BR112017017428A2 - ?método para supressão do amargor de derivado de quinolina? - Google Patents

?método para supressão do amargor de derivado de quinolina?

Info

Publication number
BR112017017428A2
BR112017017428A2 BR112017017428-6A BR112017017428A BR112017017428A2 BR 112017017428 A2 BR112017017428 A2 BR 112017017428A2 BR 112017017428 A BR112017017428 A BR 112017017428A BR 112017017428 A2 BR112017017428 A2 BR 112017017428A2
Authority
BR
Brazil
Prior art keywords
quot
bitterness
suppressing
quinoline derivative
quinoline
Prior art date
Application number
BR112017017428-6A
Other languages
English (en)
Japanese (ja)
Inventor
NAGANE Kentaro
Ueki Yosuke
SANO Shusuke
Sakaguchi Takahisa
Original Assignee
Eisai R&D Management Co., Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=56789022&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR112017017428(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Eisai R&D Management Co., Ltd. filed Critical Eisai R&D Management Co., Ltd.
Publication of BR112017017428A2 publication Critical patent/BR112017017428A2/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
    • A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Inorganic Chemistry (AREA)
  • Dispersion Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Zoology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)

Abstract

a presente invenção proporciona um método para supressão do amargor de um derivado de quinolina.
BR112017017428-6A 2015-02-25 2016-02-23 ?método para supressão do amargor de derivado de quinolina? BR112017017428A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201562120561P 2015-02-25 2015-02-25
US62/120.561 2015-02-25
PCT/JP2016/055268 WO2016136745A1 (ja) 2015-02-25 2016-02-23 キノリン誘導体の苦味抑制方法

Publications (1)

Publication Number Publication Date
BR112017017428A2 true BR112017017428A2 (pt) 2018-04-03

Family

ID=56789022

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112017017428-6A BR112017017428A2 (pt) 2015-02-25 2016-02-23 ?método para supressão do amargor de derivado de quinolina?

Country Status (23)

Country Link
US (2) US20180028662A1 (pt)
EP (1) EP3263106B1 (pt)
JP (1) JP6792546B2 (pt)
KR (1) KR20170122734A (pt)
CN (1) CN107427505A (pt)
AU (1) AU2016224583B2 (pt)
BR (1) BR112017017428A2 (pt)
CA (1) CA2976325C (pt)
DK (1) DK3263106T3 (pt)
ES (1) ES2967362T3 (pt)
FI (1) FI3263106T3 (pt)
HR (1) HRP20231692T1 (pt)
HU (1) HUE064614T2 (pt)
IL (1) IL253946A0 (pt)
LT (1) LT3263106T (pt)
MX (1) MX2017010474A (pt)
PL (1) PL3263106T3 (pt)
PT (1) PT3263106T (pt)
RS (1) RS65049B1 (pt)
RU (1) RU2017128583A (pt)
SG (1) SG11201706630UA (pt)
SI (1) SI3263106T1 (pt)
WO (1) WO2016136745A1 (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20200345637A1 (en) * 2018-01-19 2020-11-05 Aiviva Biopharma, Inc. Suspension compositions of multi-target inhibitors
CN112190583B (zh) * 2019-07-08 2021-10-29 成都苑东生物制药股份有限公司 一种乐伐替尼药物组合物及其制备方法
EP4153140A4 (en) * 2020-05-23 2024-07-17 Shilpa Medicare Ltd ORAL LIQUID FORMULATIONS OF LENVATINIB

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