EA201000494A1 - Новые гидрокси-8-гетероарилфенантридины и их применение в качестве ингибиторов pde4 - Google Patents

Новые гидрокси-8-гетероарилфенантридины и их применение в качестве ингибиторов pde4

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Publication number
EA201000494A1
EA201000494A1 EA201000494A EA201000494A EA201000494A1 EA 201000494 A1 EA201000494 A1 EA 201000494A1 EA 201000494 A EA201000494 A EA 201000494A EA 201000494 A EA201000494 A EA 201000494A EA 201000494 A1 EA201000494 A1 EA 201000494A1
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EA
Eurasian Patent Office
Prior art keywords
application
heteroarryfenanthridines
pde4 inhibitors
new hydroxy
hydroxy
Prior art date
Application number
EA201000494A
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English (en)
Other versions
EA017282B1 (ru
Inventor
Беате Шмидт
Дитер Флоккерци
Армин Хатцельманн
Кристоф Цитт
Иоганнес Барзиг
Дегенхард Маркс
Ханс-Петер Клей
Ульрих Каутц
Original Assignee
Никомед Гмбх
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Publication date
Application filed by Никомед Гмбх filed Critical Никомед Гмбх
Publication of EA201000494A1 publication Critical patent/EA201000494A1/ru
Publication of EA017282B1 publication Critical patent/EA017282B1/ru

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Abstract

В заявке описаны соединения формулы (I), в которых Rl, R2, R3, R4, R5 и Har имеют значения, указанные в описании заявки, причем указанные соединения являются эффективными ингибиторами PDE4.
EA201000494A 2004-03-03 2005-03-02 Производное гидрокси-6-гетероарилфенантридина и его применение в качестве ингибитора pde4 EA017282B1 (ru)

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