AU2003264910A1 - Process for selective alkylation of macrolide and azalide derivatives - Google Patents

Process for selective alkylation of macrolide and azalide derivatives

Info

Publication number
AU2003264910A1
AU2003264910A1 AU2003264910A AU2003264910A AU2003264910A1 AU 2003264910 A1 AU2003264910 A1 AU 2003264910A1 AU 2003264910 A AU2003264910 A AU 2003264910A AU 2003264910 A AU2003264910 A AU 2003264910A AU 2003264910 A1 AU2003264910 A1 AU 2003264910A1
Authority
AU
Australia
Prior art keywords
macrolide
selective alkylation
azalide derivatives
azalide
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2003264910A
Inventor
Marko Derek
Davor Kidemet
Marija Leljak
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fidelta doo
Original Assignee
Pliva Istrazivacki Institut doo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pliva Istrazivacki Institut doo filed Critical Pliva Istrazivacki Institut doo
Publication of AU2003264910A1 publication Critical patent/AU2003264910A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU2003264910A 2003-05-30 2003-09-04 Process for selective alkylation of macrolide and azalide derivatives Abandoned AU2003264910A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US47434803P 2003-05-30 2003-05-30
US60/474,348 2003-05-30
PCT/HR2003/000048 WO2004106353A1 (en) 2003-05-30 2003-09-04 Process for selective alkylation of macrolide and azalide derivatives

Publications (1)

Publication Number Publication Date
AU2003264910A1 true AU2003264910A1 (en) 2005-01-21

Family

ID=33490713

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2003264910A Abandoned AU2003264910A1 (en) 2003-05-30 2003-09-04 Process for selective alkylation of macrolide and azalide derivatives

Country Status (3)

Country Link
CN (1) CN100381453C (en)
AU (1) AU2003264910A1 (en)
WO (1) WO2004106353A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103923142B (en) * 2014-04-30 2017-01-11 浙江震元制药有限公司 Preparation method of roxithromycin intermediate
CN105801642B (en) * 2016-03-11 2019-03-26 北京理工大学 A method of preparing the bis--O- erythromycin A of 6,11-
EP3583099A1 (en) * 2017-02-14 2019-12-25 Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. Cyclization processes of hydroxyalkenoic aicds and products thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI9011409A (en) * 1990-07-18 1995-10-31 Pliva Pharm & Chem Works O-methyl azitromycin derivates, methods and intermediates for their preparation and methods for preparation of pharmaceuticals products which comprise them
ES2279242T3 (en) * 1997-10-16 2007-08-16 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. NEW 3,6-HEMICETALS OF THE CLASS OF 9A-AZALIDAS.

Also Published As

Publication number Publication date
WO2004106353A1 (en) 2004-12-09
CN1798755A (en) 2006-07-05
CN100381453C (en) 2008-04-16

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase