DE602008006209D1 - 1-(4-(4-benzylbenzamid)-benzyl)-azetidin-3-carboxylsäurederivate und entsprechende verbindungen als s1p-rezeptor-modulatoren zur behandlung von immunerkrankungen - Google Patents

1-(4-(4-benzylbenzamid)-benzyl)-azetidin-3-carboxylsäurederivate und entsprechende verbindungen als s1p-rezeptor-modulatoren zur behandlung von immunerkrankungen

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Publication number
DE602008006209D1
DE602008006209D1 DE602008006209T DE602008006209T DE602008006209D1 DE 602008006209 D1 DE602008006209 D1 DE 602008006209D1 DE 602008006209 T DE602008006209 T DE 602008006209T DE 602008006209 T DE602008006209 T DE 602008006209T DE 602008006209 D1 DE602008006209 D1 DE 602008006209D1
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Germany
Prior art keywords
benzylbenzamid
azetidine
benzyl
treatment
carboxylic acid
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DE602008006209T
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English (en)
Inventor
Susana C Neira
Xiang Yu
Roland Burli
Brian Lanman
Victor Cee
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Amgen Inc
Epix Pharmaceuticals Inc
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Amgen Inc
Epix Pharmaceuticals Inc
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Application filed by Amgen Inc, Epix Pharmaceuticals Inc filed Critical Amgen Inc
Publication of DE602008006209D1 publication Critical patent/DE602008006209D1/de
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    • C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
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    • C07D401/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing aromatic rings

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DE602008006209T 2007-09-20 2008-09-19 1-(4-(4-benzylbenzamid)-benzyl)-azetidin-3-carboxylsäurederivate und entsprechende verbindungen als s1p-rezeptor-modulatoren zur behandlung von immunerkrankungen Active DE602008006209D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US99481207P 2007-09-20 2007-09-20
PCT/US2008/010887 WO2009038759A2 (en) 2007-09-20 2008-09-19 1-(4-(benzylbenzamid0) -benzyl) azetidine-3-carboxylic acid derivatives and related compounds as slp receptor modulators for the treatment of immune disorders

Publications (1)

Publication Number Publication Date
DE602008006209D1 true DE602008006209D1 (de) 2011-05-26

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DE602008006209T Active DE602008006209D1 (de) 2007-09-20 2008-09-19 1-(4-(4-benzylbenzamid)-benzyl)-azetidin-3-carboxylsäurederivate und entsprechende verbindungen als s1p-rezeptor-modulatoren zur behandlung von immunerkrankungen

Country Status (10)

Country Link
US (2) US8080542B2 (de)
EP (1) EP2188252B1 (de)
JP (1) JP2010540438A (de)
AT (1) ATE505454T1 (de)
AU (1) AU2008302746B2 (de)
CA (1) CA2699417A1 (de)
DE (1) DE602008006209D1 (de)
ES (1) ES2360929T3 (de)
MX (1) MX2010002885A (de)
WO (1) WO2009038759A2 (de)

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JP2010540438A (ja) 2010-12-24
WO2009038759A2 (en) 2009-03-26
US20120088749A1 (en) 2012-04-12
AU2008302746A1 (en) 2009-03-26
ATE505454T1 (de) 2011-04-15
WO2009038759A3 (en) 2009-07-23
EP2188252B1 (de) 2011-04-13
US8080542B2 (en) 2011-12-20
ES2360929T3 (es) 2011-06-10
MX2010002885A (es) 2010-04-01
CA2699417A1 (en) 2009-03-26
EP2188252A2 (de) 2010-05-26
AU2008302746B2 (en) 2014-07-03
US20090082331A1 (en) 2009-03-26

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