CA2652980A1 - Formulations d'oxymorphone robustes a liberation prolongee - Google Patents

Formulations d'oxymorphone robustes a liberation prolongee Download PDF

Info

Publication number: CA2652980A1
Authority: CA; Canada
Prior art keywords: formulation; oxymorphone; sustained release; ethanol; drug
Prior art date: 2006-10-10
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

CA002652980A

Other languages

English (en)

Inventor

Anand R. Baichwal

Kevin Fitzmaurice

Steve Labudzinski

Michelle Howard-Sparks

William Hein

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Penwest Pharmaceuticals Co

Original Assignee

Individual

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2006-10-10

Filing date

2006-10-10

Publication date

2008-04-17

2006-10-10 Application filed by Individual filed Critical Individual

2008-04-17 Publication of CA2652980A1 publication Critical patent/CA2652980A1/fr

Status Abandoned legal-status Critical Current

Links

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Chemical Kinetics & Catalysis (AREA)
Rheumatology (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

CA002652980A 2006-10-10 2006-10-10 Formulations d'oxymorphone robustes a liberation prolongee Abandoned CA2652980A1 (fr)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US2006/039767 WO2008045046A1 (fr)	2006-10-10	2006-10-10	Formulations d'oxymorphone robustes à libération prolongée

Publications (1)

Publication Number	Publication Date
CA2652980A1 true CA2652980A1 (fr)	2008-04-17

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ID=38169509

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CA002652980A Abandoned CA2652980A1 (fr)	2006-10-10	2006-10-10	Formulations d'oxymorphone robustes a liberation prolongee

Country Status (10)

Country	Link
EP (1)	EP2097069A1 (fr)
JP (1)	JP2010505947A (fr)
KR (1)	KR20090076946A (fr)
CN (1)	CN101578095A (fr)
AU (1)	AU2006349471A1 (fr)
BR (1)	BRPI0621952A2 (fr)
CA (1)	CA2652980A1 (fr)
IL (1)	IL198169A0 (fr)
MX (1)	MX2009003772A (fr)
WO (1)	WO2008045046A1 (fr)

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KR20030034171A (ko)	2001-07-06	2003-05-01	엔도 파마슈티걸즈, 인크.	옥시모르폰 제어 방출 제형
BRPI0621951A2 (pt) *	2006-10-10	2011-10-18	Penwest Pharmaceuticals Co	Formulações com liberação prolongada de oximorfona e formas de dosagem
EP3473246A1 (fr)	2017-10-19	2019-04-24	Capsugel Belgium NV	Formulations anti-abus à libération immédiate

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* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL208484B1 (pl) *	2001-07-06	2011-05-31	Penwest Pharmaceuticals Company	Sposoby wytwarzania preparatów oksymorfonu o przedłużonym uwalnianiu
KR20030034171A (ko) *	2001-07-06	2003-05-01	엔도 파마슈티걸즈, 인크.	옥시모르폰 제어 방출 제형
AU2002337686B2 (en) *	2001-09-26	2008-05-15	Penwest Pharmaceuticals Company	Opioid formulations having reduced potential for abuse
BRPI0621951A2 (pt) *	2006-10-10	2011-10-18	Penwest Pharmaceuticals Co	Formulações com liberação prolongada de oximorfona e formas de dosagem

2006
- 2006-10-10 CN CNA2006800560524A patent/CN101578095A/zh active Pending
- 2006-10-10 EP EP06816745A patent/EP2097069A1/fr not_active Withdrawn
- 2006-10-10 CA CA002652980A patent/CA2652980A1/fr not_active Abandoned
- 2006-10-10 BR BRPI0621952-7A patent/BRPI0621952A2/pt not_active Application Discontinuation
- 2006-10-10 KR KR1020097008716A patent/KR20090076946A/ko not_active Application Discontinuation
- 2006-10-10 WO PCT/US2006/039767 patent/WO2008045046A1/fr active Application Filing
- 2006-10-10 JP JP2009532329A patent/JP2010505947A/ja active Pending
- 2006-10-10 AU AU2006349471A patent/AU2006349471A1/en not_active Abandoned
- 2006-10-10 MX MX2009003772A patent/MX2009003772A/es not_active Application Discontinuation
2009
- 2009-04-16 IL IL198169A patent/IL198169A0/en unknown

Also Published As

Publication number	Publication date
JP2010505947A (ja)	2010-02-25
EP2097069A1 (fr)	2009-09-09
AU2006349471A1 (en)	2008-04-17
IL198169A0 (en)	2009-12-24
MX2009003772A (es)	2009-07-22
CN101578095A (zh)	2009-11-11
WO2008045046A1 (fr)	2008-04-17
KR20090076946A (ko)	2009-07-13
BRPI0621952A2 (pt)	2011-10-18

Legal Events

Date	Code	Title	Description
2008-02-26	EEER	Examination request
2015-03-29	FZDE	Discontinued	Effective date: 20150130

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