AR113688A1 - Proceso para la preparación de compuestos de piridiminio ópticamente activo - Google Patents
Proceso para la preparación de compuestos de piridiminio ópticamente activoInfo
- Publication number
- AR113688A1 AR113688A1 ARP180101083A ARP180101083A AR113688A1 AR 113688 A1 AR113688 A1 AR 113688A1 AR P180101083 A ARP180101083 A AR P180101083A AR P180101083 A ARP180101083 A AR P180101083A AR 113688 A1 AR113688 A1 AR 113688A1
- Authority
- AR
- Argentina
- Prior art keywords
- compounds
- optically active
- pyridiminium
- preparation
- unsubstituted
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 2
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000006656 (C2-C4) alkenyl group Chemical group 0.000 abstract 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 150000001721 carbon Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- -1 pyrimidinium compound Chemical class 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
- C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
- C07F15/0033—Iridium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
- C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
- C07F15/0046—Ruthenium compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F15/00—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table
- C07F15/0006—Compounds containing elements of Groups 8, 9, 10 or 18 of the Periodic Table compounds of the platinum group
- C07F15/0073—Rhodium compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Abstract
Un proceso para preparar un compuesto de pirimidinio ópticamente activo de la fórmula (1) y sus intermediarios, en donde: C* es un átomo de carbono asimétrico de configuración S o R; R¹ es C₁₋₄-alquilo, C₃₋₆-cicloalquilo, C₂₋₄-alquenilo o -CH₂-fenilo, en donde los grupos son no sustituidos o sustituidos con halógeno o C₁₋₄-alquilo; R² es un anillo carbocíclico o heterocíclico saturado, parcialmente insaturado o aromático de 5 ó 6 miembros, en donde el anillo es no sustituido o sustituido con R²ᵃ; Het se selecciona de los compuestos de fórmula (2), (3) y (4).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP17168354 | 2017-04-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR113688A1 true AR113688A1 (es) | 2020-06-03 |
Family
ID=58638745
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP180101083A AR113688A1 (es) | 2017-04-27 | 2018-04-26 | Proceso para la preparación de compuestos de piridiminio ópticamente activo |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US11124528B2 (es) |
| EP (1) | EP3615543B1 (es) |
| JP (1) | JP7263250B2 (es) |
| KR (1) | KR102591738B1 (es) |
| CN (1) | CN110546153B (es) |
| AR (1) | AR113688A1 (es) |
| AU (1) | AU2018260180B2 (es) |
| CA (1) | CA3058083A1 (es) |
| IL (1) | IL270134B (es) |
| MX (1) | MX2019012815A (es) |
| PH (1) | PH12019502286A1 (es) |
| WO (1) | WO2018197541A1 (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2019011785A (es) * | 2017-03-31 | 2019-11-18 | Basf Se | Proceso para preparar compuestos de 2,3-dihidrotiazolo[3,2-a]pirim idin-4-io quirales. |
| CN110621677B (zh) | 2017-05-03 | 2022-06-07 | 巴斯夫欧洲公司 | 制备手性2,3-二氢噻唑并[3,2-a]嘧啶-4-鎓化合物的方法 |
| WO2018234202A1 (en) | 2017-06-19 | 2018-12-27 | Basf Se | SUBSTITUTED PYRIMIDINIUM COMPOUNDS AND DERIVATIVES FOR CONTROLLING HARMFUL ANIMALS |
| US11358922B2 (en) | 2017-11-02 | 2022-06-14 | Basf Se | Process for preparing 4-chlorobenzyl propargyl ether |
| CN110041365B (zh) * | 2018-12-05 | 2020-12-22 | 华东师范大学 | 吡咯啉类手性双膦配体及其制备方法和应用 |
| US11187127B2 (en) | 2019-06-28 | 2021-11-30 | Deere & Company | Exhaust gas treatment system and method with four-way catalyzed filter element |
| US20240051929A1 (en) * | 2019-10-04 | 2024-02-15 | Basf Se | Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone |
| EP4081037A1 (en) * | 2019-12-23 | 2022-11-02 | Basf Se | Enzyme enhanced root uptake of agrochemical active compound |
| EP3974417A1 (en) | 2020-09-29 | 2022-03-30 | Basf Se | Preparation of 2-chloro-1-(2-chlorothiazol-5-yl)ethanone |
| EP4032878A1 (en) | 2021-01-22 | 2022-07-27 | Basf Se | Method for preparing 2-[2-(2-chlorothiazol-5-yl)-2-oxo-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one |
| EP4032886A1 (en) | 2021-01-22 | 2022-07-27 | Basf Se | Method for preparing an enantiomerically enriched form of 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one |
| EP4032894A1 (en) | 2021-01-22 | 2022-07-27 | Basf Se | Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate |
| EP4032893A1 (en) | 2021-01-22 | 2022-07-27 | Basf Se | Method for preparing an enantiomerically enriched form of 3-(2-chlorothiazol-5-yl)-8-methyl-7-oxo-6-phenyl-2,3-dihydrothiazolo[3,2-a]pyrimidin-4-ium-5-olate |
| EP4063362A1 (en) | 2021-03-25 | 2022-09-28 | Basf Se | Method for preparing enantiomerically enriched 2-[2-(2-chlorothiazol-5-yl)-2-hydroxy-ethyl]sulfanyl-6-hydroxy-3-methyl-5-phenyl-pyrimidin-4-one by hydrogenation of the 2-oxo derivative in the presence of a chiral transition metal catalyst |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9019095D0 (en) * | 1990-09-01 | 1990-10-17 | Beecham Group Plc | Novel compounds |
| UA107804C2 (en) * | 2009-08-05 | 2015-02-25 | Du Pont | Mixtures of pesticides mezoionnyh |
| MX2012001646A (es) * | 2009-08-05 | 2012-03-21 | Du Pont | Pesticidas mesoionicos. |
| JP6067733B2 (ja) * | 2011-11-21 | 2017-01-25 | ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ | Ｎ置換１ｈ−ピラゾール−５−カルボキシラート化合物及びその誘導体を製造する方法 |
| JP6389830B2 (ja) | 2013-03-01 | 2018-09-12 | アムジエン・インコーポレーテツド | ベータ−セクレターゼ阻害剤としてのパーフルオロ化５，６−ジヒドロ−４ｈ−１，３−オキサジン−２−アミン化合物および使用方法 |
| AR096022A1 (es) | 2013-04-11 | 2015-12-02 | Basf Se | Compuestos de pirimidinio sustituido, útiles para combatir plagas de animales |
| US10149477B2 (en) * | 2014-10-06 | 2018-12-11 | Basf Se | Substituted pyrimidinium compounds for combating animal pests |
| CN110621677B (zh) * | 2017-05-03 | 2022-06-07 | 巴斯夫欧洲公司 | 制备手性2,3-二氢噻唑并[3,2-a]嘧啶-4-鎓化合物的方法 |
-
2018
- 2018-04-25 JP JP2019557819A patent/JP7263250B2/ja active Active
- 2018-04-25 KR KR1020197034153A patent/KR102591738B1/ko active IP Right Grant
- 2018-04-25 CA CA3058083A patent/CA3058083A1/en active Pending
- 2018-04-25 EP EP18718479.1A patent/EP3615543B1/en active Active
- 2018-04-25 CN CN201880027777.3A patent/CN110546153B/zh active Active
- 2018-04-25 AU AU2018260180A patent/AU2018260180B2/en active Active
- 2018-04-25 US US16/608,290 patent/US11124528B2/en active Active
- 2018-04-25 MX MX2019012815A patent/MX2019012815A/es unknown
- 2018-04-25 WO PCT/EP2018/060555 patent/WO2018197541A1/en unknown
- 2018-04-26 AR ARP180101083A patent/AR113688A1/es unknown
-
2019
- 2019-10-03 PH PH12019502286A patent/PH12019502286A1/en unknown
- 2019-10-24 IL IL270134A patent/IL270134B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20190141711A (ko) | 2019-12-24 |
| JP7263250B2 (ja) | 2023-04-24 |
| AU2018260180B2 (en) | 2021-12-09 |
| KR102591738B1 (ko) | 2023-10-19 |
| MX2019012815A (es) | 2020-01-14 |
| EP3615543B1 (en) | 2021-10-20 |
| US20200055872A1 (en) | 2020-02-20 |
| IL270134B (en) | 2022-05-01 |
| PH12019502286A1 (en) | 2020-09-14 |
| BR112019021122A2 (pt) | 2020-05-12 |
| JP2020517684A (ja) | 2020-06-18 |
| CA3058083A1 (en) | 2018-11-01 |
| WO2018197541A1 (en) | 2018-11-01 |
| EP3615543A1 (en) | 2020-03-04 |
| AU2018260180A1 (en) | 2019-10-31 |
| US11124528B2 (en) | 2021-09-21 |
| CN110546153B (zh) | 2022-09-06 |
| CN110546153A (zh) | 2019-12-06 |
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