE54173B1 (es)
IL (1) IL67285A (es)
MA (1) MA19659A1 (es)
NO (1) NO159857C (es)
NZ (1) NZ202658A (es)
OA (1) OA07262A (es)
PH (1) PH18949A (es)
PL (1) PL132054B1 (es)
PT (1) PT75905B (es)
SG (1) SG12188G (es)
SU (1) SU1114338A3 (es)
YU (1) YU265482A (es)
ZA (1) ZA828598B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS60142987A (ja) * 1983-12-29 1985-07-29 Mochida Pharmaceut Co Ltd セフアロスポリン誘導体
DE3485860T2 (de) * 1983-12-29 1993-01-14 Mochida Pharm Co Ltd Cephalosporinverbindungen, verfahren zu ihrer herstellung und pharmazeutishe praeparate.
US4840945A (en) * 1985-04-01 1989-06-20 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives
US4812562A (en) * 1985-07-25 1989-03-14 Taisho Pharmaceutical Co., Ltd. Cephalosporin derivatives
HU196814B (en) * 1985-10-22 1989-01-30 Biogal Gyogyszergyar Process for producing new cepheme-carboxylic acid derivatives
US4880798A (en) * 1986-11-25 1989-11-14 Mochida Pharmaceutical Co., Ltd. Cephalosporin derivatives
JPS63132893A (ja) * 1986-11-25 1988-06-04 Mochida Pharmaceut Co Ltd 新規セフアロスポリン誘導体、その製法およびそれらを有効成分とする抗菌剤

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB694060A (en) * 1949-12-27 1953-07-15 Bataafsche Petroleum Process for the manufacture of ethers of glycerols
US4165430A (en) * 1976-03-19 1979-08-21 Glaxo Laboratories Limited Cephalosporins having a 7-carboxy substituted α-etherified oximinoarylacetamido) group
DE2716677C2 (de) * 1977-04-15 1985-10-10 Hoechst Ag, 6230 Frankfurt Cephemderivate und Verfahren zu ihrer Herstellung
DK123480A (da) * 1979-03-22 1980-09-23 Glaxo Group Ltd Fremgangsmaade til fremstilling af cephalosporinforbindelser
US4237128A (en) * 1979-04-12 1980-12-02 E. R. Squibb & Sons, Inc. 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides

Also Published As

Publication number Publication date
SG12188G (en) 1989-01-27
AU564235B2 (en) 1987-08-06
GR76739B (es) 1984-08-30
YU265482A (en) 1985-03-20
FR2517309A1 (fr) 1983-06-03
US4609654A (en) 1986-09-02
ES517840A0 (es) 1983-08-16
EP0080944B1 (fr) 1985-08-28
IE54173B1 (en) 1989-07-05
PL132054B1 (en) 1985-01-31
KR840002406A (ko) 1984-07-21
ZA828598B (en) 1983-09-28
FI824043A0 (fi) 1982-11-24
FI73221B (fi) 1987-05-29
NO159857B (no) 1988-11-07
CS232743B2 (en) 1985-02-14
FI824043L (fi) 1983-06-02
HU186998B (en) 1985-10-28
EG15644A (en) 1986-09-30
CS859582A2 (en) 1984-02-13
DE3265901D1 (en) 1985-10-03
CA1189854A (en) 1985-07-02
FI73221C (fi) 1987-09-10
NZ202658A (en) 1985-07-12
PT75905A (fr) 1982-12-01
IL67285A (en) 1985-11-29
DK532282A (da) 1983-06-02
MA19659A1 (fr) 1983-07-01
PL239271A1 (en) 1983-06-06
IL67285A0 (en) 1983-03-31
AU9094882A (en) 1983-06-09
KR880001775B1 (ko) 1988-09-15
SU1114338A3 (ru) 1984-09-15
JPS58103392A (ja) 1983-06-20
NO823930L (no) 1983-06-02
ES8308331A1 (es) 1983-08-16
ATE15199T1 (de) 1985-09-15
NO159857C (no) 1989-02-15
FR2517309B1 (es) 1985-03-22
OA07262A (fr) 1984-04-30
EP0080944A1 (fr) 1983-06-08
PH18949A (en) 1985-11-14
PT75905B (fr) 1985-10-04
IE822721L (en) 1983-06-01
HU186999B (en) 1985-10-28

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