MX163202B - 5-aroil derivados de acidos 1,2-dihidro-3h-pirrolo(1,2-a)pirrol-1-carboxilicos - Google Patents

5-aroil derivados de acidos 1,2-dihidro-3h-pirrolo(1,2-a)pirrol-1-carboxilicos

Info

Publication number: MX163202B
Authority: MX; Mexico
Prior art keywords: carboxilicos; aroil; pirrol; pirrolo; dihidro
Prior art date: 1976-07-14

Application number

MX9100104A

Other languages

English (en)

Spanish (es)

Inventor

Joseph M Muchowski

Arthur F Kluge

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-07-14

Filing date

1991-07-05

Publication date

1992-02-20

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX163202(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1977-02-23 Priority claimed from US05/771,286 external-priority patent/US4089969A/en

1991-07-05 Application filed by Syntex Inc filed Critical Syntex Inc

1992-02-20 Publication of MX163202B publication Critical patent/MX163202B/es

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)

MX9100104A 1976-07-14 1991-07-05 5-aroil derivados de acidos 1,2-dihidro-3h-pirrolo(1,2-a)pirrol-1-carboxilicos MX163202B (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US70490976A	1976-07-14	1976-07-14
US05/771,286 US4089969A (en)	1976-07-14	1977-02-23	5-Aroyl-1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid derivatives and process for the production thereof

Publications (1)

Publication Number	Publication Date
MX163202B true MX163202B (es)	1992-02-20

Family

ID=27107410

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
MX9100104A MX163202B (es)	1976-07-14	1991-07-05	5-aroil derivados de acidos 1,2-dihidro-3h-pirrolo(1,2-a)pirrol-1-carboxilicos

Country Status (27)

Country	Link
JP (1)	JPS539788A (de)
AR (1)	AR224997A1 (de)
CA (1)	CA1102809A (de)
CH (3)	CH641458A5 (de)
CS (1)	CS204954B2 (de)
DE (2)	DE2760330C2 (de)
DK (1)	DK151886C (de)
ES (2)	ES460706A1 (de)
FI (1)	FI63406C (de)
FR (2)	FR2358406A1 (de)
GB (1)	GB1554075A (de)
GR (1)	GR61111B (de)
HK (1)	HK15981A (de)
HU (1)	HU174224B (de)
IE (1)	IE45253B1 (de)
IL (2)	IL52493A (de)
IT (1)	IT1117313B (de)
MX (1)	MX163202B (de)
MY (1)	MY8100357A (de)
NL (2)	NL186318C (de)
NO (1)	NO147564C (de)
NZ (1)	NZ184610A (de)
PL (4)	PL109390B1 (de)
PT (1)	PT66780B (de)
SE (1)	SE434643B (de)
SU (1)	SU695558A3 (de)
YU (1)	YU40816B (de)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4140698A (en) *	1977-07-25	1979-02-20	Syntex (Usa) Inc.	1,2-Dihydro-3H-pyrrolo[1,2-a]pyrrole-1-nitriles
JPS55124633A (en) *	1979-03-19	1980-09-25	Sohachi Takeuchi	Manufacturing method of tubular vessel
US4344943A (en) *	1980-06-09	1982-08-17	Syntex (U.S.A.) Inc.	6-Chloro- or 6-bromo-1,2-dihydro-3H-pyrrolo[1,2-a]-pyrrole-1-carboxylic acids and derivatives thereof
US4353829A (en) *	1980-11-21	1982-10-12	Syntex (U.S.A.) Inc.	Process for 5-aroylation of 1,2-dihydro-3H-pyrrolo[1,2-a]pyrrole-1-carboxylic esters
US4511724A (en) *	1982-06-10	1985-04-16	Merck & Co., Inc.	5-(Pyrrol-2-oyl)-1,2-dihydro-3H-pyrrolo [1,2-a]pyrrole derivatives as anti-inflammatory and analgesic agents
JPS5910589A (ja) *	1982-06-10	1984-01-20	メルク　エンド　カムパニー　インコーポレーテツド	抗炎症剤および鎮痛剤として新規な５−（ピロ−ル−２−オイル）−１，２−ジヒドロ−３Ｈ−ピロロ〔１，２−ａ〕ピロ−ル誘導体
US4874871A (en) *	1987-03-25	1989-10-17	Syntex (U.S.A.) Inc.	Process for preparing (+)-2,3-Dihydro-1H-pyrrolo[1,2-a]pyrrole-1-carboxylic acid and related compounds
JPH0739418B2 (ja) *	1987-09-10	1995-05-01	久光製薬株式会社	新規な３−アロイル−６，７−ジヒドロ−５Ｈ−ピロロ〔１，２−ｃ〕イミダゾール−７−カルボン酸誘導体
JP2649168B2 (ja) *	1988-02-25	1997-09-03	久光製薬株式会社	新規な５，６−ジフェニル−１，２−ジヒドロ−３Ｈ−ピロロ［１，２−ａ］ピロール−１−カルボン酸誘導体
IT1250691B (it) *	1991-07-22	1995-04-21	Giancarlo Santus	Composizioni terapeutiche per somministrazione intranasale comprendenti ketorolac.
JP2902113B2 (ja) *	1991-11-11	1999-06-07	久光製薬株式会社	ケトロラク含有シップ剤
DE4300697C1 (de) *	1993-01-13	1994-05-19	Roemmers Sa	Keterolac-Derivat mit wesentlich geringerer gastrointestinaler Reizung und Ulzeration
US5622948A (en) *	1994-12-01	1997-04-22	Syntex (U.S.A.) Inc.	Pyrrole pyridazine and pyridazinone anti-inflammatory agents
JP2008210666A (ja) *	2007-02-27	2008-09-11	Okamura Corp	商品陳列棚における照明装置

1977
- 1977-05-17 JP JP5697777A patent/JPS539788A/ja active Granted
- 1977-07-07 GR GR53907A patent/GR61111B/el unknown
- 1977-07-07 DK DK307577A patent/DK151886C/da active
- 1977-07-07 AR AR268356A patent/AR224997A1/es active
- 1977-07-08 PT PT66780A patent/PT66780B/pt unknown
- 1977-07-08 IE IE1423/77A patent/IE45253B1/en not_active IP Right Cessation
- 1977-07-08 IL IL52493A patent/IL52493A/xx unknown
- 1977-07-08 CH CH850077A patent/CH641458A5/de not_active IP Right Cessation
- 1977-07-08 NL NLAANVRAGE7707651,A patent/NL186318C/xx not_active IP Right Cessation
- 1977-07-11 FI FI772153A patent/FI63406C/fi not_active IP Right Cessation
- 1977-07-11 GB GB28919/77A patent/GB1554075A/en not_active Expired
- 1977-07-11 NZ NZ184610A patent/NZ184610A/xx unknown
- 1977-07-11 YU YU1721/77A patent/YU40816B/xx unknown
- 1977-07-11 FR FR7721356A patent/FR2358406A1/fr active Granted
- 1977-07-12 CA CA282,599A patent/CA1102809A/en not_active Expired
- 1977-07-12 CS CS774646A patent/CS204954B2/cs unknown
- 1977-07-13 SU SU772501050A patent/SU695558A3/ru active
- 1977-07-13 PL PL1977199603A patent/PL109390B1/pl unknown
- 1977-07-13 PL PL1977227290A patent/PL124444B1/pl unknown
- 1977-07-13 ES ES460706A patent/ES460706A1/es not_active Expired
- 1977-07-13 DE DE2760330A patent/DE2760330C2/de not_active Expired
- 1977-07-13 PL PL1977227289A patent/PL124711B1/pl unknown
- 1977-07-13 SE SE7708141A patent/SE434643B/xx not_active IP Right Cessation
- 1977-07-13 IT IT68630/77A patent/IT1117313B/it active Protection Beyond IP Right Term
- 1977-07-13 PL PL1977227291A patent/PL124445B1/pl unknown
- 1977-07-13 NO NO772494A patent/NO147564C/no unknown
- 1977-07-13 DE DE19772731678 patent/DE2731678A1/de active Granted
- 1977-07-14 HU HU77SI1582A patent/HU174224B/hu unknown
- 1977-12-20 FR FR7738508A patent/FR2375234A1/fr active Granted
1978
- 1978-05-24 ES ES470214A patent/ES470214A1/es not_active Expired
1979
- 1979-11-22 IL IL58779A patent/IL58779A0/xx unknown
1981
- 1981-04-23 HK HK159/81A patent/HK15981A/xx unknown
- 1981-12-30 MY MY357/81A patent/MY8100357A/xx unknown
1984
- 1984-02-22 CH CH86584A patent/CH646972A5/de not_active IP Right Cessation
- 1984-02-22 CH CH86684A patent/CH646973A5/de not_active IP Right Cessation
1991
- 1991-07-05 MX MX9100104A patent/MX163202B/es unknown
1993
- 1993-03-23 NL NL930021C patent/NL930021I2/nl unknown

Also Published As

Publication number	Publication date
FR2375234A1 (fr)	1978-07-21
YU172177A (en)	1983-09-30
NO147564B (no)	1983-01-24
FI772153A (de)	1978-01-15
ES460706A1 (es)	1978-12-01
DK151886B (da)	1988-01-11
DE2760330C2 (de)	1989-06-15
IT1117313B (it)	1986-02-17
DE2731678C2 (de)	1989-06-08
JPS6254109B2 (de)	1987-11-13
FR2358406B1 (de)	1981-04-17
CA1102809A (en)	1981-06-09
FI63406B (fi)	1983-02-28
FI63406C (fi)	1983-06-10
IL52493A0 (en)	1977-10-31
AU513384B2 (en)	1980-11-27
FR2358406A1 (fr)	1978-02-10
YU40816B (en)	1986-06-30
NL186318B (nl)	1990-06-01
SU695558A3 (ru)	1979-10-30
NZ184610A (en)	1979-03-28
IE45253L (en)	1978-01-14
FR2375234B1 (de)	1980-11-07
ES470214A1 (es)	1979-09-16
NL7707651A (nl)	1978-01-17
PL124711B1 (en)	1983-02-28
DK151886C (da)	1988-06-06
HU174224B (hu)	1979-11-28
AR224997A1 (es)	1982-02-15
NO772494L (no)	1978-01-17
DE2731678A1 (de)	1978-03-16
GB1554075A (en)	1979-10-17
IL52493A (en)	1982-02-28
DK307577A (da)	1978-01-15
IE45253B1 (en)	1982-07-14
GR61111B (en)	1978-09-12
PL199603A1 (pl)	1978-04-24
NO147564C (no)	1983-05-18
PL124444B1 (en)	1983-01-31
SE7708141L (sv)	1978-01-15
PL109390B1 (en)	1980-05-31
HK15981A (en)	1981-05-01
CH646973A5 (en)	1984-12-28
PT66780A (fr)	1977-08-01
PL124445B1 (en)	1983-01-31
NL930021I1 (nl)	1993-05-03
CS204954B2 (en)	1981-04-30
IL58779A0 (en)	1980-02-29
SE434643B (sv)	1984-08-06
CH646972A5 (en)	1984-12-28
PT66780B (fr)	1978-12-18
NL186318C (nl)	1990-11-01
NL930021I2 (nl)	1997-03-03
AU2697577A (en)	1979-01-18
JPS539788A (en)	1978-01-28
MY8100357A (en)	1981-12-31
CH641458A5 (en)	1984-02-29

Publication	Publication Date	Title
DK343980A (da)	1981-02-10	2,4,6-triiod-isophthalsyrederivater
DK343880A (da)	1981-02-10	2,4,6-triiod-isophthalsyrederivater
NO791140L (no)	1979-10-08	Tioetiansyrederivater.
NL7806333A (nl)	1978-12-19	Olefinemaleinezuur-copolymeerderivaten.
NL7704210A (nl)	1977-10-25	Fenoxy-fenoxypropionzuurderivaten.
IL52150A0 (en)	1977-07-31	Phenoxyphenoxy-propionic acid derivatives
NL7709442A (nl)	1978-03-15	Werkwijze voor imidazo-(1,2-a)-chinoline-2- -carbonzuurderivaten.
SE7806711L (sv)	1978-12-11	7alfa-metoxi-7beta-(1,3-ditietan-2-karboxamido)-cefalosporansyraderivat
AU2241677A (en)	1978-08-24	4,5-dichloroimidazole-2-carboxylic acid derivatives
NZ183824A (en)	1980-10-24	5-phenyl-trans-1,3,4,4a,5,9b-hexahydro-2h-pyrido-(4,3-b)-indol-2-yl-alkanols-alkanones or-alkanoic acid derivatives
GB1548820A (en)	1979-07-18	9-thia11- oxo -12 - azaprotanoic acid derivatives
MX163202B (es)	1992-02-20	5-aroil derivados de acidos 1,2-dihidro-3h-pirrolo(1,2-a)pirrol-1-carboxilicos
NO774131L (no)	1978-11-07	Pyrimido(6,1-a)isokinolin-2-on-derivater
IT7848582A0 (it)	1978-03-23	Immidazo(1,2-a)-piridine eterociclo -sostituite nuove
FI772628A (fi)	1978-03-09	7-acylamino-8-oxo-3-oxa-1-azabicyklo(4.2.0)-octan-2-carboxyl-syraderivat
NO803592L (no)	1981-05-29	4,5-umettede prostansyre-derivater.
RO70629A (ro)	1981-01-30	Procedeu pentru prepararea 1,1-dioxidului de acid 3,4-dihidro-2-metil-4-oxo-2h-1,2-benzotiazin-3-carboxilic
NL7705896A (nl)	1977-11-29	Polyprenylcarbonzuurderivaten.
IL52244A0 (en)	1977-08-31	Clavam-3-carboxylic acid derivatives
NL7807871A (nl)	1979-01-30	Alpha-halogeenmethylaminozuur derivaten.
BE842782A (fr)	1976-12-10	4,5-dihydrotetrazolo (1,5-a)- quinoxalines
NL7801576A (nl)	1978-08-15	Benzoheterocyclylglyoxylzuurderivaten.
NL7810254A (nl)	1979-05-02	Olefine-maleinezuur-copolymeerderivaten.
IL51605A0 (en)	1977-05-31	Phenoxyphenoxy-alkanecarboxylic acid derivatives
DK573678A (da)	1979-06-23	3,4-methano-pyrrolidinderivater