EA201001724A1 - Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов - Google Patents

Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов

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Publication number
EA201001724A1
EA201001724A1 EA201001724A EA201001724A EA201001724A1 EA 201001724 A1 EA201001724 A1 EA 201001724A1 EA 201001724 A EA201001724 A EA 201001724A EA 201001724 A EA201001724 A EA 201001724A EA 201001724 A1 EA201001724 A1 EA 201001724A1
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EA
Eurasian Patent Office
Prior art keywords
izoxazole
derivatives
application
metabotropic glutamate
glutamate receptors
Prior art date
Application number
EA201001724A
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English (en)
Other versions
EA018412B1 (ru
Inventor
Джозеф Кассиола
Джеймс Эмпфилд
Джеймс Фолмер
Анджела М. Хантер
Скотт Тронер
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Астразенека Аб
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Application filed by Астразенека Аб filed Critical Астразенека Аб
Publication of EA201001724A1 publication Critical patent/EA201001724A1/ru
Publication of EA018412B1 publication Critical patent/EA018412B1/ru

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Abstract

Соединения формулы I, где R, R, Rи Rявляются такими, как определено в описании, их фармацевтически приемлемые соли, способы их получения, фармацевтические композиции, содержащие их, и способы их применения.
EA201001724A 2008-06-06 2009-06-08 Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов EA018412B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5948508P 2008-06-06 2008-06-06
PCT/SE2009/050682 WO2009148403A1 (en) 2008-06-06 2009-06-08 Isoxazole derivatives and their use as metabotropic glutamate receptor potentiators

Publications (2)

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EA201001724A1 true EA201001724A1 (ru) 2011-08-30
EA018412B1 EA018412B1 (ru) 2013-07-30

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EA201001724A EA018412B1 (ru) 2008-06-06 2009-06-08 Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов
EA201300342A EA201300342A1 (ru) 2008-06-06 2009-06-08 Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов

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EA201300342A EA201300342A1 (ru) 2008-06-06 2009-06-08 Производные изоксазола и их применение в качестве потенциирующих средств для метаботропных глутаматных рецепторов

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