FI852249L - FOERFARANDE FOER FRAMSTAELLNING AV NYA ISOXAZOLOKINOLINONER. - Google Patents

FOERFARANDE FOER FRAMSTAELLNING AV NYA ISOXAZOLOKINOLINONER.

Info

Publication number
FI852249L
FI852249L FI852249A FI852249A FI852249L FI 852249 L FI852249 L FI 852249L FI 852249 A FI852249 A FI 852249A FI 852249 A FI852249 A FI 852249A FI 852249 L FI852249 L FI 852249L
Authority
FI
Finland
Prior art keywords
carbon atoms
radical containing
isoxazolokinolinoner
nya
alkyl radical
Prior art date
Application number
FI852249A
Other languages
Finnish (fi)
Other versions
FI79322C (en
FI852249A0 (en
FI79322B (en
Inventor
Daniel Humbert
Jean-Claude Gasc
Peter Francis Hunt
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of FI852249A0 publication Critical patent/FI852249A0/en
Publication of FI852249L publication Critical patent/FI852249L/en
Application granted granted Critical
Publication of FI79322B publication Critical patent/FI79322B/en
Publication of FI79322C publication Critical patent/FI79322C/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Lubricants (AREA)
  • Color Television Systems (AREA)
  • Diaphragms For Electromechanical Transducers (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

1. Derivatives of isoxazoloquinolinone characterized in that they answer to the general formula l see diagramm : EP0168309,P8,F1 in which R represents a hydrogen, fluorine, chlorine or bromine atom, a linear alkyl radical containing from 1 to 5 carbon atoms, or branched alkyl radical containing from 3 to 5 carbon atoms, an alkoxy radical containing from 1 to 5 carbon atoms, a nitro or trifluoromethyl radical and R1 represents a phenyl radical possibly substituted by a linear alkyl radical containing from 1 to 5 carbon atoms, or a branched alkyl radical containing from 3 to 5 carbon atoms, by an alkoxy radical containing from 1 to 5 carbon atoms, or by a halogen atom.
FI852249A 1984-06-25 1985-06-05 Process for the preparation of novel therapeutically useful 2-phenyl-ice oxazolo / 4,5-c / quinolin-3-ones FI79322C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8409961 1984-06-25
FR8409961A FR2566407B1 (en) 1984-06-25 1984-06-25 NOVEL ISOXAZOLOQUINOLEIN DERIVATIVES, PROCESS FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS, AND COMPOSITIONS CONTAINING THEM

Publications (4)

Publication Number Publication Date
FI852249A0 FI852249A0 (en) 1985-06-05
FI852249L true FI852249L (en) 1985-12-26
FI79322B FI79322B (en) 1989-08-31
FI79322C FI79322C (en) 1989-12-11

Family

ID=9305387

Family Applications (1)

Application Number Title Priority Date Filing Date
FI852249A FI79322C (en) 1984-06-25 1985-06-05 Process for the preparation of novel therapeutically useful 2-phenyl-ice oxazolo / 4,5-c / quinolin-3-ones

Country Status (17)

Country Link
EP (1) EP0168309B1 (en)
JP (1) JPS6176491A (en)
KR (1) KR860000296A (en)
AT (1) ATE32899T1 (en)
CA (1) CA1225993A (en)
DE (1) DE3561818D1 (en)
DK (1) DK284085A (en)
ES (1) ES8604599A1 (en)
FI (1) FI79322C (en)
FR (1) FR2566407B1 (en)
GR (1) GR851530B (en)
HU (1) HU192234B (en)
IL (1) IL75562A (en)
MA (1) MA20461A1 (en)
NZ (1) NZ212532A (en)
OA (1) OA08045A (en)
PT (1) PT80690B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4920117A (en) * 1989-06-09 1990-04-24 Hoechst-Roussel Pharmaceuticals Inc. 4,5,5a,6-tetrahydro-3H-isoxazolo(5,4,3-kl)acridines, pharmaceutical compositions and use
US5182290A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain oxazoloquinolinones; a new class of GABA brain receptor ligands
IL127559A0 (en) 1996-06-20 1999-10-28 Univ Texas Compounds and methods for providing pharmacologically active preparations and uses thereof

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2537140B1 (en) * 1982-12-07 1986-07-18 Roussel Uclaf NOVEL 4-HYDROXY-3-QUINOLEINE CARBOXAMIDE DERIVATIVES, SALTS THEREOF, PROCESS FOR THEIR PREPARATION, APPLICATION AS MEDICAMENTS, AND COMPOSITIONS CONTAINING THEM

Also Published As

Publication number Publication date
FI79322C (en) 1989-12-11
HUT38948A (en) 1986-07-28
PT80690B (en) 1987-03-31
ES544488A0 (en) 1986-02-01
JPS6176491A (en) 1986-04-18
DE3561818D1 (en) 1988-04-14
FI852249A0 (en) 1985-06-05
FR2566407B1 (en) 1986-09-26
EP0168309B1 (en) 1988-03-09
OA08045A (en) 1987-01-31
HU192234B (en) 1987-05-28
GR851530B (en) 1985-11-25
IL75562A0 (en) 1985-10-31
EP0168309A1 (en) 1986-01-15
FI79322B (en) 1989-08-31
ATE32899T1 (en) 1988-03-15
PT80690A (en) 1985-07-01
KR860000296A (en) 1986-01-27
ES8604599A1 (en) 1986-02-01
CA1225993A (en) 1987-08-25
MA20461A1 (en) 1985-12-31
NZ212532A (en) 1988-08-30
FR2566407A1 (en) 1985-12-27
DK284085A (en) 1985-12-26
DK284085D0 (en) 1985-06-24
IL75562A (en) 1988-07-31

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: ROUSSEL-UCLAF