FI883672A - Menetelmä terapeuttisesti käyttökelpoisten aminoalkoksifenyylijohdannaisten valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisten aminoalkoksifenyylijohdannaisten valmistamiseksi Download PDF

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FI883672A
FI883672A FI883672A FI883672A FI883672A FI 883672 A FI883672 A FI 883672A FI 883672 A FI883672 A FI 883672A FI 883672 A FI883672 A FI 883672A FI 883672 A FI883672 A FI 883672A
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preparation
therapeutically useful
aminoalkoxyphenyl derivatives
aminoalkoxyphenyl
derivatives
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FI883672A
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English (en)
Swedish (sv)
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FI93215C (fi
FI883672A0 (fi
FI93215B (fi
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Jean Gubin
Pierre Chatelain
Henri Inion
Jean Lucchetti
Jean-Marie Mahaux
Jean-Noel Vallat
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Sanofi Sa
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Priority claimed from US07/082,554 external-priority patent/US4957925A/en
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    • C07ORGANIC CHEMISTRY
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    • C07D213/00Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62Oxygen or sulfur atoms
    • C07D213/70Sulfur atoms
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
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    • C07D207/22Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/82Benzo [b] furans; Hydrogenated benzo [b] furans with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
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    • C07D317/48Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
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  • Obesity (AREA)
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  • Neurology (AREA)
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  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Quinoline Compounds (AREA)
  • Indole Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Furan Compounds (AREA)
  • Pyrrole Compounds (AREA)
FI883672A 1987-08-07 1988-08-05 Menetelmä terapeuttisesti käyttökelpoisten aminoalkoksifenyylijohdannaisten valmistamiseksi FI93215C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US8255487 1987-08-07
US07/082,554 US4957925A (en) 1986-02-14 1987-08-07 Aminoalkoxyphenyl derivatives, process of preparation and compositions containing the same

Publications (4)

Publication Number Publication Date
FI883672A0 FI883672A0 (fi) 1988-08-05
FI883672A true FI883672A (fi) 1989-02-08
FI93215B FI93215B (fi) 1994-11-30
FI93215C FI93215C (fi) 1995-03-10

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FI883672A FI93215C (fi) 1987-08-07 1988-08-05 Menetelmä terapeuttisesti käyttökelpoisten aminoalkoksifenyylijohdannaisten valmistamiseksi

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AT (2) ATE113274T1 (fi)
AU (2) AU608873B2 (fi)
CA (2) CA1335379C (fi)
DD (1) DD278792A5 (fi)
DE (2) DE3886298T2 (fi)
DK (2) DK435588A (fi)
ES (1) ES2060667T3 (fi)
FI (1) FI93215C (fi)
HU (1) HU207990B (fi)
IE (1) IE61731B1 (fi)
IL (1) IL87181A (fi)
MA (1) MA21348A1 (fi)
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Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2594438B1 (fr) * 1986-02-14 1990-01-26 Labaz Sanofi Nv Derives d'indolizine, leur procede de preparation ainsi que les compositions en contenant
IL87181A (en) * 1987-08-07 1993-08-18 Sanofi Sa Aminoalkoxyphenyl derivatives, their preparation and pharmaceutical and veterinary compositions containing them
FR2633622B1 (fr) * 1988-07-04 1991-05-17 Sanofi Sa Derives de sulfonyl indolizine, leur procede de preparation et leur utilisation comme intermediaires de synthese
CA2008985A1 (en) * 1989-02-06 1990-08-06 Jean Gubin Aminoalkoxyphenyl derivatives, process of preparation and compositions containing the same
FR2642755B1 (fi) * 1989-02-07 1993-11-05 Sanofi
FR2642756B1 (fr) * 1989-02-07 1994-03-04 Sanofi Derives cycloaminoalkoxyphenyle, leur procede de preparation ainsi que les compositions pharmaceutiques ou veterinaires en contenant
FR2692578B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Derives d'indolizines, procede de preparation et utilisation pour la preparation de composes aminoalkoxybenzenesulfonyl-indolizines a activite pharmaceutique.
FR2692574B1 (fr) * 1992-06-23 1995-06-23 Sanofi Elf Derives hydroxy-4 benzenethio, leur preparation ainsi que leur utilisation pour la preparation de derives aminoalkoxybenzenesulfonyles.
FR2708604B1 (fr) * 1993-07-30 1995-10-20 Sanofi Elf Utilisation de dérivés de benzènesulfonyl-indole pour la préparation de médicaments.
GB9321811D0 (en) * 1993-10-22 1993-12-15 Smithkline Beecham Plc Pharmaceuticals
FR2725133B1 (fr) * 1994-09-30 1996-12-20 Sanofi Sa Composition pharmaceutique de fantofarone pour administration orale
WO1997034876A1 (en) 1996-03-15 1997-09-25 Zeneca Limited Cinnoline derivatives and use as medicine
WO1998010763A1 (en) * 1996-09-13 1998-03-19 Merck & Co., Inc. Thrombin inhibitors
DK1660057T3 (da) 2003-08-27 2012-08-20 Ophthotech Corp Kombinationsterapi til behandling af neovaskulære øjenlidelser
US9006227B2 (en) * 2011-04-19 2015-04-14 Integrative Research Laboratories Sweden Ab Modulators of cortical dopaminergic- and NMDA-receptor-mediated glutamatergic neurotransmission
CA3237199A1 (en) 2021-11-02 2023-05-11 Flare Therapeutics Inc. Pparg inverse agonists and uses thereof

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US3321478A (en) * 1963-09-20 1967-05-23 American Cyanamid Co Aminoethoxyphenyl amine, ether, and sulfide derivatives of pyrimidine
FI61030C (fi) * 1976-02-19 1982-05-10 Sanofi Sa Foerfarande foer framstaellning av terapeutiskt verkande 2-substituerade-1- eller 3-benzoyl-indolizinderivat
US4117128A (en) * 1976-08-03 1978-09-26 Smithkline Corporation Sulfonyl benzofurans and benzothiophenes having coronary vasodilator activity
FR2376145A1 (fr) * 1977-01-03 1978-07-28 Thea Therapeutiques Applic Sa Nouveaux derives de chromones a activite medicamenteuse et leur preparation
GB1560006A (en) * 1977-08-18 1980-01-30 Laroche Navarron Sa Benzoyl furan derivatives process for their preparation and therapeutic applications thereof
AU537816B2 (en) * 1980-07-01 1984-07-12 Ici Australia Limited Cinnolines having herbicidal properties
AU8165582A (en) * 1981-04-02 1982-10-07 Ici Australia Limited Quinolin derivatives
FR2594438B1 (fr) * 1986-02-14 1990-01-26 Labaz Sanofi Nv Derives d'indolizine, leur procede de preparation ainsi que les compositions en contenant
IL87181A (en) * 1987-08-07 1993-08-18 Sanofi Sa Aminoalkoxyphenyl derivatives, their preparation and pharmaceutical and veterinary compositions containing them

Also Published As

Publication number Publication date
DK435588A (da) 1989-02-08
ATE113274T1 (de) 1994-11-15
MA21348A1 (fr) 1989-04-01
ZA885781B (en) 1990-04-25
PL163114B1 (pl) 1994-02-28
ES2060667T3 (es) 1994-12-01
CA1335378C (en) 1995-04-25
AU608873B2 (en) 1991-04-18
RU2032669C1 (ru) 1995-04-10
JPH01104038A (ja) 1989-04-21
AR246250A1 (es) 1994-07-29
EP0302792B1 (en) 1994-10-26
IE61731B1 (en) 1994-11-30
PL160574B1 (pl) 1993-03-31
EP0302792A3 (en) 1990-11-28
OA09013A (en) 1991-03-31
AU620040B2 (en) 1992-02-13
FI93215C (fi) 1995-03-10
YU152188A (en) 1990-04-30
PT88181A (pt) 1989-06-30
DE3886298T2 (de) 1994-06-09
IE882274L (en) 1989-02-07
IL87181A0 (en) 1988-12-30
DK438788D0 (da) 1988-08-05
JPS6470458A (en) 1989-03-15
DK438788A (da) 1989-02-08
NO176142C (no) 1995-02-08
NO176142B (no) 1994-10-31
NO883503L (no) 1989-02-08
SG59866G (en) 1995-09-18
PT88180A (pt) 1989-06-30
HU207990B (en) 1993-07-28
PL274094A1 (en) 1989-05-02
TNSN88080A1 (fr) 1990-07-10
EP0302793A3 (en) 1990-11-28
DD278792A5 (de) 1990-05-16
NO883503D0 (no) 1988-08-05
FI883672A0 (fi) 1988-08-05
DE3886298D1 (de) 1994-01-27
EP0302793B1 (en) 1993-12-15
PT88180B (pt) 1995-03-01
NZ225625A (en) 1990-09-26
AU2024388A (en) 1989-02-09
EP0302792A2 (en) 1989-02-08
FI93215B (fi) 1994-11-30
SG58994G (en) 1994-10-28
HUT48870A (en) 1989-07-28
EP0302793A2 (en) 1989-02-08
MY103905A (en) 1993-10-30
DK435588D0 (da) 1988-08-04
DE3851925D1 (de) 1994-12-01
DE3851925T2 (de) 1995-06-08
ZA885782B (en) 1990-04-25
IL87181A (en) 1993-08-18
RU1819260C (ru) 1993-05-30
PT88181B (pt) 1995-03-01
CA1335379C (en) 1995-04-25
NZ225642A (en) 1990-03-27
ATE98643T1 (de) 1994-01-15
AU2061988A (en) 1989-02-09

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