SE0400208D0 - Chemical compounds - Google Patents
Chemical compoundsInfo
- Publication number
- SE0400208D0 SE0400208D0 SE0400208A SE0400208A SE0400208D0 SE 0400208 D0 SE0400208 D0 SE 0400208D0 SE 0400208 A SE0400208 A SE 0400208A SE 0400208 A SE0400208 A SE 0400208A SE 0400208 D0 SE0400208 D0 SE 0400208D0
- Authority
- SE
- Sweden
- Prior art keywords
- chemical compounds
- compounds
- chemokine
- modulators
- activity
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 102100024167 C-C chemokine receptor type 3 Human genes 0.000 abstract 1
- 101710149862 C-C chemokine receptor type 3 Proteins 0.000 abstract 1
- 102000019034 Chemokines Human genes 0.000 abstract 1
- 108010012236 Chemokines Proteins 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/40—Oxygen atoms
- C07D211/44—Oxygen atoms attached in position 4
- C07D211/52—Oxygen atoms attached in position 4 having an aryl radical as the second substituent in position 4
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/02—Nasal agents, e.g. decongestants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P11/14—Antitussive agents
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/16—Central respiratory analeptics
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A61P5/00—Drugs for disorders of the endocrine system
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Diabetes (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Virology (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pain & Pain Management (AREA)
- Cardiology (AREA)
- Molecular Biology (AREA)
- Psychiatry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Heart & Thoracic Surgery (AREA)
- AIDS & HIV (AREA)
- Hospice & Palliative Care (AREA)
Priority Applications (22)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0400208A SE0400208D0 (sv) | 2004-02-02 | 2004-02-02 | Chemical compounds |
PCT/SE2005/000110 WO2005073192A1 (en) | 2004-02-02 | 2005-01-31 | Novel piperidines as chemokine modulators (ccr) |
JP2006551005A JP4814109B2 (ja) | 2004-02-02 | 2005-01-31 | ケモカイン・モジュレーター(ccr)としての新規ピペリジン類 |
BRPI0507366-9A BRPI0507366A (pt) | 2004-02-02 | 2005-01-31 | novas piperidinas como moduladores de quimiocima (ccr) |
US10/587,633 US7956070B2 (en) | 2004-02-02 | 2005-01-31 | Piperidines as chemokine modulators (CCR) |
UY28731A UY28731A1 (es) | 2004-02-02 | 2005-01-31 | Compuestos quimicos |
KR1020067015578A KR20060128992A (ko) | 2004-02-02 | 2005-01-31 | 케모카인 조절제 (ccr)로서의 신규 피페리딘 |
RU2006130686/04A RU2348616C2 (ru) | 2004-02-02 | 2005-01-31 | Новые пиперидины в качестве модуляторов хемокинов (ccr) |
EP05704776A EP1713772A1 (en) | 2004-02-02 | 2005-01-31 | Novel piperidines as chemokine modulators (ccr) |
AU2005207817A AU2005207817B2 (en) | 2004-02-02 | 2005-01-31 | Novel piperidines as chemokine modulators (CCR) |
CNA2005800103948A CN1938274A (zh) | 2004-02-02 | 2005-01-31 | 用作趋化因子调节剂(ccr)的新哌啶化合物 |
CA002553089A CA2553089A1 (en) | 2004-02-02 | 2005-01-31 | Novel piperidines as chemokine modulators (ccr) |
NZ548781A NZ548781A (en) | 2004-02-02 | 2005-01-31 | Piperidine derivatives as chemokine modulators (CCR) |
TW094103106A TW200529843A (en) | 2004-02-02 | 2005-02-01 | Chemical compounds |
ARP050100391A AR049770A1 (es) | 2004-02-02 | 2005-02-02 | Derivados de piperidina como moduladores de la actividad de quimioquinas |
IL176992A IL176992A0 (en) | 2004-02-02 | 2006-07-20 | Novel piperidines as chemokine modulators (ccr) |
ZA200606199A ZA200606199B (en) | 2004-02-02 | 2006-07-26 | Novel piperidines as chemokine modulators (CCR) |
CO06073840A CO5700747A2 (es) | 2004-02-02 | 2006-07-27 | Piperidinas novedosas como moduladores de quimoquina (ccr) |
NO20063921A NO20063921L (no) | 2004-02-02 | 2006-09-01 | Nye piperidiner som kjemokinmodulatorer (CCR) |
JP2008226791A JP2009019055A (ja) | 2004-02-02 | 2008-09-04 | ケモカイン・モジュレーター(ccr)としての新規ピペリジン類 |
AU2008229856A AU2008229856A1 (en) | 2004-02-02 | 2008-10-09 | Novel piperidines as chemokine modulators (CCR) |
RU2008140910/04A RU2008140910A (ru) | 2004-02-02 | 2008-10-16 | Новые пиперидины в качестве модуляторов хемокинов (ccr) |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
SE0400208A SE0400208D0 (sv) | 2004-02-02 | 2004-02-02 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
SE0400208D0 true SE0400208D0 (sv) | 2004-02-02 |
Family
ID=31713276
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SE0400208A SE0400208D0 (sv) | 2004-02-02 | 2004-02-02 | Chemical compounds |
Country Status (19)
Country | Link |
---|---|
US (1) | US7956070B2 (sv) |
EP (1) | EP1713772A1 (sv) |
JP (2) | JP4814109B2 (sv) |
KR (1) | KR20060128992A (sv) |
CN (1) | CN1938274A (sv) |
AR (1) | AR049770A1 (sv) |
AU (2) | AU2005207817B2 (sv) |
BR (1) | BRPI0507366A (sv) |
CA (1) | CA2553089A1 (sv) |
CO (1) | CO5700747A2 (sv) |
IL (1) | IL176992A0 (sv) |
NO (1) | NO20063921L (sv) |
NZ (1) | NZ548781A (sv) |
RU (2) | RU2348616C2 (sv) |
SE (1) | SE0400208D0 (sv) |
TW (1) | TW200529843A (sv) |
UY (1) | UY28731A1 (sv) |
WO (1) | WO2005073192A1 (sv) |
ZA (1) | ZA200606199B (sv) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200303304A (en) * | 2002-02-18 | 2003-09-01 | Astrazeneca Ab | Chemical compounds |
SE0400208D0 (sv) | 2004-02-02 | 2004-02-02 | Astrazeneca Ab | Chemical compounds |
TW200812582A (en) * | 2006-04-06 | 2008-03-16 | Astrazeneca Ab | Medicaments |
US7897621B2 (en) | 2008-03-31 | 2011-03-01 | Hoffmann-La Roche Inc. | 2-trifluoromethylnicotinamide derivatives as HDL-cholesterol raising agents |
TWI433838B (zh) * | 2008-06-25 | 2014-04-11 | 必治妥美雅史谷比公司 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
US8410107B2 (en) | 2010-10-15 | 2013-04-02 | Hoffmann-La Roche Inc. | N-pyridin-3-yl or N-pyrazin-2-yl carboxamides |
US8669254B2 (en) | 2010-12-15 | 2014-03-11 | Hoffman-La Roche Inc. | Pyridine, pyridazine, pyrimidine or pyrazine carboxamides as HDL-cholesterol raising agents |
TW201418242A (zh) | 2012-10-26 | 2014-05-16 | Du Pont | 作為除草劑之經取代的三唑 |
PL3164394T3 (pl) | 2014-07-03 | 2020-09-07 | Board Of Regents, The University Of Texas System | Inhibitory GLS1 do leczenia chorób |
WO2016004417A1 (en) * | 2014-07-03 | 2016-01-07 | Board Of Regents, University Of Texas System | Gls1 inhibitors for treating disease |
EP3316887B1 (en) | 2015-06-30 | 2020-04-08 | Board of Regents, The University of Texas System | Gls1 inhibitors for treating disease |
JP6976248B2 (ja) | 2015-12-22 | 2021-12-08 | ボード オブ リージェンツ、ザ ユニバーシテイ オブ テキサス システム | (r)−1−(4−(6−(2−(4−(3,3−ジフルオロシクロブトキシ)−6−メチルピリジン−2−イル)アセトアミド)ピリダジン−3−イル)−2−フルオロブチル)−n−メチル−1h−1,2,3−トリアゾール−4−カルボキサミドの塩形態および多形体 |
US10722487B2 (en) | 2017-10-18 | 2020-07-28 | Board Of Regents, The University Of Texas System | Glutaminase inhibitor therapy |
WO2020025574A1 (en) | 2018-08-03 | 2020-02-06 | Bayer Aktiengesellschaft | Process for the preparation of 6-(haloalkyl)-2-halo-5-acylpyridines and intermediates for this process |
CN113121417A (zh) * | 2019-12-30 | 2021-07-16 | 苏州盛迪亚生物医药有限公司 | 一种新型哌啶衍生物及其药物用途 |
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- 2005-01-31 RU RU2006130686/04A patent/RU2348616C2/ru not_active IP Right Cessation
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RU2008140910A (ru) | 2010-04-27 |
IL176992A0 (en) | 2006-12-10 |
JP2007519717A (ja) | 2007-07-19 |
AU2008229856A1 (en) | 2008-11-06 |
US7956070B2 (en) | 2011-06-07 |
CA2553089A1 (en) | 2005-08-11 |
AU2005207817B2 (en) | 2008-07-24 |
RU2348616C2 (ru) | 2009-03-10 |
KR20060128992A (ko) | 2006-12-14 |
US20070054924A1 (en) | 2007-03-08 |
CO5700747A2 (es) | 2006-11-30 |
NO20063921L (no) | 2006-11-02 |
JP4814109B2 (ja) | 2011-11-16 |
AR049770A1 (es) | 2006-09-06 |
NZ548781A (en) | 2008-11-28 |
RU2006130686A (ru) | 2008-03-10 |
UY28731A1 (es) | 2005-09-30 |
WO2005073192A1 (en) | 2005-08-11 |
EP1713772A1 (en) | 2006-10-25 |
TW200529843A (en) | 2005-09-16 |
AU2005207817A1 (en) | 2005-08-11 |
JP2009019055A (ja) | 2009-01-29 |
BRPI0507366A (pt) | 2007-07-03 |
CN1938274A (zh) | 2007-03-28 |
ZA200606199B (en) | 2008-04-30 |
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