DK161147C - Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater - Google Patents

Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater

Info

Publication number: DK161147C
Authority: DK; Denmark
Prior art keywords: undiverives; oe3haa; tetrazin; daa; imidazo
Prior art date: 1981-08-24

Application number

DK377882A

Other languages

English (en)

Other versions

DK161147B (da

DK377882A (da

Inventor

Edward Lunt

Malcolm Francis Graham Stevens

Robert Stone

Kenneth Robert Harr Wooldridge

Original Assignee

May & Baker Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-08-24

Filing date

1982-08-23

Publication date

1991-11-18

1982-08-23 Application filed by May & Baker Ltd filed Critical May & Baker Ltd

1983-02-25 Publication of DK377882A publication Critical patent/DK377882A/da

1991-06-03 Publication of DK161147B publication Critical patent/DK161147B/da

1991-11-18 Application granted granted Critical

1991-11-18 Publication of DK161147C publication Critical patent/DK161147C/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Hematology (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK377882A 1981-08-24 1982-08-23 Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater DK161147C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8125791		1981-08-24
GB8125791		1981-08-24

Publications (3)

Publication Number	Publication Date
DK377882A DK377882A (da)	1983-02-25
DK161147B DK161147B (da)	1991-06-03
DK161147C true DK161147C (da)	1991-11-18

Family

ID=10524141

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK377882A DK161147C (da)	1981-08-24	1982-08-23	Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater

Country Status (29)

Country	Link
JP (1)	JPS5843975A (da)
KR (1)	KR890000094B1 (da)
AT (1)	AT380256B (da)
AU (1)	AU571430B2 (da)
BE (1)	BE894175A (da)
CA (1)	CA1197247A (da)
CH (1)	CH655114A5 (da)
DE (2)	DE19975037I2 (da)
DK (1)	DK161147C (da)
ES (1)	ES8400438A1 (da)
FI (1)	FI73434C (da)
FR (1)	FR2511679A1 (da)
GB (1)	GB2104522B (da)
GE (1)	GEP19960641B (da)
GR (1)	GR76863B (da)
HU (1)	HU186107B (da)
IE (1)	IE53408B1 (da)
IL (1)	IL66606A (da)
IT (1)	IT1152505B (da)
LT (1)	LT2436B (da)
LU (1)	LU84347A1 (da)
LV (2)	LV5511A3 (da)
NL (2)	NL192739C (da)
NZ (1)	NZ201668A (da)
OA (1)	OA07174A (da)
SE (1)	SE448543B (da)
SU (1)	SU1447284A3 (da)
UA (1)	UA5971A1 (da)
ZA (1)	ZA826120B (da)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5260291A (en) *	1981-08-24	1993-11-09	Cancer Research Campaign Technology Limited	Tetrazine derivatives
GB2125402B (en) *	1982-08-17	1985-11-13	May & Baker Ltd	New tetrazine derivatives
FR2531958B1 (fr) *	1982-08-17	1986-10-31	May & Baker Ltd	Nouveaux derive
US4517182A (en) *	1983-05-24	1985-05-14	Warner-Lambert Company	3-(Haloethyl)-4-oxopyrazolo-[5,1-d]-1,2,3,5-tetrazine-8-carboxamide composition
GB8616125D0 (en) *	1986-07-02	1986-08-06	May & Baker Ltd	Compositions of matter
AU622330B2 (en) *	1989-06-23	1992-04-02	Takeda Chemical Industries Ltd.	Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
EP2275425A1 (en) *	2003-12-30	2011-01-19	Chemagis Ltd.	Novel crystalline forms of temozolomide
ES2552338T3 (es)	2005-01-21	2015-11-27	Astex Therapeutics Limited	Compuestos farmacéuticos
PE20080695A1 (es)	2006-04-27	2008-06-28	Banyu Pharma Co Ltd	Derivados de dihidropirazolopirimidinona como inhibidores de quinasa weel
JP2008081492A (ja)	2006-08-31	2008-04-10	Banyu Pharmaceut Co Ltd	オーロラａ選択的阻害作用を有する新規アミノピリジン誘導体
WO2008044045A1 (en)	2006-10-12	2008-04-17	Astex Therapeutics Limited	Pharmaceutical combinations
JP5528806B2 (ja)	2006-10-12	2014-06-25	アステックス、セラピューティックス、リミテッド	複合薬剤
AU2008315048A1 (en)	2007-10-23	2009-04-30	Msd K.K.	Pyridone-substituted-dihydropyrazolopyrimidinone derivative
PE20091101A1 (es) *	2007-12-18	2009-07-26	Pharminox Ltd	AMIDAS DE ACIDO 3-SUBSTITUIDO-4-OXO-3,4-DIHIDRO-IMIDAZO[5,1-d] [1,2,3,5-TETRACINA-8-CARBOXILICO Y SU EMPLEO
WO2010058430A1 (en) *	2008-11-24	2010-05-27	Reliance Life Sciences Pvt. Ltd.	Process for the preparation of tetrazine derivatives
US8481503B2 (en)	2009-03-06	2013-07-09	Merck Sharp & Dohme Corp.	Combination cancer therapy with an AKT inhibitor and other anticancer agents
EP2445915B1 (en)	2009-06-23	2016-04-20	Pharminox Limited	3-substituted-8-substituted-3h imidazo[5,1-d][1,2,3,5-tetrazin-4-one compounds and their use
RU2462466C1 (ru) *	2011-06-24	2012-09-27	Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан"	Замещенные азоло[1,2,4,5]тетразины - ингибиторы актинобактериальных серин-треониновых протеинкиназ
US20140271657A1 (en)	2011-10-12	2014-09-18	Children's Medical Center Corporation	Combinatorial compositions and methods of treating hemoglobinopathies
SG11201807965YA (en)	2016-03-15	2018-10-30	Oryzon Genomics Sa	Combinations of lsd1 inhibitors for use in the treatment of solid tumors
KR101847342B1 (ko) *	2017-05-08	2018-04-11	(주)센텍코리아	웨어러블 체지방 연소량 측정기

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2932305A1 (de) *	1979-08-09	1981-02-26	Basf Ag	Azolo- eckige klammer auf 5,1-d eckige klammer zu - eckige klammer auf 1,2,3,5 eckige klammer zu -tetrazin-4-one und verfahren zur herstellung dieser verbindungen

1982
- 1982-08-05 OA OA57766BISD patent/OA07174A/xx unknown
- 1982-08-12 IL IL66606A patent/IL66606A/xx not_active IP Right Cessation
- 1982-08-23 LU LU84347A patent/LU84347A1/fr unknown
- 1982-08-23 CA CA000409950A patent/CA1197247A/fr not_active Expired
- 1982-08-23 GB GB08224155A patent/GB2104522B/en not_active Expired
- 1982-08-23 IT IT22938/82A patent/IT1152505B/it active Protection Beyond IP Right Term
- 1982-08-23 DE DE1999175037 patent/DE19975037I2/de active Active
- 1982-08-23 SE SE8204817A patent/SE448543B/sv not_active IP Right Cessation
- 1982-08-23 FR FR8214461A patent/FR2511679A1/fr active Granted
- 1982-08-23 AU AU87493/82A patent/AU571430B2/en not_active Expired
- 1982-08-23 FI FI822921A patent/FI73434C/fi not_active IP Right Cessation
- 1982-08-23 ES ES515176A patent/ES8400438A1/es not_active Expired
- 1982-08-23 NL NL8203286A patent/NL192739C/nl not_active IP Right Cessation
- 1982-08-23 BE BE0/208860A patent/BE894175A/fr not_active IP Right Cessation
- 1982-08-23 KR KR8203774A patent/KR890000094B1/ko active
- 1982-08-23 ZA ZA826120A patent/ZA826120B/xx unknown
- 1982-08-23 SU SU823482389A patent/SU1447284A3/ru active
- 1982-08-23 CH CH5007/82A patent/CH655114A5/fr not_active IP Right Cessation
- 1982-08-23 AT AT0319182A patent/AT380256B/de not_active IP Right Cessation
- 1982-08-23 JP JP57144902A patent/JPS5843975A/ja active Granted
- 1982-08-23 HU HU822708A patent/HU186107B/hu unknown
- 1982-08-23 DE DE19823231255 patent/DE3231255A1/de active Granted
- 1982-08-23 IE IE2026/82A patent/IE53408B1/en not_active IP Right Cessation
- 1982-08-23 NZ NZ201668A patent/NZ201668A/en unknown
- 1982-08-23 GR GR69093A patent/GR76863B/el unknown
- 1982-08-23 UA UA3482389A patent/UA5971A1/uk unknown
- 1982-08-23 DK DK377882A patent/DK161147C/da not_active IP Right Cessation
1993
- 1993-06-19 LV LV930621A patent/LV5511A3/xx unknown
- 1993-09-29 LT LTRP1286A patent/LT2436B/xx not_active IP Right Cessation
- 1993-11-16 GE GEAP19931653A patent/GEP19960641B/en unknown
- 1993-12-03 LV LV931303A patent/LV5621A3/xx unknown
1999
- 1999-04-01 NL NL990010C patent/NL990010I2/nl unknown

Also Published As

Publication number	Publication date
ZA826120B (en)	1983-07-27
NL8203286A (nl)	1983-03-16
HU186107B (en)	1985-06-28
FR2511679A1 (fr)	1983-02-25
DK161147B (da)	1991-06-03
IT1152505B (it)	1987-01-07
DE3231255A1 (de)	1983-03-03
ES515176A0 (es)	1983-11-01
FI73434B (fi)	1987-06-30
NL990010I2 (nl)	1999-09-01
LT2436B (lt)	1994-02-15
CH655114A5 (fr)	1986-03-27
CA1197247A (fr)	1985-11-26
NL192739B (nl)	1997-09-01
GEP19960641B (en)	1996-11-15
NZ201668A (en)	1985-08-16
IE822026L (en)	1983-02-24
ES8400438A1 (es)	1983-11-01
SE8204817L (sv)	1983-02-25
SU1447284A3 (ru)	1988-12-23
FI822921A0 (fi)	1982-08-23
GR76863B (da)	1984-09-04
ATA319182A (de)	1985-09-15
FI73434C (fi)	1987-10-09
AU571430B2 (en)	1988-04-21
FR2511679B1 (da)	1985-02-01
LU84347A1 (fr)	1983-06-07
IL66606A0 (en)	1982-12-31
KR840001175A (ko)	1984-03-28
LV5511A3 (lv)	1994-03-10
BE894175A (fr)	1983-02-23
GB2104522B (en)	1985-06-12
LV5621A3 (lv)	1994-05-10
FI822921L (fi)	1983-02-25
NL192739C (nl)	1998-01-06
AU8749382A (en)	1983-03-03
AT380256B (de)	1986-05-12
NL990010I1 (nl)	1999-07-01
DE19975037I2 (de)	2001-06-13
KR890000094B1 (ko)	1989-03-07
IT8222938A0 (it)	1982-08-23
GB2104522A (en)	1983-03-09
IE53408B1 (en)	1988-11-09
SE448543B (sv)	1987-03-02
DK377882A (da)	1983-02-25
DE3231255C2 (da)	1992-02-27
JPS5843975A (ja)	1983-03-14
IL66606A (en)	1987-07-31
JPH045029B2 (da)	1992-01-30
OA07174A (fr)	1984-04-30
UA5971A1 (uk)	1994-12-29
SE8204817D0 (sv)	1982-08-23

Legal Events

Date	Code	Title	Description
1999-08-16	CTFF	Application for supplementary protection certificate (spc) filed	Free format text: CA 1999 00012, 19990511, EXPIRES: 20070823
2002-09-09	PUP	Patent expired

Publication	Publication Date	Title
DK159442C (da)	1991-03-18	Analogifremgangsmaade til fremstilling af 6,7-substitueret-4-ethyl-quinazoliner
DK162389C (da)	1992-03-09	Analogifremgangsmaade til fremstilling af 2-oe4-oe(4,4-dialkyl-2,6-piperidindion-1-yl)butylaa-1-piperazinylaapyrimidiner
DK162601C (da)	1992-05-11	Analogifremgangsmaade til fremstilling af 8-oe4-oe4-(2,1-benzisothiazol-3-yl)-1-piperazinylaabutylaa-8-azaspirooe4.5aadecan-7,9-dion
DK528982A (da)	1983-05-28	Fremgangsmaade til fremstilling af 13,14-didehydro-prostaglandiner
DK149949C (da)	1987-06-15	Analogifremgangsmaade til fremstilling af n-aryl-piperazinalkanamider
DK219382A (da)	1982-11-19	Fremgangsmaade til fremstilling af 1,2-diaminocyclobuten-3,4-dioner
DK260682A (da)	1982-12-13	Fremgangsmaade til fremstilling af partikelformige geler
DK151341C (da)	1988-05-09	Analogifremgangsmaade til fremstilling af d-phenylalanyl-l-prolyl-l-argininaldehydsulfat
DK65882A (da)	1982-08-18	Fremgangsmaade til fremstilling af substituerede phosphonamider
DK161147C (da)	1991-11-18	Analogifremgangsmaade til fremstilling af oe3haa-imidazo-oe5,1-daa-1,2,3,5-tetrazin-4-onderivater
DK149846C (da)	1987-06-29	Analogifremgangsmaade til fremstilling af n,n'-bis-tetrahydro-isoquinolyldisulfonylimider
DK153282A (da)	1982-10-07	Fremgangsmaade til fremstilling af bismethinisoindoliner
DK155281C (da)	1989-07-24	Fremgangsmaade til fremstilling af 1,2-dihydro-6-methyl-2-oxo-5-(pyridinyl)nicotinonitriler
DK239382A (da)	1982-11-29	Fremgangsmaade til fremstilling af anthracyclinglycosider
DK152132C (da)	1988-06-20	Analogifremgangsmaade til fremstilling af derivater af 5,6,7,7a-tetrahydro-4h-thienooe3,2-caapyridin-2-on
DK157855C (da)	1990-07-30	Fremgangsmaade til fremstilling af 2,3-dichlor-5-trichlormethylpyridin
DK305982A (da)	1983-01-09	Fremgangsmaade til fremstilling af amidobenzamider
DK162581A (da)	1981-10-12	Fr&mgangsmaade til fremstilling af substituerede 1,4-dihydropyridiner
DK159158C (da)	1991-03-11	Fremgangsmaade til fremstilling af penicillanoyloxy-methylpenicillanat-1,1,1',1'-tetraoxid
DK151256C (da)	1988-06-06	Analogifremgangsmaade til fremstilling af alkylendioxybenzenderivater
DK113483D0 (da)	1983-03-08	Fremgangsmade til fremstilling af 3,4-diphenyl-5-methylpyrazolderivater
DK158740C (da)	1990-11-19	Analogifremgangsmaade til fremstilling af 1,3-propandioletheren af antibiotikum x-14868a
DK156219C (da)	1989-12-04	Analogifremgangsmaade til fremstilling af spirothiazolidinylpiperazinderivater
DK146067C (da)	1983-11-14	Analogifremgangsmaade til fremstilling af 2,4-diamino-5-phenoxypropoxypyrimidiner
DK157873C (da)	1990-08-06	Analogifremgangsmaade til fremstilling af azinorifamycin-forbindelser