JPS5473780A - Novel benzamide derivative - Google Patents
Novel benzamide derivativeInfo
- Publication number
- JPS5473780A JPS5473780A JP13769777A JP13769777A JPS5473780A JP S5473780 A JPS5473780 A JP S5473780A JP 13769777 A JP13769777 A JP 13769777A JP 13769777 A JP13769777 A JP 13769777A JP S5473780 A JPS5473780 A JP S5473780A
- Authority
- JP
- Japan
- Prior art keywords
- group
- imino
- alkyl
- formula
- alkyl group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pyrrole Compounds (AREA)
Abstract
NEW MATERIAL:A benzamide derivative of formula I: (R is alkyl group; R1 is alkyl, aralkyl, or dialkylamino-alkyl group; R2 is H, alkyl or halogen; X is H, halogen, alkyl group, amino, imino, mercapto, thioxo, OH, or oxo group; Y is nitrylo, imino, alkylimino, dialkylaminoalkyl imino; the broken line is single or double bond; however, Y is a group other than nitrylo group when X is imino, thioxo, or oxo group).
EXAMPLE: N-(1-Ethyl-2-pyrrolidinyl methyl)-2-methoxy-5-(1-tetrazolyl)benzamide.
USE: Anti-peptic ulcer drugs, psychotropic drugs (Major tranquilizer).
PROCESS: An aminobenzamide of formula II is reacted with sodium azide in the presence of acetic acid and ethyl orthoformate to give the compound of formula I.
COPYRIGHT: (C)1979,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP13769777A JPS5473780A (en) | 1977-11-15 | 1977-11-15 | Novel benzamide derivative |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP13769777A JPS5473780A (en) | 1977-11-15 | 1977-11-15 | Novel benzamide derivative |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5473780A true JPS5473780A (en) | 1979-06-13 |
Family
ID=15204685
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP13769777A Pending JPS5473780A (en) | 1977-11-15 | 1977-11-15 | Novel benzamide derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5473780A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0869118A1 (en) * | 1997-04-04 | 1998-10-07 | Shiseido Company Limited | Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug |
-
1977
- 1977-11-15 JP JP13769777A patent/JPS5473780A/en active Pending
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0869118A1 (en) * | 1997-04-04 | 1998-10-07 | Shiseido Company Limited | Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug |
US5925667A (en) * | 1997-04-04 | 1999-07-20 | Shiseido Co., Ltd. | Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug |
US6043243A (en) * | 1997-04-04 | 2000-03-28 | Shiseido Co., Ltd. | Pyrrolidine derivative, anti-ulcer drug, and antibacterial drug |
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