BR9810592A - Composto, processos para preparar um composto, para tratar ou prevenir doenças do sistema endócrino e para a fabricação de um medicamento, composição farmacêutica, e, uso de um composto - Google Patents

Composto, processos para preparar um composto, para tratar ou prevenir doenças do sistema endócrino e para a fabricação de um medicamento, composição farmacêutica, e, uso de um composto

Info

Publication number
BR9810592A
BR9810592A BR9810592-2A BR9810592A BR9810592A BR 9810592 A BR9810592 A BR 9810592A BR 9810592 A BR9810592 A BR 9810592A BR 9810592 A BR9810592 A BR 9810592A
Authority
BR
Brazil
Prior art keywords
compound
processes
preparing
manufacture
pharmaceutical composition
Prior art date
Application number
BR9810592-2A
Other languages
English (en)
Inventor
Fleming Elmedlund Nielsen
John Bondo Hansen
Holger Claus Hansen
Tina Mueller Tagmose
John Patrick Mogensen
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of BR9810592A publication Critical patent/BR9810592A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

"COMPOSTO, PROCESSOS PARA PREPARAR UM COMPOSTO, PARA TRATAR OU PREVENIR DOENçAS DO SISTEMA ENDóCRINO E PARA A FABRICAçãO DE UM MEDICAMENTO, COMPOSIçãO FARMACêUTICA, E, USO DE UM COMPOSTO". Os derivados de 1,2,4-tiadiazina e de 1,4-tiazina, representados pela fórmula (I): em que A, B, D, R , R , R e R^ 4^ são definidos na descrição, suas composições e processos para preparar os compostos são descritos. Os compostos são úteis no tratamento de doenças do sistema nervoso central, do sistema cardiovascular, do sistema pulmonar, do sistema gastrointestinal e do sistema endócrino.
BR9810592-2A 1997-07-16 1998-06-30 Composto, processos para preparar um composto, para tratar ou prevenir doenças do sistema endócrino e para a fabricação de um medicamento, composição farmacêutica, e, uso de um composto BR9810592A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DK87297 1997-07-16
DK36898 1998-03-17
PCT/DK1998/000288 WO1999003861A1 (en) 1997-07-16 1998-06-30 Fused 1,2,4-thiadiazine derivatives, their preparation and use

Publications (1)

Publication Number Publication Date
BR9810592A true BR9810592A (pt) 2000-09-12

Family

ID=26063863

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9810592-2A BR9810592A (pt) 1997-07-16 1998-06-30 Composto, processos para preparar um composto, para tratar ou prevenir doenças do sistema endócrino e para a fabricação de um medicamento, composição farmacêutica, e, uso de um composto

Country Status (13)

Country Link
EP (1) EP1000066A1 (pt)
JP (1) JP2001510195A (pt)
KR (1) KR20010021936A (pt)
CN (1) CN1264384A (pt)
AU (1) AU757693B2 (pt)
BR (1) BR9810592A (pt)
CA (1) CA2294830A1 (pt)
HU (1) HUP0003999A3 (pt)
IL (1) IL133604A0 (pt)
NO (1) NO315470B1 (pt)
PL (1) PL338013A1 (pt)
RU (1) RU2215004C2 (pt)
WO (1) WO1999003861A1 (pt)

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