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TAK1 Biochemical Assay (1mM ATP) from US Patent US20240279233: "MACROCYCLIC TAK1 INHIBITORS"
Assay data:48 Active, 48 Activity ≤ 1 µM, 48 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
TAK1 Biochemical Assay (100uM ATP) from US Patent US20240279233: "MACROCYCLIC TAK1 INHIBITORS"
Assay data:120 Active, 6 Activity ≤ 1 nM, 120 Activity ≤ 1 µM, 120 Tested
5-HT2 Receptor Assays from US Patent US20240279226: "ERGOLINE-DERIVED AGONISTS OF THE 5-HT2A RECEPTOR"
Assay data:5 Active, 1 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Surface Plasmon Resonance (SPR) SOS1 Binding Assay from US Patent US20240279221: "HETEROCYCLIC COMPOUNDS AND METHODS OF USE"
Assay data:64 Active, 64 Activity ≤ 1 µM, 64 Tested
SOS1-KRas(G12C) FRET Assay from US Patent US20240279221: "HETEROCYCLIC COMPOUNDS AND METHODS OF USE"
Assay data:133 Active, 120 Activity ≤ 1 µM, 136 Tested
Binding Assay from US Patent US20240279218: "ISOXAZOLYL ETHER DERIVATIVES AS GABA A ALPHA5 PAM"
Assay data:194 Active, 3 Activity ≤ 1 nM, 194 Activity ≤ 1 µM, 194 Tested
NMN Fluorescence Biochemical Assay from US Patent US20240279215: "NAMPT MODULATORS"
Assay data:229 Active, 14 Activity ≤ 1 µM, 468 Tested
TBD from US Patent US20240279201: "DUAL WNT SIGNALING PATHWAY INHIBITORS AND AMPK ACTIVATORS FOR TREATMENTS OF DISEASE"
Assay data:51 Active, 9 Activity ≤ 1 nM, 115 Activity ≤ 1 µM, 115 Tested
Enzymatic Assay for KpLpxH Inhibition from US Patent US20240279174: "ANTIBIOTICS COMPRISING LPXH-TARGETING COMPOUNDS AND METHODS OF MAKING AND USING THE SAME"
Assay data:26 Active, 1 Activity ≤ 1 nM, 24 Activity ≤ 1 µM, 26 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibition Activity from US Patent US20240277852: "INHIBITORS AND DEGRADERS OF PIP4K PROTEIN"
Assay data:19 Active, 1 Activity ≤ 1 nM, 18 Activity ≤ 1 µM, 19 Tested
Acetyltransferase Biochemical Assay from US Patent US20240277683: "COMPOUNDS"
Assay data:77 Active, 41 Activity ≤ 1 µM, 125 Tested
Cell Viability Test from US Patent US12065447: "Heterocyclic amide for inhibiting RIP1 kinase and uses thereof"
Assay data:26 Active, 19 Activity ≤ 1 nM, 26 Activity ≤ 1 µM, 26 Tested
BTK kinase lanthascreen binding assay from US Patent US12065446: "Inhibitors of Bruton's tyrosine kinase and method of their use"
Assay data:375 Active, 400 Activity ≤ 1 µM, 416 Tested
Myofibril Assays from US Patent US12065436: "Cardiac sarcomere inhibitors"
Assay data:486 Active, 52 Activity ≤ 1 µM, 696 Tested
Evaluation of Inhibitory Activity of Compounds on KRAS G12C Nucleotide (GDP-GTP) Exchange Reaction from US Patent US12065430: "Indazole compound or salt thereof"
Assay data:120 Active, 109 Activity ≤ 1 µM, 123 Tested
Ki Estimation from US Patent US12065407: "Dual acting FKBP12 and FKBP52 inhibitors"
Assay data:31 Active, 15 Activity ≤ 1 µM, 43 Tested
Intracellular Ca2+ Mobilization Assay (FLIPR) from US Patent US12065399: "Arylsulfonamide derivatives"
Assay data:52 Active, 12 Activity ≤ 1 µM, 59 Tested
TBD from US Patent US12064420: "Tie-2 activators targeting the Schlemm's canal"
Assay data:97 Active, 32 Activity ≤ 1 nM, 95 Activity ≤ 1 µM, 97 Tested
MTase-Glo Methyl Transferase Assay from US Patent US20240262835: "PRMT5 INHIBITING COMPOUNDS AND USES THEREOF"
Assay data:26 Active, 26 Activity ≤ 1 µM, 26 Tested
PRMT5/MEP50 HotSpot Methyltransferase Assay from US Patent US20240262835: "PRMT5 INHIBITING COMPOUNDS AND USES THEREOF"
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
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