NO20052888L - Diamintriazoler anvendelige som inhibitorer av proteinkinaser - Google Patents

Diamintriazoler anvendelige som inhibitorer av proteinkinaser

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Publication number
NO20052888L
NO20052888L NO20052888A NO20052888A NO20052888L NO 20052888 L NO20052888 L NO 20052888L NO 20052888 A NO20052888 A NO 20052888A NO 20052888 A NO20052888 A NO 20052888A NO 20052888 L NO20052888 L NO 20052888L
Authority
NO
Norway
Prior art keywords
inhibitors
protein kinases
diamin
triazoles useful
triazoles
Prior art date
Application number
NO20052888A
Other languages
English (en)
Other versions
NO20052888D0 (no
Inventor
Michael J Arnost
Cornelia J Forster
Robert J Davies
Albert Pierce
Hayley Binch
Mark Ledeboer
Brian E Ledford
Vincent Galullo
Ronald Grey
Shi-Kai Tian
Jinwang Xu
David Messersmith
Sughanthi Nanthakumar
Andrew Jayaraj
Original Assignee
Vertex Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vertex Pharma filed Critical Vertex Pharma
Publication of NO20052888D0 publication Critical patent/NO20052888D0/no
Publication of NO20052888L publication Critical patent/NO20052888L/no

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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D487/04—Ortho-condensed systems
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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Abstract

Foreliggende oppfinnelse vedrører inhibitorer av proteinkinaser. Oppfinnelsen tilveiebringer også farmasøytiske sammensetninger omfattende forbindelsene ifølge oppfinnelsen og metoder for anvendelse av sammensetningene i behandlingen av forskjellige forstyrrelser.
NO20052888A 2002-11-15 2005-06-10 Diamintriazoler anvendelige som inhibitorer av proteinkinaser NO20052888L (no)

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AU2003294329B2 (en) 2010-04-29
BR0316350A (pt) 2005-09-27
JP4783020B2 (ja) 2011-09-28
US7902239B2 (en) 2011-03-08
WO2004046120A2 (en) 2004-06-03
ES2318189T3 (es) 2009-05-01
DK1562589T3 (da) 2009-02-16
US20080014189A1 (en) 2008-01-17
EP1562589B1 (en) 2009-01-07
RU2350606C2 (ru) 2009-03-27
NO20052888D0 (no) 2005-06-10
CA2505789A1 (en) 2004-06-03
EP1562589A2 (en) 2005-08-17
ATE419849T1 (de) 2009-01-15
JP2006515313A (ja) 2006-05-25
SI1562589T1 (sl) 2009-06-30
US7279469B2 (en) 2007-10-09
TWI335913B (en) 2011-01-11
AU2003294329A1 (en) 2004-06-15
WO2004046120A3 (en) 2004-08-12
NZ540662A (en) 2008-04-30
PT1562589E (pt) 2009-04-15
US20040214817A1 (en) 2004-10-28
DE60325761D1 (de) 2009-02-26
PL377825A1 (pl) 2006-02-20
RU2005118418A (ru) 2006-02-10
AR042052A1 (es) 2005-06-08
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JP2011132263A (ja) 2011-07-07

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