DK492783D0 - Fremgangsmade til fremstilling af 3-aryl-5-pyrazol-derivater - Google Patents
Fremgangsmade til fremstilling af 3-aryl-5-pyrazol-derivaterInfo
- Publication number
- DK492783D0 DK492783D0 DK4927/83A DK492783A DK492783D0 DK 492783 D0 DK492783 D0 DK 492783D0 DK 4927/83 A DK4927/83 A DK 4927/83A DK 492783 A DK492783 A DK 492783A DK 492783 D0 DK492783 D0 DK 492783D0
- Authority
- DK
- Denmark
- Prior art keywords
- aryl
- preparing
- pyrazole derivatives
- pyrazole
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/16—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Physical Education & Sports Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/437,994 US4495195A (en) | 1982-11-01 | 1982-11-01 | Xanthine oxidase inhibiting 3(5)-phenyl-substituted-5(3)-pyrazole-carboxylic acid derivatives, compositions, and methods of use |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK492783D0 true DK492783D0 (da) | 1983-10-27 |
Family
ID=23738785
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK4927/83A DK492783D0 (da) | 1982-11-01 | 1983-10-27 | Fremgangsmade til fremstilling af 3-aryl-5-pyrazol-derivater |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US4495195A (da) |
| EP (1) | EP0112623A2 (da) |
| JP (1) | JPS5995272A (da) |
| KR (1) | KR840006629A (da) |
| AU (1) | AU2068583A (da) |
| DD (1) | DD210265A5 (da) |
| DK (1) | DK492783D0 (da) |
| ES (1) | ES8601900A1 (da) |
| FI (1) | FI833931A (da) |
| GB (1) | GB2130205A (da) |
| GR (1) | GR79640B (da) |
| IL (1) | IL70075A0 (da) |
| PT (1) | PT77583B (da) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ208555A (en) * | 1983-06-23 | 1987-06-30 | American Cyanamid Co | (3-amino-1h-pyrazol-4-yl)-arylmethanone derivatives |
| IE59813B1 (en) * | 1986-05-09 | 1994-04-06 | Warner Lambert Co | Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxy-genase inhibitors and pharmaceutical compositions containing them |
| JPS6425763A (en) | 1987-04-24 | 1989-01-27 | Mitsubishi Chem Ind | Pyrazoles and insecticide and acaricide containing said pyrazoles as active ingredient |
| US4861777A (en) * | 1987-09-11 | 1989-08-29 | Mitsubishi Kasei Corporation | Pyrazole derivative and insecticidal and miticidal composition containing the derivative as active ingredient |
| JP2751309B2 (ja) * | 1988-02-16 | 1998-05-18 | 三菱化学株式会社 | ピラゾール類およびこれを有効成分とする殺虫、殺ダニ、殺菌剤 |
| JP2784925B2 (ja) * | 1988-09-07 | 1998-08-13 | 日本農薬株式会社 | ３又は５−フェニルピラゾール類又はその塩及び除草剤 |
| US4956379A (en) * | 1990-02-13 | 1990-09-11 | Bristol-Myers Squibb Company | Pyrazole carboxylic acids and esters and inhibition of blood platelet aggregation therewith |
| EP0442448A3 (en) | 1990-02-13 | 1992-08-12 | Bristol-Myers Squibb Company | Heterocyclic carboxylic acids and esters |
| FR2665898B1 (fr) * | 1990-08-20 | 1994-03-11 | Sanofi | Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant. |
| US5294630A (en) * | 1992-07-07 | 1994-03-15 | Eli Lilly And Company | Treatment of inflammatory bowel disease |
| US5436258A (en) * | 1992-09-09 | 1995-07-25 | Eli Lilly And Company | Prevention of bone resorption |
| GB9312853D0 (en) * | 1993-06-22 | 1993-08-04 | Euro Celtique Sa | Chemical compounds |
| US5591776A (en) * | 1994-06-24 | 1997-01-07 | Euro-Celtique, S.A. | Pheynl or benzyl-substituted rolipram-based compounds for and method of inhibiting phosphodiesterase IV |
| HRP950330A2 (en) * | 1994-07-05 | 1997-10-31 | Ciba Geigy Ag | New herbicides |
| US6025361A (en) * | 1994-12-13 | 2000-02-15 | Euro-Celtique, S.A. | Trisubstituted thioxanthines |
| WO1996018399A1 (en) * | 1994-12-13 | 1996-06-20 | Euro-Celtique, S.A. | Aryl thioxanthines |
| JP2001523213A (ja) * | 1994-12-13 | 2001-11-20 | ユーロ−セルティーク，エス．エイ． | 三置換チオキサンチン類 |
| US6166041A (en) * | 1995-10-11 | 2000-12-26 | Euro-Celtique, S.A. | 2-heteroaryl and 2-heterocyclic benzoxazoles as PDE IV inhibitors for the treatment of asthma |
| US6075016A (en) * | 1996-04-10 | 2000-06-13 | Euro-Celtique S.A. | 6,5-fused aromatic ring systems having enhanced phosphodiesterase IV inhibitory activity |
| ID21775A (id) * | 1996-10-25 | 1999-07-22 | Yoshitomi Pharmaceutical | Senyawa-senyawa 1-fenilpirazol dan penggunaan farmasinya |
| US5723608A (en) * | 1996-12-31 | 1998-03-03 | Neurogen Corporation | 3-aryl substituted pyrazolo 4,3-d!pyrimidine derivatives; corticotropin-releasing factor receptor (CRF1) specific ligands |
| WO1999024038A1 (en) | 1997-11-07 | 1999-05-20 | Johns Hopkins University | Methods for treatment of disorders of cardiac contractility |
| MX2007002160A (es) * | 2004-08-27 | 2007-05-10 | Astellas Pharma Inc | Derivado de 2-fenilpiridina. |
| US7612108B2 (en) * | 2004-08-27 | 2009-11-03 | Astellas Pharma Inc. | 2-phenylthiophene derivative |
| DE602006018635D1 (de) | 2005-10-07 | 2011-01-13 | Astellas Pharma Inc | Triarylcarbonsäurederivat |
| KR20080097456A (ko) | 2006-02-24 | 2008-11-05 | 아스텔라스세이야쿠 가부시키가이샤 | 소화관 궤양의 치료제 또는 예방제 |
| AU2010218748B2 (en) | 2009-02-27 | 2015-03-26 | Teijin Limited | Process for producing phenyl-substituted heterocyclic derivative through coupling using transition metal catalyst |
| JP5654601B2 (ja) | 2010-08-27 | 2015-01-14 | 帝人ファーマ株式会社 | パラジウム化合物を用いたカップリング法によるフェニル置換複素環誘導体の製造法 |
| NO2980085T3 (da) | 2013-03-29 | 2018-08-11 | ||
| EP2944635B1 (en) * | 2014-05-15 | 2018-11-28 | Council of Scientific & Industrial Research | Pyrazole linked benzimidazole conjugates and a process for preparation thereof |
| CN106632245B (zh) * | 2016-09-30 | 2019-11-15 | 华南理工大学 | 氮取代基苯基吡唑类黄嘌呤氧化还原酶抑制剂及制备与应用 |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1261124B (de) * | 1961-09-22 | 1968-02-15 | Hoechst Ag | Verfahren zur Herstellung von Pyrazolen |
| IT1053661B (it) * | 1966-09-27 | 1981-10-10 | Farmacosmici S P A | Ammidi dell acido 3 5 metil 5 3 pirazol carbossilico |
| FR2104931B1 (da) * | 1970-09-08 | 1975-01-10 | Ferlux | |
| DE2508934A1 (de) * | 1974-03-04 | 1975-09-11 | Byk Gulden Lomberg Chem Fab | Neue substituierte 5-amino-4- formyl-carbamoyl-pyrazole, verfahren zu ihrer herstellung und sie enthaltende arzneimittel |
| DE2410653A1 (de) * | 1974-03-06 | 1975-10-30 | Byk Gulden Lomberg Chem Fab | Neue heterocyclisch substituierte 5amino-4-formylcarbamoyl-pyrazole, verfahren zu ihrer herstellung und sie enthaltende arzneimittel |
| US3899508A (en) * | 1974-04-12 | 1975-08-12 | Lilly Co Eli | 5-(2-Aminophenyl)pyrazole-3-carboxylic acids and esters thereof |
| US3903106A (en) * | 1974-04-12 | 1975-09-02 | Lilly Co Eli | Pyrazole-3-carboxylic acids |
| US3895027A (en) * | 1974-04-12 | 1975-07-15 | Lilly Co Eli | Process for preparing pyrazole-3-carboxylic acids |
| FR2320093A1 (fr) * | 1975-08-05 | 1977-03-04 | Sogeras | Nouveaux acides diphenyl-pyrazole-5-acetiques |
| FR2353292A1 (fr) * | 1975-08-05 | 1977-12-30 | Sogeras | Nouveaux derives du benzoyl-3 pyrazole |
| US4134987A (en) * | 1976-01-14 | 1979-01-16 | Huppatz John L | Compounds and compositions |
| US4214090A (en) * | 1976-01-14 | 1980-07-22 | Commonwealth Scientific And Industrial Research Organization | Fungicidal carboxamidopyrazoles |
| US4245106A (en) * | 1979-07-05 | 1981-01-13 | Monsanto Company | Process for the preparation of 1-alkyl-3-aryl-4-pyrazolecarboxylates |
| US4346097A (en) * | 1980-09-30 | 1982-08-24 | Warner-Lambert Company | Method for treating convulsions with pyrazole-4-carboxamide derivatives |
-
1982
- 1982-11-01 US US06/437,994 patent/US4495195A/en not_active Expired - Fee Related
-
1983
- 1983-10-26 GR GR72796A patent/GR79640B/el unknown
- 1983-10-27 IL IL70075A patent/IL70075A0/xx unknown
- 1983-10-27 DK DK4927/83A patent/DK492783D0/da not_active Application Discontinuation
- 1983-10-27 FI FI833931A patent/FI833931A/fi not_active Application Discontinuation
- 1983-10-27 EP EP83306530A patent/EP0112623A2/en not_active Withdrawn
- 1983-10-27 GB GB08328755A patent/GB2130205A/en not_active Withdrawn
- 1983-10-28 DD DD83256094A patent/DD210265A5/de unknown
- 1983-10-28 JP JP58203575A patent/JPS5995272A/ja active Pending
- 1983-10-28 PT PT77583A patent/PT77583B/pt unknown
- 1983-10-28 AU AU20685/83A patent/AU2068583A/en not_active Abandoned
- 1983-10-28 KR KR1019830005109A patent/KR840006629A/ko not_active IP Right Cessation
- 1983-10-28 ES ES526869A patent/ES8601900A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES526869A0 (es) | 1985-05-01 |
| PT77583A (en) | 1983-11-01 |
| IL70075A0 (en) | 1984-01-31 |
| US4495195A (en) | 1985-01-22 |
| DD210265A5 (de) | 1984-06-06 |
| EP0112623A2 (en) | 1984-07-04 |
| GB2130205A (en) | 1984-05-31 |
| FI833931A0 (fi) | 1983-10-27 |
| GR79640B (da) | 1984-10-31 |
| ES8601900A1 (es) | 1985-05-01 |
| FI833931A (fi) | 1984-05-02 |
| GB8328755D0 (en) | 1983-11-30 |
| KR840006629A (ko) | 1984-12-01 |
| JPS5995272A (ja) | 1984-06-01 |
| PT77583B (en) | 1986-05-27 |
| AU2068583A (en) | 1984-05-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK470583D0 (da) | Fremgangsmade til fremstilling af 1-phenyl-2-piperidinopropanolderivater | |
| DK492783D0 (da) | Fremgangsmade til fremstilling af 3-aryl-5-pyrazol-derivater | |
| DK95483D0 (da) | Fremgangsmade til fremstilling af tetrahydropyranderivater | |
| DK280182A (da) | Fremgangsmaade til fremstilling af n-aryl-piperazinalkanamider | |
| DK183583D0 (da) | Fremgangsmade til fremstilling af benzoazacycloalkyl-spiro-imidazolidiner | |
| DK210083D0 (da) | Fremgangsmade til fremstilling af 6a,10a-trans-hexahydrodibenzopyranoner | |
| DK262782A (da) | Fremgangsmaade til fremstilling af n-dihydrothiazolyl-3-quinolincarboxamidderivater | |
| DK153583A (da) | Fremgangsmaade til fremstilling af substituerede penemderivater | |
| DK370582A (da) | Fremgangsmaade til fremstilling af 2-beta-d-ribofuranosylthiazol-4-carboxamid | |
| DK159309C (da) | Fremgangsmaade til fremstilling af 4-metyl-5-alkylthiometyl-imidazoler | |
| DK271183D0 (da) | Fremgangsmade til fremstilling af dihydropyridinderivater | |
| DK115581A (da) | Fremgangsmaade til fremstilling af pyrimidylquinazoliner | |
| DK40883D0 (da) | Fremgangsmade til fremstilling af benzothienylallylaminer | |
| DK188881A (da) | Fremgangsmaade til fremstilling af 2-guanidinthiazol-derivater | |
| DK71783D0 (da) | Fremgangsmade til fremstilling af pyrimidonderivater | |
| DK449881A (da) | Fremgangsmaade til fremstilling af moroxydinphenoxyisobutyrater | |
| DK399783A (da) | Fremgangsmaade til fremstilling af substituerede 1-pyridyloxy-3-indolylalkylamino-2-propanoler | |
| DK518883A (da) | Fremgangsmaade til fremstilling af 1-oxa-beta-lactam-forbindelser | |
| DK457983D0 (da) | Fremgangsmade til fremstilling af beta-lactam | |
| DK454183D0 (da) | Fremgangsmade til fremstilling af 15-cycloaliphatiske derivater af 13,14-didehydro-carboprostancycliner | |
| DK63583D0 (da) | Fremgangsmade til fremstilling af dihydropyridinderivater | |
| DK432683D0 (da) | Fremgangsmade til fremstilling af 2-hydroxy-2-phenylethylaminer | |
| DK156061C (da) | Fremgangsmaade til fremstilling af 2-alkyl-4-amino-5-aminomethylpyrimidin | |
| DK400481A (da) | Fremgangsmaade til fremstilling af 4-carbamoyloxy-oxazaphosporiner | |
| DK493384D0 (da) | Fremgangsmaade til fremstilling af bis-dioxopiperazin-derivater |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHS | Application shelved for other reasons than non-payment |