ES2000187A6 - Un procedimiento para preparar derivados de benzamida - Google Patents

Un procedimiento para preparar derivados de benzamida

Info

Publication number
ES2000187A6
ES2000187A6 ES8600108A ES8600108A ES2000187A6 ES 2000187 A6 ES2000187 A6 ES 2000187A6 ES 8600108 A ES8600108 A ES 8600108A ES 8600108 A ES8600108 A ES 8600108A ES 2000187 A6 ES2000187 A6 ES 2000187A6
Authority
ES
Spain
Prior art keywords
benzamides
hydrogen atom
preparation
alkyl
therapeutical use
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8600108A
Other languages
English (en)
Inventor
Jacqueline Franceschini
Renne Gardaix-Luthereau
Josette Margarit
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Original Assignee
Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe dEtudes Scientifiques et Industrielles de lIle de France SA filed Critical Societe dEtudes Scientifiques et Industrielles de lIle de France SA
Publication of ES2000187A6 publication Critical patent/ES2000187A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/20—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D233/24—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Nutrition Science (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrrole Compounds (AREA)

Abstract

LA PREPARACION DE NUEVOS DERIVADOS DE BENZAMIDA DE FORMULA GENERAL (I): EN LA CUAL R1 REPRESENTA ALQUILO INFERIOR, ALQUENILO INFERIOR O HIDROGENO; R2 REPRESENTA ALQUILO, ALQUENILO INFERIOR, BENCILO, CICLOALQUILALQUILO, CICLOALQUENILALQUILO O HIDROGENO; R3, R4, R5, R6, R7 Y R8 REPRESENTAN ALQUILO INFERIOR O HIDROGENO; Y X REPRESENTA HALOGENO, SE EFECTUA HACIENDO REACCIONAR UN DERIVADO DEL ACIDO P-AMINOBENZOICO CON UN NITRILOAMINADO Y HACIENDO REACCIONAR EL COMPUESTO INTERMEDIO OBTENIDO CON UNA DIAMINA SUSTITUIDA. LOS COMPUESTOS DE FORMULA (I) PUEDEN UTILIZARSE COMO MEDICAMENTOS DE ACCION GASTROMOTORA.
ES8600108A 1985-07-04 1986-07-03 Un procedimiento para preparar derivados de benzamida Expired ES2000187A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8510199A FR2584401B1 (fr) 1985-07-04 1985-07-04 Nouveau benzamide, son procede de preparation et son application dans le domaine therapeutique

Publications (1)

Publication Number Publication Date
ES2000187A6 true ES2000187A6 (es) 1988-01-01

Family

ID=9320954

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8600108A Expired ES2000187A6 (es) 1985-07-04 1986-07-03 Un procedimiento para preparar derivados de benzamida

Country Status (42)

Country Link
US (1) US4703055A (es)
EP (1) EP0210893B1 (es)
JP (1) JPS62103069A (es)
KR (1) KR920007271B1 (es)
CN (1) CN1021441C (es)
AR (1) AR241906A1 (es)
AT (1) ATE57181T1 (es)
AU (1) AU582253B2 (es)
BE (1) BE905018A (es)
BG (1) BG45853A3 (es)
CA (2) CA1276644C (es)
CH (1) CH667873A5 (es)
CS (1) CS274658B2 (es)
DD (1) DD251554A5 (es)
DE (2) DE3620215A1 (es)
DK (2) DK316386A (es)
EG (1) EG18057A (es)
ES (1) ES2000187A6 (es)
FI (1) FI86422C (es)
FR (1) FR2584401B1 (es)
GB (1) GB2178035B (es)
GR (1) GR861714B (es)
HU (1) HU198023B (es)
IE (1) IE58577B1 (es)
IL (1) IL79241A (es)
IN (1) IN163430B (es)
IS (1) IS1374B6 (es)
IT (1) IT1214686B (es)
LU (1) LU86499A1 (es)
MA (1) MA20725A1 (es)
NO (1) NO166124C (es)
NZ (1) NZ216704A (es)
OA (1) OA08355A (es)
PH (2) PH23435A (es)
PL (1) PL147410B1 (es)
PT (1) PT82853B (es)
SU (1) SU1605924A3 (es)
TN (1) TNSN86099A1 (es)
YU (1) YU44790B (es)
ZA (1) ZA864874B (es)
ZM (1) ZM5086A1 (es)
ZW (1) ZW12286A1 (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2057324A1 (en) * 1990-12-18 1992-06-19 Lora Louise Fitch Benzamide and sulfonamide hypoglycemic agents
US5214189A (en) * 1992-06-15 1993-05-25 The United States Of America As Represented By The Secretary Of The Navy N-(2-hydroxyethyl nitrate)-2,4,6,-trinitrobenzamide
US7507727B2 (en) * 2003-04-07 2009-03-24 Cylene Pharmaceuticals, Inc. Substituted quinobenzoxazine analogs and methods of using thereof
AU2006223482A1 (en) * 2005-03-14 2006-09-21 Janssen Pharmaceutica, N.V. Process for the preparation of opioid modulators

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2376424A (en) * 1940-12-23 1945-05-22 Parke Davis & Co Biological product and process of obtaining same
GB1268259A (en) * 1969-11-18 1972-03-29 Beecham Group Ltd Imidazoline derivatives
AT311338B (de) * 1971-03-08 1973-11-12 Malesci Sas Verfahren zum Herstellen eines neuen Imidazolinderivates und seiner Salze
CA1008856A (en) * 1971-11-15 1977-04-19 Ciba-Geigy Ag Triazolo-benzodiazepines
US3885040A (en) * 1973-02-28 1975-05-20 Univ Toledo Methods and benzamide compositions for producing hypotensive activity
GB1513631A (en) * 1976-02-17 1978-06-07 Gallardo Antonio Sa Piperidine derivatives
DK189677A (da) * 1976-05-07 1977-11-08 Sumitomo Chemical Co M-phenoxybenzamid-derivater
FR2415099A1 (fr) * 1978-01-20 1979-08-17 Ile De France Nouveaux derives de 4-amino-5-alkylsulfonyl ortho-anisamides, leurs procedes de preparation et leur application comme psychotropes

Also Published As

Publication number Publication date
PT82853B (pt) 1988-04-21
GR861714B (en) 1986-11-04
YU115086A (en) 1988-02-29
PL147410B1 (en) 1989-05-31
OA08355A (fr) 1988-02-29
DK204891D0 (da) 1991-12-20
IE861796L (en) 1987-01-04
FI862793A (fi) 1987-01-05
MA20725A1 (fr) 1987-04-01
KR920007271B1 (ko) 1992-08-29
CH667873A5 (fr) 1988-11-15
CS274658B2 (en) 1991-09-15
BE905018A (fr) 1987-01-02
HUT42451A (en) 1987-07-28
PH23435A (en) 1989-08-07
DK204891A (da) 1991-12-20
YU44790B (en) 1991-02-28
NO166124C (no) 1991-06-12
JPS62103069A (ja) 1987-05-13
IE58577B1 (en) 1993-10-06
BG45853A3 (en) 1989-08-15
IL79241A0 (en) 1986-09-30
CN1021441C (zh) 1993-06-30
IT1214686B (it) 1990-01-18
GB2178035A (en) 1987-02-04
NO862676D0 (no) 1986-07-02
IS1374B6 (is) 1989-06-30
AU5977986A (en) 1987-01-08
EG18057A (en) 1991-08-30
CN86105682A (zh) 1987-02-04
ZA864874B (en) 1987-02-25
DK316386A (da) 1987-01-05
EP0210893A1 (fr) 1987-02-04
LU86499A1 (fr) 1986-12-02
ATE57181T1 (de) 1990-10-15
KR870001172A (ko) 1987-03-11
FR2584401A1 (fr) 1987-01-09
CA1276644C (fr) 1990-11-20
JPH0586942B2 (es) 1993-12-14
ZM5086A1 (en) 1986-11-28
CA1300162C (fr) 1992-05-05
IT8648189A0 (it) 1986-06-27
SU1605924A3 (ru) 1990-11-07
TNSN86099A1 (fr) 1990-01-01
DD251554A5 (de) 1987-11-18
DE3620215A1 (de) 1987-01-08
DE3674667D1 (de) 1990-11-08
NZ216704A (en) 1990-03-27
EP0210893B1 (fr) 1990-10-03
AR241906A1 (es) 1993-01-29
CS504086A2 (en) 1990-09-12
IS3116A7 (is) 1987-01-05
HU198023B (en) 1989-07-28
GB2178035B (en) 1989-02-08
ZW12286A1 (en) 1986-11-05
IL79241A (en) 1990-04-29
US4703055A (en) 1987-10-27
FR2584401B1 (fr) 1987-11-20
FI86422C (fi) 1992-08-25
IN163430B (es) 1988-09-17
AU582253B2 (en) 1989-03-16
FI862793A0 (fi) 1986-07-01
PH25219A (en) 1991-03-27
PT82853A (fr) 1986-07-01
GB8616287D0 (en) 1986-08-13
DK316386D0 (da) 1986-07-03
NO862676L (no) 1987-01-05
FI86422B (fi) 1992-05-15
NO166124B (no) 1991-02-25

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20000601