DK134984B - Analogifremgangsmåde til fremstilling af alfa-alkylaminopropiophenoner eller syreadditionssalte heraf. - Google Patents

Analogifremgangsmåde til fremstilling af alfa-alkylaminopropiophenoner eller syreadditionssalte heraf.

Info

Publication number
DK134984B
DK134984B DK617070AA DK617070A DK134984B DK 134984 B DK134984 B DK 134984B DK 617070A A DK617070A A DK 617070AA DK 617070 A DK617070 A DK 617070A DK 134984 B DK134984 B DK 134984B
Authority
DK
Denmark
Prior art keywords
alkylaminopropiophenones
alpha
preparation
acid addition
addition salts
Prior art date
Application number
DK617070AA
Other languages
English (en)
Other versions
DK134984C (da
Inventor
Nariman Bomanshaw Mehta
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=10483336&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK134984(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wellcome Found filed Critical Wellcome Found
Priority to DK193076A priority Critical patent/DK193076A/da
Publication of DK134984B publication Critical patent/DK134984B/da
Application granted granted Critical
Publication of DK134984C publication Critical patent/DK134984C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
    • C07C225/02—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C225/14—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated
    • C07C225/16—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being unsaturated and containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C07C49/807—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen all halogen atoms bound to the ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/004—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reaction with organometalhalides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK617070AA 1969-12-04 1970-12-03 Analogifremgangsmåde til fremstilling af alfa-alkylaminopropiophenoner eller syreadditionssalte heraf. DK134984B (da)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DK193076A DK193076A (da) 1969-12-04 1976-04-29 M-halogen-alfa-chlorpropiophenon, blandt andet til anvendelse som mellemprodukt til fremstilling af alfa-alkylaminopropiophenoner

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB5923169 1969-12-04

Publications (2)

Publication Number Publication Date
DK134984B true DK134984B (da) 1977-02-21
DK134984C DK134984C (da) 1977-07-11

Family

ID=10483336

Family Applications (1)

Application Number Title Priority Date Filing Date
DK617070AA DK134984B (da) 1969-12-04 1970-12-03 Analogifremgangsmåde til fremstilling af alfa-alkylaminopropiophenoner eller syreadditionssalte heraf.

Country Status (29)

Country Link
US (1) US3819706A (da)
JP (1) JPS4825179B1 (da)
AR (2) AR192302A1 (da)
AT (2) AT302276B (da)
BE (1) BE759838A (da)
CA (1) CA977777A (da)
CH (2) CH574907A5 (da)
CS (1) CS172338B2 (da)
DE (2) DE2059618C3 (da)
DK (1) DK134984B (da)
EG (1) EG10507A (da)
ES (1) ES386127A1 (da)
FI (1) FI53813C (da)
FR (1) FR2081326B1 (da)
HK (1) HK78476A (da)
IE (1) IE34788B1 (da)
IL (1) IL35781A (da)
IT (1) IT8047948A0 (da)
MT (1) MTP680B (da)
MY (1) MY7700107A (da)
NL (1) NL172148C (da)
NO (1) NO131127C (da)
PH (1) PH9351A (da)
PL (1) PL74637B1 (da)
RO (1) RO57979A (da)
SE (1) SE377933B (da)
YU (1) YU34269B (da)
ZA (1) ZA708179B (da)
ZM (1) ZM14070A1 (da)

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HK78476A (en) 1976-12-17
NL7017687A (da) 1971-06-08
IL35781A0 (en) 1971-02-25
RO57979A (da) 1975-03-15
PL74637B1 (da) 1974-12-31
FI53813B (fi) 1978-05-02
MTP680B (en) 1971-09-11
AT307389B (de) 1973-05-25
CS172338B2 (da) 1976-12-29
SE377933B (da) 1975-08-04
IE34788L (en) 1971-06-04
NO131127C (da) 1975-04-09
DE2059618B2 (de) 1980-07-10
FR2081326B1 (da) 1974-08-30
ES386127A1 (es) 1973-12-16
DE2064934A1 (de) 1971-10-21
YU34269B (en) 1979-04-30
NL172148C (nl) 1983-07-18
IT8047948A0 (it) 1980-02-19
ZA708179B (en) 1972-07-26
DK134984C (da) 1977-07-11
IL35781A (en) 1973-06-29
FR2081326A1 (da) 1971-12-03
BE759838A (fr) 1971-06-03
PH9351A (en) 1975-10-06
JPS4825179B1 (da) 1973-07-26
DE2059618A1 (de) 1971-10-07
MY7700107A (en) 1977-12-31
AT302276B (de) 1972-10-10
CH574907A5 (da) 1976-04-30
YU294570A (en) 1978-10-31
FI53813C (fi) 1978-08-10
US3819706A (en) 1974-06-25
NL172148B (nl) 1983-02-16
CH569693A5 (da) 1975-11-28
EG10507A (en) 1976-03-31
NO131127B (da) 1974-12-30
CA977777A (en) 1975-11-11
IE34788B1 (en) 1975-08-20
AR192302A1 (es) 1973-02-14
DE2059618C3 (de) 1981-04-16
AR198945A1 (es) 1974-07-31
ZM14070A1 (en) 1972-08-21

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