| CYP3A4 inhibitor |
| Clotrimazole (JP18/USP/INN) <JP/US> |
| Cimetidine |
| Cimetidine (JP18/USP/INN) <JP/US> |
| Cimetidine hydrochloride (USP) <US> |
| Omeprazole, clarithromycin and amoxicillin <US> |
| Amoxicillin hydrate, clarithromycin and lansoprazole <US> |
| Rabeprazole, amoxicillin and clarithromycin <JP> |
| Vonoprazan, amoxicillin and clarithromycin <JP> |
| Aprepitant |
| Aprepitant (JAN/USP/INN) <JP/US> |
| Fosaprepitant (INN) |
| Fosaprepitant dimeglumine (USAN); Fosaprepitant meglumine (JAN) <JP/US> |
| Fidaxomicin (JAN/USAN) <JP/US> |
| Teneligliptin |
| Teneligliptin (INN) |
| Teneligliptin hydrobromide hydrate (JAN) <JP> |
| Teneligliptin hydrobromide (JAN) |
| Berotralstat |
| Berotralstat (USAN/INN) |
| Berotralstat hydrochloride (JAN/USAN) <JP/US> |
| Verapamil |
| Verapamil (USAN/INN) |
| Verapamil hydrochloride (JP18/USP) <JP/US> |
| Ketoconazole (JP18/USP) <JP/US> |
| Fluconazole |
| Fluconazole (JP18/USP/INN) <JP/US> |
| Fosfluconazole (JAN/INN) <JP> |
| Luliconazole (JAN/USAN/INN) <JP/US> |
| Bromocriptine |
| Bromocriptine (USAN/INN) |
| Bromocriptine mesylate (USP); Bromocriptine mesilate (JP18) <JP/US> |
| Ethinylestradiol |
| Ethinyl estradiol (USP); Ethinylestradiol (JP18/INN) <JP> |
| Ethinylestradiol propanesulfonate |
| Midecamycin |
| Midecamycin (JP18/INN) |
| Midecamycin acetate (JP18) |
| Josamycin |
| Josamycin (JP18/USAN/INN) |
| Josamycin propionate (JP18) |
| Troleandomycin (USAN/INN); Triacetyloleandomycin (JAN) |
| Clarithromycin |
| Clarithromycin (JP18/USP/INN) <JP/US> |
| Clarithromycin lactobionate |
| Quinupristin and dalfopristin |
| Itraconazole (JP18/USP) <JP/US> |
| Posaconazole (JAN/USAN/INN) <JP/US> |
| Indinavir |
| Indinavir |
| Indinavir (USAN) |
| Indinavir sulfate (USP) |
| Indinavir sulfate ethanolate (JAN) |
| Nelfinavir |
| Nelfinavir (INN) |
| Nelfinavir mesylate (USAN/INN); Nelfinavir mesilate (JAN) <US> |
| Fosamprenavir |
| Fosamprenavir (INN) |
| Fosamprenavir calcium hydrate (JAN) |
| Fosamprenavir calcium (USAN) <US> |
| Fosamprenavir sodium (USAN) |
| Atazanavir |
| Atazanavir (INN) |
| Atazanavir sulfate (JAN/USAN) <US> |
| Darunavir |
| Darunavir (USAN/INN) <US> |
| Darunavir ethanolate (JAN) <JP/US> |
| Darunavir hydrate <US> |
| Darunavir propylene glycolate <US> |
| Telaprevir (JAN/USAN/INN) |
| Dasabuvir, ombitasvir, paritaprevir and ritonavir |
| Ombitasvir, paritaprevir and ritonavir |
| Sirolimus (JAN/USAN/INN) <JP/US> |
| Bicalutamide (JP18/USP/INN) <JP/US> |
| Anastrozole (JP18/USP/INN) <JP/US> |
| Cyclosporine (USP); Ciclosporin (JP18) <JP/US> |
| Stiripentol (JAN/USAN/INN) <JP/US> |
| Istradefylline (JAN/USAN/INN) <JP/US> |
| Fluvoxamine |
| Fluvoxamine (INN) |
| Fluvoxamine maleate (JP18/USP) <JP/US> |
| Aclidinium bromide (JAN/USAN/INN) <JP/US> |
| Fomepizole (JAN/USAN/INN) <JP/US> |
| Carotegrast methyl (JAN) <JP> |
| Miconazole |
| Miconazole (JP18/USP/INN) <JP/US> |
| Miconazole nitrate (JP18/USP) <JP/US> |
| Ranitidine |
| Ranitidine (USAN/INN) |
| Ranitidine hydrochloride (JP18/USP) <US> |
| Ranitidine bismuth citrate (USAN) |
| Lonafarnib (JAN/USAN/INN) <JP/US> |
| Ticagrelor (JAN/USAN/INN) <JP/US> |
| Fostamatinib |
| Fostamatinib (USAN) |
| Fostamatinib disodium (USAN); Fostamatinib sodium hydrate (JAN) <JP/US> |
| Dronedarone |
| Dronedarone (INN) |
| Dronedarone hydrochloride (USP) <US> |
| Conivaptan |
| Conivaptan (INN) |
| Conivaptan hydrochloride (JAN/USAN) |
| Mibefradil |
| Mibefradil (INN) |
| Mibefradil dihydrochloride (USAN) |
| Ravuconazole |
| Ravuconazole (prop.INN) |
| Fosravuconazole L-lysine ethanolate (JAN) <JP> |
| Erythromycin |
| Erythromycin (JP18/USP/INN) <JP/US> |
| Erythromycin estolate (USP); Erythromycin estorate (JAN) |
| Erythromycin ethylsuccinate (JP18/USP) <JP/US> |
| Erythromycin lactobionate (JP18/USP) <JP/US> |
| Erythromycin stearate (JP18/USP) <JP> |
| Erythromycin acistrate (USAN) |
| Erythromycin gluceptate (USP) |
| Erythromycin propionate (USAN) |
| Berythromycin (USAN/INN) |
| Erythromycin salnacedin (USAN) |
| Erythromycin thiocyanate |
| Erythromycin stinoprate (INN) |
| Mifepristone (JAN/USAN/INN) <US> |
| Mifepristone and misoprostol <JP> |
| Telithromycin (JAN/USAN/INN) |
| Norfloxacin |
| Norfloxacin (JP18/USP/INN) <JP> |
| Norfloxacin nicotinate |
| Voriconazole (JP18/USP/INN) <JP/US> |
| Ritonavir (JAN/USP/INN) <JP/US> |
| Amprenavir (JAN/USAN/INN) |
| Ensitrelvir |
| Ensitrelvir (USAN/INN) |
| Ensitrelvir fumarate (USAN); Ensitrelvir fumaric acid (JAN) <JP> |
| Nirmatrelvir and ritonavir <JP/US> |
| Delavirdine |
| Delavirdine (INN) |
| Delavirdine mesylate (USAN); Delavirdine mesilate (JAN) |
| Boceprevir (INN/USAN) |
| Simeprevir |
| Simeprevir (JAN/USAN) |
| Simeprevir sodium (JAN) |
| Daclatasvir |
| Daclatasvir (USAN) |
| Daclatasvir dihydrochloride (USAN); Daclatasvir hydrochloride (JAN) |
| Grazoprevir |
| Grazoprevir (USAN/INN) |
| Grazoprevir (USAN); Grazoprevir hydrate (JAN) |
| Elvitegravir, cobicistat, emtricitabine and tenofovir disoproxil <US> |
| Lopinavir and ritonavir <JP/US> |
| Darunavir and cobicistat <JP/US> |
| Atazanavir and cobicistat <US> |
| Elvitegravir, cobicistat, emtricitabine and tenofovir alafenamide <JP/US> |
| Darunavir, cobicistat, emtricitabine and tenofovir alafenamide <JP/US> |
| Letermovir (JAN/USAN/INN) <JP/US> |
| Crizotinib (JAN/USAN/INN) <JP/US> |
| Ceritinib (JAN/USAN/INN) <JP/US> |
| Pirtobrutinib (JAN/USAN) <JP/US> |
| Entrectinib (JAN/USAN/INN) <JP/US> |
| Ritlecitinib tosylate (USAN); Ritlecitinib tosilate (JAN) <JP/US> |
| Fluoxetine |
| Fluoxetine (USAN/INN) |
| Fluoxetine hydrochloride (JAN/USP) <US> |
| Cobicistat (JAN/USAN/INN) <US> |
| Isavuconazonium |
| Isavuconazonium (USAN) |
| Isavuconazonium sulfate (JAN/USAN) <JP/US> |
| Pimitespib (JAN) <JP> |
| Lopinavir (JAN/USP/INN) |
| Netupitant (USAN/INN) |