PT1259512E - Compostos de pteridin para o tratamento da psoriase - Google Patents

Compostos de pteridin para o tratamento da psoriase

Info

Publication number: PT1259512E
Authority: PT; Portugal
Prior art keywords: compounds; pteridin; psoriasis treatment; formula; psoriasis
Prior art date: 2000-02-23

Application number

PT01906493T

Other languages

English (en)

Inventor

Roger Bonnert

Stewart Gardiner

Fraser Hunt

Iain Walters

Original Assignee

Astrazeneca Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-02-23

Filing date

2001-02-20

Publication date

2004-02-27

2001-02-20 Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab

2004-02-27 Publication of PT1259512E publication Critical patent/PT1259512E/pt

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
- C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D475/00—Heterocyclic compounds containing pteridine ring systems
- C07D475/06—Heterocyclic compounds containing pteridine ring systems with a nitrogen atom directly attached in position 4

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Immunology (AREA)
Psychiatry (AREA)
Pulmonology (AREA)
Pain & Pain Management (AREA)
Dermatology (AREA)
Addiction (AREA)
Rheumatology (AREA)
Diabetes (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Cardiology (AREA)
Vascular Medicine (AREA)
Psychology (AREA)
Hematology (AREA)
Orthopedic Medicine & Surgery (AREA)
Physical Education & Sports Medicine (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

PT01906493T 2000-02-23 2001-02-20 Compostos de pteridin para o tratamento da psoriase PT1259512E (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB0004128A GB2359551A (en)	2000-02-23	2000-02-23	Pharmaceutically active pyrimidine derivatives

Publications (1)

Publication Number	Publication Date
PT1259512E true PT1259512E (pt)	2004-02-27

Family

ID=9886153

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
PT01906493T PT1259512E (pt)	2000-02-23	2001-02-20	Compostos de pteridin para o tratamento da psoriase

Country Status (33)

Country	Link
US (2)	US6875868B2 (pt)
EP (1)	EP1259512B1 (pt)
JP (1)	JP2003524012A (pt)
KR (1)	KR100795758B1 (pt)
CN (1)	CN1190437C (pt)
AR (1)	AR029805A1 (pt)
AT (1)	ATE250605T1 (pt)
AU (1)	AU782509B2 (pt)
BG (1)	BG107002A (pt)
BR (1)	BR0108600A (pt)
CA (1)	CA2400217C (pt)
CO (1)	CO5290258A1 (pt)
CZ (1)	CZ20022839A3 (pt)
DE (1)	DE60100851T2 (pt)
DK (1)	DK1259512T3 (pt)
EE (1)	EE200200461A (pt)
ES (1)	ES2206402T3 (pt)
GB (1)	GB2359551A (pt)
HK (1)	HK1050899A1 (pt)
HU (1)	HUP0204399A3 (pt)
IL (2)	IL151132A0 (pt)
IS (1)	IS6491A (pt)
MX (1)	MXPA02008233A (pt)
NO (1)	NO329898B1 (pt)
NZ (1)	NZ520355A (pt)
PL (1)	PL358004A1 (pt)
PT (1)	PT1259512E (pt)
RU (1)	RU2002125451A (pt)
SK (1)	SK12152002A3 (pt)
TR (1)	TR200302214T4 (pt)
UA (1)	UA72590C2 (pt)
WO (1)	WO2001062758A1 (pt)
ZA (1)	ZA200206590B (pt)

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2000
- 2000-02-23 GB GB0004128A patent/GB2359551A/en not_active Withdrawn
2001
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- 2001-02-20 EE EEP200200461A patent/EE200200461A/xx unknown
- 2001-02-20 CN CNB018054676A patent/CN1190437C/zh not_active Expired - Fee Related
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- 2001-02-20 JP JP2001562540A patent/JP2003524012A/ja active Pending
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- 2001-02-20 TR TR2003/02214T patent/TR200302214T4/xx unknown
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Also Published As

Publication number	Publication date
AU782509B2 (en)	2005-08-04
PL358004A1 (en)	2004-08-09
DK1259512T3 (da)	2003-12-29
NZ520355A (en)	2005-01-28
US20030055250A1 (en)	2003-03-20
NO20024005D0 (no)	2002-08-22
UA72590C2 (uk)	2005-03-15
NO20024005L (no)	2002-10-22
CN1190437C (zh)	2005-02-23
SK12152002A3 (sk)	2003-03-04
KR100795758B1 (ko)	2008-01-21
MXPA02008233A (es)	2004-04-05
TR200302214T4 (tr)	2004-01-21
DE60100851D1 (de)	2003-10-30
EE200200461A (et)	2003-12-15
HUP0204399A2 (en)	2003-05-28
AU3431601A (en)	2001-09-03
BR0108600A (pt)	2002-11-12
GB0004128D0 (en)	2000-04-12
GB2359551A (en)	2001-08-29
IS6491A (is)	2002-08-07
CA2400217A1 (en)	2001-08-30
WO2001062758A1 (en)	2001-08-30
EP1259512B1 (en)	2003-09-24
EP1259512A1 (en)	2002-11-27
US6875868B2 (en)	2005-04-05
KR20030005207A (ko)	2003-01-17
US7579342B2 (en)	2009-08-25
CA2400217C (en)	2009-02-17
HUP0204399A3 (en)	2004-11-29
HK1050899A1 (en)	2003-07-11
IL151132A0 (en)	2003-04-10
CZ20022839A3 (cs)	2002-11-13
ATE250605T1 (de)	2003-10-15
IL151132A (en)	2010-11-30
RU2002125451A (ru)	2004-01-10
US20050171345A1 (en)	2005-08-04
JP2003524012A (ja)	2003-08-12
CN1404482A (zh)	2003-03-19
NO329898B1 (no)	2011-01-24
BG107002A (bg)	2003-04-30
CO5290258A1 (es)	2003-06-27
ES2206402T3 (es)	2004-05-16
DE60100851T2 (de)	2004-07-15
AR029805A1 (es)	2003-07-16
ZA200206590B (en)	2003-11-17

Publication	Publication Date	Title
PT1259512E (pt)	2004-02-27	Compostos de pteridin para o tratamento da psoriase
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BG66080B1 (bg)	2011-03-31	Заместени тиоацетамиди
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BR9911488A (pt)	2001-03-20	Composto, uso do mesmo, composição farmacêutica, e, processos para tratamento ou de profilaxia de doenças inflamatórias, e para a preparação de um composto
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ATE358668T1 (de)	2007-04-15	Drogen zur behandlung maligner tumoren
BRPI0410316A (pt)	2006-05-23	composto, composição farmacêutica, uso dos compostos, e, método de tratamento de distúrbios mediados por vr1 e para o tratamento de distúrbios de dores
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SE9804212D0 (sv)	1998-12-04	Compounds
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