AU1624992A - Amino acid azetidinyl substituted pyridone derivatives, their preparation and their application as medications - Google Patents

Amino acid azetidinyl substituted pyridone derivatives, their preparation and their application as medications

Info

Publication number
AU1624992A
AU1624992A AU16249/92A AU1624992A AU1624992A AU 1624992 A AU1624992 A AU 1624992A AU 16249/92 A AU16249/92 A AU 16249/92A AU 1624992 A AU1624992 A AU 1624992A AU 1624992 A AU1624992 A AU 1624992A
Authority
AU
Australia
Prior art keywords
medications
preparation
amino acid
application
pyridone derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
AU16249/92A
Other versions
AU660311B2 (en
Inventor
Jordi Frigola Constansa
Jordi Corbera-Arjona
Juan Pares Corominas
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Esteve Pharmaceuticals SA
Original Assignee
Laboratorios del Dr Esteve SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratorios del Dr Esteve SA filed Critical Laboratorios del Dr Esteve SA
Publication of AU1624992A publication Critical patent/AU1624992A/en
Application granted granted Critical
Publication of AU660311B2 publication Critical patent/AU660311B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
  • Peptides Or Proteins (AREA)
AU16249/92A 1991-05-16 1992-05-14 Amino acid azetidinyl substituted pyridone derivatives, their preparation and their application as medications Ceased AU660311B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9105937A FR2676445B1 (en) 1991-05-16 1991-05-16 SUBSTITUTED PYRIDONE AMINO ACID AZETIDINYL DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS.
FR9105937 1991-05-16

Publications (2)

Publication Number Publication Date
AU1624992A true AU1624992A (en) 1992-11-19
AU660311B2 AU660311B2 (en) 1995-06-22

Family

ID=9412841

Family Applications (1)

Application Number Title Priority Date Filing Date
AU16249/92A Ceased AU660311B2 (en) 1991-05-16 1992-05-14 Amino acid azetidinyl substituted pyridone derivatives, their preparation and their application as medications

Country Status (20)

Country Link
EP (1) EP0514268A1 (en)
JP (1) JPH05132479A (en)
KR (1) KR920021528A (en)
CN (1) CN1066656A (en)
AU (1) AU660311B2 (en)
CA (1) CA2068853A1 (en)
CZ (1) CZ147992A3 (en)
ES (1) ES2039192B1 (en)
FI (1) FI922225A (en)
FR (1) FR2676445B1 (en)
HU (1) HUT61304A (en)
IL (1) IL101886A0 (en)
IS (1) IS3862A (en)
MA (1) MA22526A1 (en)
MX (1) MX9202273A (en)
NO (1) NO921908L (en)
NZ (1) NZ242733A (en)
OA (1) OA09794A (en)
PL (1) PL294561A1 (en)
ZA (1) ZA923538B (en)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100488284B1 (en) 1996-07-12 2005-05-11 다이이찌 세이야꾸 가부시기가이샤 cis-Substituted aminocyclopropane derivatives and an antimicrobial agent containing the same
KR100613690B1 (en) * 2004-07-30 2006-08-21 한국화학연구원 4-quinolinone derivative and fungicidal composition for agriculture and horticulture comprising same
KR100613688B1 (en) * 2004-08-30 2006-08-21 한국화학연구원 2-amino-4-quinolinone derivative and fungicidal composition for agriculture and horticulture comprising same
EP1814575A4 (en) 2004-11-24 2010-07-07 Neopro Labs Llc Methods and compositions for treating conditions
WO2007112453A2 (en) 2006-03-28 2007-10-04 Neopro Labs, Llc Methods amd compositions for treating conditions
WO2008144675A1 (en) 2007-05-17 2008-11-27 Neopro Labs, Llc Crystalline and amorphous forms of peptide
CN101898990B (en) * 2009-06-01 2012-12-19 中国科学院化学研究所 Method for catalyzing and synthesizing chirality azetidine amide and carboxylic acid compound by microorganism system
US12036286B2 (en) 2021-03-18 2024-07-16 Seagen Inc. Selective drug release from internalized conjugates of biologically active compounds

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5746986A (en) * 1980-09-02 1982-03-17 Dai Ichi Seiyaku Co Ltd Pyrido(1,2,3-de)(1,4)benzoxazine derivative
IE55898B1 (en) * 1982-09-09 1991-02-14 Warner Lambert Co Antibacterial agents
DE3306771A1 (en) * 1983-02-25 1984-08-30 Bayer Ag, 5090 Leverkusen CHINOLONIC CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM
JPH0665676B2 (en) * 1984-04-26 1994-08-24 アボツト ラボラトリーズ Quinoline-benoxazine antibacterial compounds
US4617308A (en) * 1985-01-25 1986-10-14 Warner-Lambert Company 7-substituted amino-1-aryl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids and derivatives thereof as antibacterial agents
US4851418A (en) * 1987-08-21 1989-07-25 Warner-Lambert Company Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
FR2634483B2 (en) * 1987-12-29 1994-03-04 Esteve Labor Dr DERIVATIVES OF ACIDS 7- (1-AZETIDINYL) -1,4-DIHYDRO-4-OXOQUINOLEINE-3-CARBOXYLIQUES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS
IL91648A (en) * 1988-09-22 1997-03-18 Abbott Lab Amino acid quinoline and naphthyridine derivatives, their preparation and pharmaceutical compositions containing them
FI901201A0 (en) * 1989-03-13 1990-03-09 Bristol Myers Squibb Co ANTIBAKTERIELLA 5-SUBSTITUERADE 1,4-DIHYDRO-4-OXONAFTYRIDIN-3-CARBOXYLATDERIVAT OCH DERAS FRAMSTAELLNING.
NO177302C (en) * 1989-03-16 1995-08-23 Esteve Labor Dr Analogous Process for Preparing Therapeutically Active Substituted Azetidinyl Quinolone (Naphthyridone) Carboxylic Acid Derivatives
FR2645862B1 (en) * 1989-04-18 1991-07-12 Esteve Labor Dr SUBSTITUTED ISOTHIAZOLO-PYRYDONE AZETIDINYL DERIVATIVES, THEIR PREPARATION AND THEIR APPLICATION AS MEDICAMENTS
FR2649100B1 (en) * 1989-06-29 1994-03-04 Laboratorios Dr Esteve Sa NOVEL AZETIDINES, THEIR PREPARATION AND THEIR APPLICATION AS INTERMEDIATES FOR THE PREPARATION OF COMPOUNDS WITH ANTIMICROBIAL ACTIVITY

Also Published As

Publication number Publication date
EP0514268A1 (en) 1992-11-19
KR920021528A (en) 1992-12-18
FI922225A (en) 1992-11-17
FR2676445A1 (en) 1992-11-20
HUT61304A (en) 1992-12-28
OA09794A (en) 1994-04-15
MA22526A1 (en) 1992-12-31
CA2068853A1 (en) 1992-11-17
PL294561A1 (en) 1993-05-04
NO921908L (en) 1992-11-17
CZ147992A3 (en) 1993-09-15
IS3862A (en) 1992-11-17
ES2039192B1 (en) 1994-04-01
MX9202273A (en) 1993-05-01
NO921908D0 (en) 1992-05-14
AU660311B2 (en) 1995-06-22
HU9201621D0 (en) 1992-08-28
FI922225A0 (en) 1992-05-15
ES2039192A1 (en) 1993-09-01
CN1066656A (en) 1992-12-02
IL101886A0 (en) 1992-12-30
ZA923538B (en) 1993-01-27
NZ242733A (en) 1994-06-27
JPH05132479A (en) 1993-05-28
FR2676445B1 (en) 1995-02-03

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