BR0311479A - Derivados de tiofeno antelmìnticos e inseticidas - Google Patents

Derivados de tiofeno antelmìnticos e inseticidas

Info

Publication number
BR0311479A
BR0311479A BR0311479-1A BR0311479A BR0311479A BR 0311479 A BR0311479 A BR 0311479A BR 0311479 A BR0311479 A BR 0311479A BR 0311479 A BR0311479 A BR 0311479A
Authority
BR
Brazil
Prior art keywords
thiophene derivatives
anthelmintic
insecticidal
derivatives
thiophene
Prior art date
Application number
BR0311479-1A
Other languages
English (en)
Inventor
Byung H Lee
Timothy G Geary
John P Davis
Original Assignee
Pharmacia & Upjohn Co Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia & Upjohn Co Llc filed Critical Pharmacia & Upjohn Co Llc
Publication of BR0311479A publication Critical patent/BR0311479A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A61P33/12—Schistosomicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62—Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/78—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
    • C07D333/80—Seven-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

"DERIVADOS DE TIOFENO ANTELMìNTICOS E INSETICIDAS". Descreve-se composições antelmíticas inusitadas que contêm derivados de tiofeno como ingredientes ativos.
BR0311479-1A 2002-05-31 2003-05-28 Derivados de tiofeno antelmìnticos e inseticidas BR0311479A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38501702P 2002-05-31 2002-05-31
PCT/US2003/016701 WO2003101979A1 (en) 2002-05-31 2003-05-28 Anthelmintic and insecticidal thiophene derivatives

Publications (1)

Publication Number Publication Date
BR0311479A true BR0311479A (pt) 2005-02-22

Family

ID=29712123

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0311479-1A BR0311479A (pt) 2002-05-31 2003-05-28 Derivados de tiofeno antelmìnticos e inseticidas

Country Status (10)

Country Link
US (1) US20040014740A1 (pt)
EP (1) EP1509514A1 (pt)
JP (1) JP2005538056A (pt)
AR (1) AR040123A1 (pt)
AU (1) AU2003234657A1 (pt)
BR (1) BR0311479A (pt)
CA (1) CA2487666A1 (pt)
MX (1) MXPA04011122A (pt)
PL (1) PL374201A1 (pt)
WO (1) WO2003101979A1 (pt)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ540161A (en) * 2002-10-30 2008-03-28 Vertex Pharma Compositions useful as inhibitors of rock and other protein kinases
US20050085531A1 (en) * 2003-10-03 2005-04-21 Hodge Carl N. Thiophene-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof
WO2009035818A1 (en) 2007-09-10 2009-03-19 Calcimedica, Inc. Compounds that modulate intracellular calcium
EP2280952B1 (en) 2008-05-05 2012-06-27 Merck Patent GmbH Thienopyridone derivatives as amp-activated protein kinase (ampk) activators
CN102256969A (zh) * 2008-08-27 2011-11-23 钙医学公司 调节胞内钙的化合物
US8524763B2 (en) 2008-09-22 2013-09-03 Calcimedica, Inc. Inhibitors of store operated calcium release
US8618307B2 (en) 2009-09-16 2013-12-31 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9079891B2 (en) 2010-08-27 2015-07-14 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9512116B2 (en) 2012-10-12 2016-12-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2023101556A1 (en) 2021-12-02 2023-06-08 Rijksuniversiteit Groningen Novel inhibitors of aspartate transcarbamoylase (atcase) and compositions, methods and uses related thereto.

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6414013B1 (en) * 2000-06-19 2002-07-02 Pharmacia & Upjohn S.P.A. Thiophene compounds, process for preparing the same, and pharmaceutical compositions containing the same background of the invention

Also Published As

Publication number Publication date
US20040014740A1 (en) 2004-01-22
WO2003101979A1 (en) 2003-12-11
CA2487666A1 (en) 2003-12-11
AU2003234657A1 (en) 2003-12-19
AR040123A1 (es) 2005-03-16
JP2005538056A (ja) 2005-12-15
PL374201A1 (en) 2005-10-03
MXPA04011122A (es) 2005-07-14
EP1509514A1 (en) 2005-03-02

Similar Documents

Publication Publication Date Title
BR0209057A (pt) Composições herbicidas contendo benzoilciclohexanodionas e protetores
HRP20080564T3 (en) Dihydrotetrabenazines and pharmaceutical compositions containing them
CY1111800T1 (el) Συνδυασμοι δραστικων ουσιων με νηματοδοκτονες, εντομοκτονες και μυκητοκτονες ιδιοτητες με βαση τριφθοροβουτενυλικες ενωσεις
BR0212921A (pt) Composição farmacêutica com base em fondant
CR7864A (es) Piridodiacinas como fungicidas de plantas
CU22869A3 (es) 1-aril-pirazoles plaguicidas
UY24553A1 (es) Compuestos insecticidas de tipo 5- amino -4-etilsulfinil-pirazol
ATE404057T1 (de) Insektenabweisende zusammensetzungen mit verzögerter freisetzung
HRP20050510A2 (en) Microbicide substances
BRPI0518395A2 (pt) inseticidas
GT200000001A (es) Derivados de eter propargilico novedosos.
ECSP066860A (es) Formulaciones de matriz oral que comprenden licarbazepina
BR0111678A (pt) Composições medicinais contendo derivados de propenona
BR0311479A (pt) Derivados de tiofeno antelmìnticos e inseticidas
CO5221025A1 (es) 4-trifluorometil-3-oxazolilpiridinas, procedimiento para su preparacion, agentes que las contienen y su uso como agente para la lucha contra organismos daninos
AR019304A1 (es) Mezclas herbicidas a base de aclonifen y clomazona.
TR200301650T4 (tr) Ziraat ve bahçecilikte kullanım için okzim O-eter bileşikleri ve fungusitler
ITMI20031714A1 (it) Formazioni ad azione antitumorale.
CU23309B7 (es) Compuestos anã logos de astrobilurinas y su uso como acaricida e insecticida
TW200509794A (en) Novel anthelmintic and insecticidal compositions
TR199901374T2 (xx) B�cek �ld�r�c� ve mitisidal kompozisyonlar
ES2183709B1 (es) Composicion para el control de artropodos.
AR034097A1 (es) Composiciones y metodos para reprimir insectos que deterioran cultivos de arroz y otros
BRPI0417106A (pt) granulos de pesticida com surfactante melhorado de soltura rápida
BR0311245B1 (pt) Composição inseticida compreendendo fosfonatos e seus derivados como realçadores da atividade de inseticidas

Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 4A,5A,6A E 7A ANUIDADES

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO PUBLICADO NA RPI 2064 DE 27/07/2010.