NO930816L - Nye aminokarboksylsyrederivater med antiallergisk/antiastmatisk virkning og fremgangsmaate for deres fremstilling - Google Patents
Nye aminokarboksylsyrederivater med antiallergisk/antiastmatisk virkning og fremgangsmaate for deres fremstillingInfo
- Publication number
- NO930816L NO930816L NO93930816A NO930816A NO930816L NO 930816 L NO930816 L NO 930816L NO 93930816 A NO93930816 A NO 93930816A NO 930816 A NO930816 A NO 930816A NO 930816 L NO930816 L NO 930816L
- Authority
- NO
- Norway
- Prior art keywords
- carbon atoms
- preparation
- acid derivatives
- aminocarboxylic acid
- antiastmatic
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C07D237/30—Phthalazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/26—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings condensed with carbocyclic rings or ring systems
- C07D237/30—Phthalazines
- C07D237/32—Phthalazines with oxygen atoms directly attached to carbon atoms of the nitrogen-containing ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Pulmonology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Forbindelse med generell formel I der R1 betyr hydrogen, en rettkjedet eller forgrenet alkylrest med 1-6 karbonatomer, benzyl eller fenyletyl, R2 betyr hydrogen, en rettkjedet eller forgrenet alkylrest med 1-6 karbonatomer, benzyl eller fenyletyl, R3 betyr hydrogen, en rettkjedet eller forgrenet alkylrest med 1-6 karbonatomer eller utgjøre benzyl, Ri og R2 kan være like eller forskjellige, X har betydningen hydrogen, halogen, C1-C^)-alkyl eller alkoksy, der alkylkjeden har en lengde på 1-6 karbon- atomer , Y! og Y2 kan være like eller forskjellige og betyr hydrogen, halogen, alkyl med 1-6 karbonatomer eller alkoksy med 1-6 karbonatomer, der m, n og o kan anta verdier fra 0-4. Forbindelsene er nye 6-aminokarboksylsyre-derivater med antiastmatiske og antiallergiske egenskaper, og de kan bli anvendt for fremstilling av legemidler.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4207234A DE4207234A1 (de) | 1992-03-07 | 1992-03-07 | Neue aminocarbonsaeure-derivate mit antiallergischer/antiasthmatischer wirkung und verfahren zu deren herstellung |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO930816D0 NO930816D0 (no) | 1993-03-05 |
| NO930816L true NO930816L (no) | 1993-09-08 |
Family
ID=6453459
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO93930816A NO930816L (no) | 1992-03-07 | 1993-03-05 | Nye aminokarboksylsyrederivater med antiallergisk/antiastmatisk virkning og fremgangsmaate for deres fremstilling |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US5464838A (no) |
| EP (1) | EP0564805A1 (no) |
| JP (1) | JPH069575A (no) |
| KR (1) | KR930019639A (no) |
| CN (1) | CN1080286A (no) |
| AU (1) | AU659717B2 (no) |
| CA (1) | CA2091105A1 (no) |
| DE (1) | DE4207234A1 (no) |
| FI (1) | FI930993A (no) |
| HU (1) | HUT63617A (no) |
| MX (1) | MX9301237A (no) |
| NO (1) | NO930816L (no) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HUE030388T2 (en) | 2004-11-24 | 2017-05-29 | Meda Pharmaceuticals Inc | Preparations and methods of use containing azelastine |
| US20070020330A1 (en) | 2004-11-24 | 2007-01-25 | Medpointe Healthcare Inc. | Compositions comprising azelastine and methods of use thereof |
| US8758816B2 (en) | 2004-11-24 | 2014-06-24 | Meda Pharmaceuticals Inc. | Compositions comprising azelastine and methods of use thereof |
| WO2010019417A2 (en) * | 2008-08-13 | 2010-02-18 | Boehringer Ingelheim International Gmbh | Chymase inhibitors |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3017411A (en) * | 1962-01-16 | New substituted phthalazones and proc- | ||
| DE1046625B (de) * | 1957-08-15 | 1958-12-18 | Hydrierwerk Rodleben Veb | Verfahren zur Herstellung basisch substituierter Phthalazone |
| CH572914A5 (no) * | 1971-01-22 | 1976-02-27 | Asta Werke Ag Chem Fab | |
| US4207112A (en) * | 1974-01-29 | 1980-06-10 | Fuji Photo Film Co., Ltd. | Heat developable light-sensitive materials |
| US4665181A (en) * | 1984-05-17 | 1987-05-12 | Pennwalt Corporation | Anti-inflammatory phthalazinones |
| DE3575135D1 (de) * | 1984-09-14 | 1990-02-08 | Asta Pharma Ag | Substituierte benzylphthalazinon-derivate. |
| ATE60598T1 (de) * | 1985-11-11 | 1991-02-15 | Asta Pharma Ag | 4-benzyl-1-(2h)-phthalazinon-derivate. |
| ZA882639B (en) * | 1987-05-02 | 1988-09-30 | Asta-Pharma Aktiengesellschaft | New 2-aminoalkyl-4-benzyl-1(2h)-phthalazinone derivatives |
| DE3813531A1 (de) * | 1987-05-02 | 1988-11-10 | Asta Pharma Ag | Neue 2-aminoalkyl-4-benzyl-1-(2h)-phthalazinon-derivate |
| EP0289939A1 (de) * | 1987-05-08 | 1988-11-09 | ASTA Pharma AG | Neue 4-Benzyl-1-(2H)-phthalazinon-Derivate mit einem Aminosäurerest |
| MC2025A1 (fr) * | 1988-04-20 | 1990-04-25 | Asta Pharma Ag | Medicament contenant de l'azelastine et capable de liberer celle-ci de facon controlee |
| JPH04198180A (ja) * | 1990-11-28 | 1992-07-17 | Eezai Kagaku Kk | ベンジルフタラゾン誘導体の製造方法 |
-
1992
- 1992-03-07 DE DE4207234A patent/DE4207234A1/de not_active Withdrawn
-
1993
- 1993-02-27 EP EP93103179A patent/EP0564805A1/de not_active Withdrawn
- 1993-03-04 US US08/027,487 patent/US5464838A/en not_active Expired - Fee Related
- 1993-03-05 MX MX9301237A patent/MX9301237A/es unknown
- 1993-03-05 JP JP5044841A patent/JPH069575A/ja active Pending
- 1993-03-05 CA CA002091105A patent/CA2091105A1/en not_active Abandoned
- 1993-03-05 NO NO93930816A patent/NO930816L/no unknown
- 1993-03-05 FI FI930993A patent/FI930993A/fi not_active Application Discontinuation
- 1993-03-05 HU HU9300626A patent/HUT63617A/hu unknown
- 1993-03-06 CN CN93103493A patent/CN1080286A/zh not_active Withdrawn
- 1993-03-06 KR KR1019930003363A patent/KR930019639A/ko not_active Application Discontinuation
- 1993-03-08 AU AU34052/93A patent/AU659717B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| FI930993A0 (fi) | 1993-03-05 |
| AU659717B2 (en) | 1995-05-25 |
| MX9301237A (es) | 1993-09-01 |
| HUT63617A (en) | 1993-09-28 |
| DE4207234A1 (de) | 1993-09-09 |
| CN1080286A (zh) | 1994-01-05 |
| NO930816D0 (no) | 1993-03-05 |
| JPH069575A (ja) | 1994-01-18 |
| AU3405293A (en) | 1993-09-09 |
| FI930993A (fi) | 1993-09-08 |
| US5464838A (en) | 1995-11-07 |
| CA2091105A1 (en) | 1993-09-08 |
| KR930019639A (ko) | 1993-10-18 |
| EP0564805A1 (de) | 1993-10-13 |
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