BR0111206A - Derivados de arilmetilamina para uso como inibidores de triptase - Google Patents
Derivados de arilmetilamina para uso como inibidores de triptaseInfo
- Publication number
- BR0111206A BR0111206A BR0111206-6A BR0111206A BR0111206A BR 0111206 A BR0111206 A BR 0111206A BR 0111206 A BR0111206 A BR 0111206A BR 0111206 A BR0111206 A BR 0111206A
- Authority
- BR
- Brazil
- Prior art keywords
- tryptase inhibitors
- arylmethylamine
- derivatives
- arylmethylamine derivatives
- compounds
- Prior art date
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- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
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- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
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- Life Sciences & Earth Sciences (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
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- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
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- Pulmonology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Hospice & Palliative Care (AREA)
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Abstract
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0012362.0A GB0012362D0 (en) | 2000-05-22 | 2000-05-22 | Chemical compounds |
US09/843,126 US6977263B2 (en) | 2000-05-22 | 2001-04-26 | Chemical compounds |
PCT/US2001/013811 WO2001090101A1 (en) | 2000-05-22 | 2001-04-27 | Arylmethylamine derivatives for use as tryptase inhibitors |
Publications (1)
Publication Number | Publication Date |
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BR0111206A true BR0111206A (pt) | 2003-04-15 |
Family
ID=26244322
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0111206-6A BR0111206A (pt) | 2000-05-22 | 2001-04-27 | Derivados de arilmetilamina para uso como inibidores de triptase |
Country Status (19)
Country | Link |
---|---|
US (1) | US20050228018A1 (pt) |
EP (1) | EP1296972B1 (pt) |
KR (1) | KR100858642B1 (pt) |
CN (1) | CN1230431C (pt) |
AR (1) | AR033525A1 (pt) |
AU (2) | AU2001257413B2 (pt) |
BR (1) | BR0111206A (pt) |
CA (1) | CA2409827C (pt) |
DZ (1) | DZ3347A1 (pt) |
HK (1) | HK1057899A1 (pt) |
HR (1) | HRP20020926B1 (pt) |
HU (1) | HU227630B1 (pt) |
IL (1) | IL152830A0 (pt) |
MA (1) | MA25809A1 (pt) |
MX (1) | MXPA02011400A (pt) |
NO (1) | NO327378B1 (pt) |
OA (1) | OA12274A (pt) |
PL (1) | PL360495A1 (pt) |
WO (1) | WO2001090101A1 (pt) |
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SG11201504231PA (en) | 2012-11-30 | 2015-07-30 | Kyowa Hakko Kirin Co Ltd | Nitrogen-containing heterocyclic compound |
TW201441193A (zh) * | 2012-12-06 | 2014-11-01 | Kyowa Hakko Kirin Co Ltd | 吡啶酮化合物 |
KR20160110357A (ko) | 2013-11-15 | 2016-09-21 | 더 위스타 인스티튜트 오브 아나토미 앤드 바이올로지 | Ebna1 억제제 및 그의 사용 방법 |
EP3113619A4 (en) | 2014-03-06 | 2017-09-13 | PTC Therapeutics, Inc. | Pharmaceutical compositions and salts of a 1,2,4-oxadiazole benzoic acid |
AU2016262572B2 (en) | 2015-05-14 | 2020-04-30 | The Wistar Institute Of Anatomy And Biology | EBNA1 inhibitors and methods using same |
AU2016287584B2 (en) | 2015-07-02 | 2020-03-26 | Centrexion Therapeutics Corporation | (4-((3R,4R)-3-methoxytetrahydro-pyran-4-ylamino)piperidin-1-yl)(5-methyl-6-(((2R,6S)-6-(p-tolyl)tetrahydro-2H-pyran-2-yl)methylamino)pyrimidin-4yl)methanone citrate |
MX2018005361A (es) | 2015-10-30 | 2018-06-07 | Ptc Therapeutics Inc | Metodos para tratar epilepsia. |
US11242338B2 (en) | 2018-05-17 | 2022-02-08 | The Wistar Institute | EBNA1 inhibitor crystalline forms, and methods of preparing and using same |
CN110357833B (zh) * | 2019-06-03 | 2022-05-24 | 杭州维坦医药科技有限公司 | 芳杂乙酰胺类衍生物及其制备和应用 |
TW202115086A (zh) | 2019-06-28 | 2021-04-16 | 美商輝瑞大藥廠 | Bckdk抑制劑 |
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DE4407139A1 (de) * | 1994-03-04 | 1995-09-07 | Thomae Gmbh Dr K | Aryl-1-azacycloalkane und deren Salze, diese Verbindungen enthaltende Arzneimittel und deren Verwendung sowie Verfahren zu ihrer Herstellung |
US6673908B1 (en) * | 1999-02-22 | 2004-01-06 | Nuvelo, Inc. | Tumor necrosis factor receptor 2 |
-
2001
- 2001-04-27 EP EP01930925A patent/EP1296972B1/en not_active Expired - Lifetime
- 2001-04-27 AU AU2001257413A patent/AU2001257413B2/en not_active Ceased
- 2001-04-27 IL IL15283001A patent/IL152830A0/xx unknown
- 2001-04-27 AU AU5741301A patent/AU5741301A/xx active Pending
- 2001-04-27 KR KR1020027015683A patent/KR100858642B1/ko not_active IP Right Cessation
- 2001-04-27 BR BR0111206-6A patent/BR0111206A/pt not_active IP Right Cessation
- 2001-04-27 PL PL36049501A patent/PL360495A1/xx not_active Application Discontinuation
- 2001-04-27 MX MXPA02011400A patent/MXPA02011400A/es active IP Right Grant
- 2001-04-27 CA CA2409827A patent/CA2409827C/en not_active Expired - Lifetime
- 2001-04-27 HU HU0302485A patent/HU227630B1/hu not_active IP Right Cessation
- 2001-04-27 WO PCT/US2001/013811 patent/WO2001090101A1/en active IP Right Grant
- 2001-04-27 DZ DZ013347A patent/DZ3347A1/fr active
- 2001-04-27 AR ARP010102009A patent/AR033525A1/es active IP Right Grant
- 2001-04-27 CN CNB018119522A patent/CN1230431C/zh not_active Expired - Lifetime
- 2001-04-27 OA OA1200200357A patent/OA12274A/en unknown
-
2002
- 2002-11-21 NO NO20025601A patent/NO327378B1/no not_active IP Right Cessation
- 2002-11-21 MA MA26919A patent/MA25809A1/fr unknown
- 2002-11-21 HR HR20020926A patent/HRP20020926B1/xx not_active IP Right Cessation
-
2004
- 2004-02-06 HK HK04100765A patent/HK1057899A1/xx unknown
-
2005
- 2005-02-14 US US11/057,809 patent/US20050228018A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
EP1296972B1 (en) | 2009-12-23 |
HK1057899A1 (en) | 2004-04-23 |
CA2409827C (en) | 2010-06-01 |
HU227630B1 (hu) | 2011-10-28 |
CN1439003A (zh) | 2003-08-27 |
OA12274A (en) | 2006-05-09 |
AU5741301A (en) | 2001-12-03 |
AU2001257413B2 (en) | 2007-01-18 |
PL360495A1 (en) | 2004-09-06 |
KR100858642B1 (ko) | 2008-09-17 |
HUP0302485A2 (hu) | 2003-12-29 |
KR20030003294A (ko) | 2003-01-09 |
MXPA02011400A (es) | 2003-05-23 |
NO20025601L (no) | 2003-01-06 |
IL152830A0 (en) | 2003-06-24 |
WO2001090101A1 (en) | 2001-11-29 |
EP1296972A1 (en) | 2003-04-02 |
HUP0302485A3 (en) | 2007-09-28 |
MA25809A1 (fr) | 2003-07-01 |
NO20025601D0 (no) | 2002-11-21 |
CN1230431C (zh) | 2005-12-07 |
HRP20020926A2 (en) | 2005-02-28 |
US20050228018A1 (en) | 2005-10-13 |
DZ3347A1 (fr) | 2001-11-29 |
HRP20020926B1 (en) | 2011-01-31 |
NO327378B1 (no) | 2009-06-22 |
AR033525A1 (es) | 2003-12-26 |
CA2409827A1 (en) | 2001-11-29 |
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Free format text: PARA:INT.CI. A61K31/451; A61K31/4525; A61K31/453; A61K31/4535; A61K31/454; A61K31/4545; A61K31/4709; A61K31/473; A61K31/496; A61K31/501; A61K31/519; A61K31/5377; A61K45/00; A61P1/02; A61P1/16; A61P11/00; A61P17/00; A61P17/06; A61P19/06; A61P25/28; A61P27/02; A61P29/00; A61P29/02; A61P31/12; A61P35/00; A61P37/00; A61P37/08; A61P43/00; A61P9/10; C07D211/26; C07D211/32; C07D211/58; C07D401/06; C07D401/10; C07D401/12; C07D401/14; C07D405/06; C07D405/10; C07D405/12; C07D405/14; C07D409/06; C07D409/14; C07D411/06; C07D413/10; C07D413/12; C07D413/14; C07D417/06; C07D471/04; C07D487/04; C07D495/04; C07D513/04 Ipc: A61K 31/451 (2006.01), A61K 31/4525 (2006.01), A61 |
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