ZA201803942B - Novel processes for preparation of integrase inhibitor - Google Patents
Novel processes for preparation of integrase inhibitorInfo
- Publication number
- ZA201803942B ZA201803942B ZA2018/03942A ZA201803942A ZA201803942B ZA 201803942 B ZA201803942 B ZA 201803942B ZA 2018/03942 A ZA2018/03942 A ZA 2018/03942A ZA 201803942 A ZA201803942 A ZA 201803942A ZA 201803942 B ZA201803942 B ZA 201803942B
- Authority
- ZA
- South Africa
- Prior art keywords
- preparation
- integrase inhibitor
- novel processes
- integrase
- inhibitor
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IN201721020606 | 2017-06-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA201803942B true ZA201803942B (en) | 2021-05-26 |
Family
ID=62981290
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA2018/03942A ZA201803942B (en) | 2017-06-13 | 2018-06-13 | Novel processes for preparation of integrase inhibitor |
Country Status (2)
| Country | Link |
|---|---|
| WO (1) | WO2018229798A1 (en) |
| ZA (1) | ZA201803942B (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20220144851A1 (en) * | 2019-02-07 | 2022-05-12 | Cipla Limited | Novel polymorphs of integrase inhibitor |
| CN110041210A (en) * | 2019-05-06 | 2019-07-23 | 凯瑞斯德生化(苏州)有限公司 | A kind of Bictegravir intermediate and preparation method thereof |
| WO2020255004A1 (en) * | 2019-06-18 | 2020-12-24 | Laurus Labs Limited | Process and polymorphic forms of bictegravir and its pharmaceutically acceptable salts or co-crystals thereof |
| US11248005B2 (en) | 2019-07-08 | 2022-02-15 | Lupin Limited | Process for preparation of intermediates used for the synthesis of HIV integrase inhibitor |
| CN111978333B (en) * | 2019-09-30 | 2021-06-18 | 常州制药厂有限公司 | Crystal form A of Bictegravir sodium salt, preparation method and application |
| WO2022059028A1 (en) * | 2020-09-19 | 2022-03-24 | Msn Laboratories Private Limited, R&D Center | Novel polymorph of bictegravir sodium and process for preparation thereof |
| US20240309017A1 (en) * | 2021-01-22 | 2024-09-19 | Laurus Labs Limited | Processes for purification of bictegravir intermediates |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103154004B (en) * | 2010-08-05 | 2016-07-06 | 盐野义制药株式会社 | There is the manufacture method of the compound of hiv integrase inhibitory activity |
| AU2013361401C1 (en) | 2012-12-21 | 2018-08-09 | Gilead Sciences, Inc. | Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
| TWI744723B (en) | 2014-06-20 | 2021-11-01 | 美商基利科學股份有限公司 | Synthesis of polycyclic-carbamoylpyridone compounds |
-
2018
- 2018-06-13 ZA ZA2018/03942A patent/ZA201803942B/en unknown
- 2018-06-13 WO PCT/IN2018/050390 patent/WO2018229798A1/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| WO2018229798A1 (en) | 2018-12-20 |
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