Eisenach, 1994 - Google Patents

Alpha-2 agonists and analgesia

Eisenach, 1994

Document ID
17365463031755241226
Author
Eisenach J
Publication year
Publication venue
Expert Opinion on Investigational Drugs

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In addition to their anti-hypertensive effects, alpha-2 agonists also cause analgesia. Since analgesia from these drugs is due primarily to actions in the spinal cord, it is not surprising that analgesia is poor after systemic administration, but profound after injection near the cord …
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
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