DOP2002000460A - 2,5-REPLACED DIAMIDOINDOLS AND ITS USE. - Google Patents

2,5-REPLACED DIAMIDOINDOLS AND ITS USE.

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Publication number
DOP2002000460A
DOP2002000460A DO2002000460A DO2002000460A DOP2002000460A DO P2002000460 A DOP2002000460 A DO P2002000460A DO 2002000460 A DO2002000460 A DO 2002000460A DO 2002000460 A DO2002000460 A DO 2002000460A DO P2002000460 A DOP2002000460 A DO P2002000460A
Authority
DO
Dominican Republic
Prior art keywords
disorders
obesity
nitrogen
diseases
disease
Prior art date
Application number
DO2002000460A
Other languages
Spanish (es)
Inventor
Jorg Keldenich
Johannes-Peter Stasch
Michael Brands
Stefan Weigand
Jens-Kerim Erguden
Thomas Krahn
Stephan Siegel
Dirk Heimbach
Christian Schroder
Hanno Wild
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Priority to DO2002000460A priority Critical patent/DOP2002000460A/en
Publication of DOP2002000460A publication Critical patent/DOP2002000460A/en

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Abstract

La presente invención se relaciona con un compuesto de la fórmula (I): (en donde A. B. C y D son independientemente nitrógeno u opcionalmente metino substituido; E es nitrógeno, metino o metino substituido con hidróxi; n es O o 1; T, U, V y W son independientemente nitrógeno u opcionalmente metino substituido; X es -N(S02R4)-, -N(COR5)- o -CO-; ¥ es -C(R6)(R7)-, -O- o -N(R8)-, siempre que el compuesto (I) es excluido cuando E es nitrógeno, n es O, X es -CO-, e Y es -O-) y similares, eI cual es útil como un agente para el tratamiento de varias enfermedades relacionadas con el NPY, por ejemplo. desórdenes cardiovasculares tales como angina. insuficiencia cardiaca aguda o congestiva. infarto miocárdico. hipertensión, nefropatía, anormalidad de electrólitos. vasospasmo. arteriosclerosis, etc.; desórdenes del sistema nervioso central tales corno la bulimia. depresión, ansiedad. acceso, epilepsia, demencia, dolor, alcoholismo, síndrome de abstinencia. desórdenes de Ios ritmos circadianos, esquizofrenia, deterioro de la memoria, desórdenes del sueño. deterioro cognoscitivo, etc.; enfermedades metabólicas tales como la obesidad. diabetes, anormalidades hormonales, hipercolesterolemia, hiperlipidernia, gota, hígado adiposo, etc.; desórdenes genitales o reproductivos tales como Ia infertilidad. parto prematuro, di sfunción sexual, etc., desórdenes gastrointestinales; desórdenes respiratorios, enfermedades inflamatorias o glaucoma y similares, así como también, por ejemplo. ateroesclerosis. hipogonadismo, hiperandrogenismo, síndrome de ovario poliquístico. hirsutismo. desórdenes de la motilidad gastrointestinal, reflujo gastro-esofágeo relacionado con la obesidad, hipoventilación por obesidad (síndrome de Pickwick), apnea del sueño, inflamación, inflamación sistémica de la vasculatura. osteoartritis, resistencia a Ia insulina, broncoconstricción, preferencia por el alcohol, síndrome metabólico. enfermedad de Alzheimer. hipertropia cardiaca, hipertropia del ventrícu1o izquierdo, hipertrigliceridemia, colesterol HDL bajo; desórdenes cardiovasculares tales como enfermedad coronaria del corazón (CHD), enfermedad cerebrovascular, ataque, enfermedad vascular periférica, muerte repentina, enfermedades de la vesícula biliar, cáncer (de pech~o, del endometrio y del colon), sofocación, hiperuricemia, fertilidad daflada, dolor de la espalda baja, o riesgo anestésico aumentado, y similaresThe present invention relates to a compound of the formula (I): (wherein AB C and D are independently nitrogen or optionally substituted methine; E is nitrogen, methine or hydroxy substituted methine; n is O or 1; T, U , V and W are independently nitrogen or optionally substituted methine; X is -N (S02R4) -, -N (COR5) - or -CO-; ¥ is -C (R6) (R7) -, -O- or -N (R8) -, provided that compound (I) is excluded when E is nitrogen, n is O, X is -CO-, and Y is -O-) and the like, which is useful as an agent for the treatment of several diseases related to NPY, for example. cardiovascular disorders such as angina. acute or congestive heart failure. myocardial infarction hypertension, nephropathy, electrolyte abnormality. vasospasm arteriosclerosis, etc .; Central nervous system disorders such as bulimia. depression, anxiety access, epilepsy, dementia, pain, alcoholism, withdrawal symptoms. disorders of circadian rhythms, schizophrenia, memory impairment, sleep disorders. cognitive impairment, etc .; metabolic diseases such as obesity. diabetes, hormonal abnormalities, hypercholesterolemia, hyperlipidernia, gout, adipose liver, etc .; genital or reproductive disorders such as infertility. premature birth, sexual function, etc., gastrointestinal disorders; respiratory disorders, inflammatory diseases or glaucoma and the like, as well as, for example. atherosclerosis hypogonadism, hyperandrogenism, polycystic ovary syndrome. hirsutism gastrointestinal motility disorders, gastro-esophageal reflux related to obesity, hypoventilation due to obesity (Pickwick syndrome), sleep apnea, inflammation, systemic inflammation of the vasculature. osteoarthritis, insulin resistance, bronchoconstriction, preference for alcohol, metabolic syndrome. Alzheimer disease. cardiac hypertropia, left ventricular hypertropia, hypertriglyceridemia, low HDL cholesterol; Cardiovascular disorders such as coronary heart disease (CHD), cerebrovascular disease, attack, peripheral vascular disease, sudden death, gallbladder diseases, cancer (breast, endometrial and colon), suffocation, hyperuricemia, impaired fertility , lower back pain, or increased anesthetic risk, and the like

DO2002000460A 2002-09-04 2002-09-04 2,5-REPLACED DIAMIDOINDOLS AND ITS USE. DOP2002000460A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DO2002000460A DOP2002000460A (en) 2002-09-04 2002-09-04 2,5-REPLACED DIAMIDOINDOLS AND ITS USE.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DO2002000460A DOP2002000460A (en) 2002-09-04 2002-09-04 2,5-REPLACED DIAMIDOINDOLS AND ITS USE.

Publications (1)

Publication Number Publication Date
DOP2002000460A true DOP2002000460A (en) 2003-03-31

Family

ID=44261095

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2002000460A DOP2002000460A (en) 2002-09-04 2002-09-04 2,5-REPLACED DIAMIDOINDOLS AND ITS USE.

Country Status (1)

Country Link
DO (1) DOP2002000460A (en)

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