PE20160026A1 - Compuestos heterociclicos como agentes para control de plagas - Google Patents

Compuestos heterociclicos como agentes para control de plagas

Info

Publication number
PE20160026A1
PE20160026A1 PE2015002428A PE2015002428A PE20160026A1 PE 20160026 A1 PE20160026 A1 PE 20160026A1 PE 2015002428 A PE2015002428 A PE 2015002428A PE 2015002428 A PE2015002428 A PE 2015002428A PE 20160026 A1 PE20160026 A1 PE 20160026A1
Authority
PE
Peru
Prior art keywords
hydrogen
alkyl
heterocyclic compounds
agents
pest control
Prior art date
Application number
PE2015002428A
Other languages
English (en)
Inventor
Olga Malsam
Peter Losel
Kerstin Ilg
Mehmet Gueclue
Peter Reinisch
Christoph Grondal
Martin Fublein
Reiner Fischer
Thomas Bretschneider
Silvia Cerezo-Galvez
Arnd Voerste
Peter Jeschke
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of PE20160026A1 publication Critical patent/PE20160026A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Dentistry (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

La presente solicitud esta referida a compuestos heterociclicos de formula (I), en donde Het es un radical de formula como se indica. G1 es N, etc. A1 es hidrogeno, halogeno, etc. A2 es hidrogeno, halogeno, etc. R es hidrogeno, alquilo, etc. R1 es hidrogeno, alquilo, etc. R2 es hidrogeno o alquilo, Q es N o C-R3, R3 es hidrogeno, alquilo, etc. V es un radical oxigeno, azufre, etc. Estos compuestos son empleados para el control de plagas de animales. La solicitud tambien esta orientada a la preparacion de los mismos. Son compuestos preferidos: 5-Etil-2-(piridin-3-il)-6-(trifluorometil)-2,5-dihidro-4H-pirazolo[3,4-d]pirimidin-4-ona (32), 3-Isopropil-6-(3-piridyl)pirazolo[3,4-d]triazin-4-ona(36)
PE2015002428A 2013-05-28 2014-05-23 Compuestos heterociclicos como agentes para control de plagas PE20160026A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP13169415 2013-05-28

Publications (1)

Publication Number Publication Date
PE20160026A1 true PE20160026A1 (es) 2016-02-03

Family

ID=48520750

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2015002428A PE20160026A1 (es) 2013-05-28 2014-05-23 Compuestos heterociclicos como agentes para control de plagas

Country Status (16)

Country Link
US (1) US9688681B2 (es)
EP (1) EP3003042B1 (es)
JP (1) JP6466921B2 (es)
KR (1) KR20160012170A (es)
CN (1) CN105744838B (es)
AR (1) AR096446A1 (es)
AU (1) AU2014273299A1 (es)
BR (1) BR112015029258A2 (es)
CA (1) CA2913509A1 (es)
CL (1) CL2015003405A1 (es)
EA (1) EA201501142A1 (es)
ES (1) ES2640794T3 (es)
MX (1) MX2015016029A (es)
PE (1) PE20160026A1 (es)
PH (1) PH12015502649A1 (es)
WO (1) WO2014191301A1 (es)

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BR112015020242A2 (pt) 2013-02-28 2017-07-18 Janssen Sciences Ireland Uc sulfamoil-arilamidas e seu uso como medicamentos para o tratamento da hepatite b
EP2981536B1 (en) 2013-04-03 2017-06-14 Janssen Sciences Ireland UC N-phenyl-carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis b
CN105960400B (zh) 2013-05-17 2019-05-31 爱尔兰詹森科学公司 氨磺酰基噻吩酰胺衍生物及其作为药物用于治疗乙型肝炎的用途
JO3603B1 (ar) 2013-05-17 2020-07-05 Janssen Sciences Ireland Uc مشتقات سلفامويل بيرولاميد واستخدامها كادوية لمعالجة التهاب الكبد نوع بي
SG10201805033XA (en) 2013-07-25 2018-07-30 Janssen Sciences Ireland Uc Glyoxamide substituted pyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis b
TWI652014B (zh) 2013-09-13 2019-03-01 美商艾佛艾姆希公司 雜環取代之雙環唑殺蟲劑
WO2015059212A1 (en) 2013-10-23 2015-04-30 Janssen R&D Ireland Carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis b
US10392349B2 (en) 2014-01-16 2019-08-27 Novira Therapeutics, Inc. Azepane derivatives and methods of treating hepatitis B infections
US9169212B2 (en) 2014-01-16 2015-10-27 Novira Therapeutics, Inc. Azepane derivatives and methods of treating hepatitis B infections
RU2702109C1 (ru) 2014-02-05 2019-10-04 Новира Терапьютикс, Инк. Комбинированная терапия для лечения инфекций вгв
AP2016009257A0 (en) 2014-02-06 2016-06-30 Janssen Sciences Ireland Uc Sulphamoylpyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis b
JP6445040B2 (ja) * 2014-03-10 2018-12-26 バイエル・クロップサイエンス・アクチェンゲゼルシャフト 殺虫剤としてのヘテロ環化合物
ES2778628T3 (es) 2015-03-12 2020-08-11 Fmc Corp Pesticidas de azol bicíclico sustituido con heterociclo
CN107847762A (zh) 2015-03-19 2018-03-27 诺维拉治疗公司 氮杂环辛烷和氮杂环壬烷衍生物以及治疗乙型肝炎感染的方法
WO2016164200A1 (en) 2015-04-09 2016-10-13 E I Du Pont De Nemours And Company Bicyclic pyrazole pesticides
US10875876B2 (en) 2015-07-02 2020-12-29 Janssen Sciences Ireland Uc Cyclized sulfamoylarylamide derivatives and the use thereof as medicaments for the treatment of hepatitis B
EP3356328A1 (en) 2015-09-29 2018-08-08 Novira Therapeutics, Inc. Crystalline forms of a hepatitis b antiviral agent
BR112018071048A2 (pt) 2016-04-15 2019-05-07 Janssen Sciences Ireland Uc combinações e métodos que compreendem um inibidor da montagem de capsídeos
SG11202007097QA (en) 2018-03-14 2020-08-28 Janssen Sciences Ireland Unlimited Co Capsid assembly modulator dosing regimen
TW202045499A (zh) 2019-02-22 2020-12-16 愛爾蘭商健生科學愛爾蘭無限公司 用於治療ｈｂｖ感染或ｈｂｖ誘發疾病之醯胺衍生物
MA55879A (fr) 2019-05-06 2022-03-16 Janssen Sciences Ireland Unlimited Co Dérivés d'amide utiles dans le traitement d'une infection par le virus de l'hépatite b ou de maladies induites par le virus de l'hépatite b
UY39475A (es) * 2020-10-19 2022-05-31 Adama Makhteshim Ltd Compuestos útiles para la preparación de pirazolopirimidinonas
CN112939980A (zh) * 2021-03-10 2021-06-11 南开大学 一类3,4-二氯异噻唑杂环嘌呤类衍生物及其制备方法和用途
WO2024214046A1 (en) 2023-04-14 2024-10-17 Takeda Pharmaceutical Company Limited Pyrazolopyrimidine derivatives as inhibitors of nlrp3

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JP2006525966A (ja) * 2003-05-09 2006-11-16 バイエル・ヘルスケア・アクチェンゲゼルシャフト ６−シクリルメチル−および６−アルキルメチル置換ピラゾロピリミジン類
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Also Published As

Publication number Publication date
CA2913509A1 (en) 2014-12-04
EP3003042A1 (de) 2016-04-13
EA201501142A1 (ru) 2016-05-31
AR096446A1 (es) 2015-12-30
AU2014273299A1 (en) 2015-12-17
CN105744838A (zh) 2016-07-06
JP6466921B2 (ja) 2019-02-06
US20160122353A1 (en) 2016-05-05
EP3003042B1 (de) 2017-06-21
BR112015029258A2 (pt) 2017-07-25
PH12015502649A1 (en) 2016-03-07
CL2015003405A1 (es) 2016-09-09
JP2016524613A (ja) 2016-08-18
ES2640794T3 (es) 2017-11-06
WO2014191301A1 (de) 2014-12-04
KR20160012170A (ko) 2016-02-02
US9688681B2 (en) 2017-06-27
CN105744838B (zh) 2017-12-08
MX2015016029A (es) 2016-03-21

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