EA201301355A1 - Композиция и таблетка, содержащая ралтегравир - Google Patents
Композиция и таблетка, содержащая ралтегравирInfo
- Publication number
- EA201301355A1 EA201301355A1 EA201301355A EA201301355A EA201301355A1 EA 201301355 A1 EA201301355 A1 EA 201301355A1 EA 201301355 A EA201301355 A EA 201301355A EA 201301355 A EA201301355 A EA 201301355A EA 201301355 A1 EA201301355 A1 EA 201301355A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- composition
- tablet containing
- raltegravir
- containing raltegravir
- tablet
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
В заявке описаны композиция и таблетка, содержащая ралтегравир, и способ изготовления такой таблетки.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP11168543.4A EP2529741B1 (en) | 2011-06-01 | 2011-06-01 | Composition and Tablet Comprising Raltegravir |
PCT/EP2012/059991 WO2012163893A1 (en) | 2011-06-01 | 2012-05-29 | Composition and tablet comprising raltegravir |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201301355A1 true EA201301355A1 (ru) | 2014-05-30 |
Family
ID=44188025
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201301355A EA201301355A1 (ru) | 2011-06-01 | 2012-05-29 | Композиция и таблетка, содержащая ралтегравир |
Country Status (7)
Country | Link |
---|---|
US (1) | US20140094478A1 (ru) |
EP (2) | EP2529741B1 (ru) |
CA (1) | CA2837241A1 (ru) |
EA (1) | EA201301355A1 (ru) |
ES (1) | ES2450944T3 (ru) |
IL (1) | IL229206A0 (ru) |
WO (1) | WO2012163893A1 (ru) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2014014933A1 (en) * | 2012-07-20 | 2014-01-23 | Merck Sharp & Dohme Corp. | Hiv treatment with amido-substituted pyrimidinone derivatives |
WO2014064711A2 (en) * | 2012-10-22 | 2014-05-01 | Hetero Research Foundation | Methods of administering raltegravir and raltegravir compositions |
EP4093380A1 (en) * | 2020-01-23 | 2022-11-30 | Lupin Limited | Pharmaceutical compositions of raltegravir |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2003035077A1 (en) | 2001-10-26 | 2003-05-01 | Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa | N-substituted hydroxypyrimidinone carboxamide inhibitors of hiv integrase |
UA87884C2 (ru) | 2004-12-03 | 2009-08-25 | Мерк Энд Ко., Инк. | Безводная кристаллическая калиевая соль ингибитора вич-интегразы |
RU2382648C2 (ru) * | 2004-12-03 | 2010-02-27 | Мерк Энд Ко., Инк. | Фармацевтический состав карбоксамидных ингибиторов интегразы вич, содержащий композицию с контролируемой скоростью высвобождения |
WO2007087188A2 (en) * | 2006-01-20 | 2007-08-02 | Merck & Co., Inc. | Taste-masked tablets and granules |
WO2009079412A2 (en) * | 2007-12-14 | 2009-06-25 | Ardea Biosciences Inc. | Reverse transcriptase inhibitors |
CA2795157C (en) * | 2010-04-01 | 2015-11-24 | Teva Pharmaceutical Industries Ltd. | Raltegravir salts and crystalline forms thereof |
AU2012241050B2 (en) * | 2011-04-06 | 2016-05-19 | Lupin Limited | Novel salts of raltegravir |
-
2011
- 2011-06-01 EP EP11168543.4A patent/EP2529741B1/en not_active Not-in-force
- 2011-06-01 ES ES11168543.4T patent/ES2450944T3/es active Active
-
2012
- 2012-05-29 CA CA2837241A patent/CA2837241A1/en not_active Abandoned
- 2012-05-29 US US14/118,959 patent/US20140094478A1/en not_active Abandoned
- 2012-05-29 EA EA201301355A patent/EA201301355A1/ru unknown
- 2012-05-29 EP EP12726061.0A patent/EP2714044A1/en not_active Withdrawn
- 2012-05-29 WO PCT/EP2012/059991 patent/WO2012163893A1/en active Application Filing
-
2013
- 2013-10-31 IL IL229206A patent/IL229206A0/en unknown
Also Published As
Publication number | Publication date |
---|---|
EP2529741B1 (en) | 2014-02-12 |
US20140094478A1 (en) | 2014-04-03 |
EP2714044A1 (en) | 2014-04-09 |
ES2450944T3 (es) | 2014-03-25 |
WO2012163893A1 (en) | 2012-12-06 |
CA2837241A1 (en) | 2012-12-06 |
IL229206A0 (en) | 2014-01-30 |
EP2529741A1 (en) | 2012-12-05 |
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