PT770615E - Processo para a preparacao de di-haloazolopirimidinas - Google Patents

Processo para a preparacao de di-haloazolopirimidinas

Info

Publication number
PT770615E
PT770615E PT96307528T PT96307528T PT770615E PT 770615 E PT770615 E PT 770615E PT 96307528 T PT96307528 T PT 96307528T PT 96307528 T PT96307528 T PT 96307528T PT 770615 E PT770615 E PT 770615E
Authority
PT
Portugal
Prior art keywords
haloazolopyrimidines
preparation
Prior art date
Application number
PT96307528T
Other languages
English (en)
Inventor
Karl-Otto Stumm
Gunther Krummel
Klaus-Jurgen Pees
Peter Heinz Rudi Liers
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Publication of PT770615E publication Critical patent/PT770615E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PT96307528T 1995-10-27 1996-10-16 Processo para a preparacao de di-haloazolopirimidinas PT770615E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US802295P 1995-10-27 1995-10-27

Publications (1)

Publication Number Publication Date
PT770615E true PT770615E (pt) 2003-10-31

Family

ID=21729405

Family Applications (1)

Application Number Title Priority Date Filing Date
PT96307528T PT770615E (pt) 1995-10-27 1996-10-16 Processo para a preparacao de di-haloazolopirimidinas

Country Status (22)

Country Link
US (1) US5808066A (pt)
EP (1) EP0770615B1 (pt)
JP (1) JP4018182B2 (pt)
KR (1) KR100443182B1 (pt)
AR (1) AR004122A1 (pt)
AT (1) ATE243211T1 (pt)
BR (1) BR9605258A (pt)
CA (1) CA2188905C (pt)
DE (1) DE69628712T2 (pt)
DK (1) DK0770615T3 (pt)
ES (1) ES2202419T3 (pt)
HU (1) HU217773B (pt)
IL (1) IL119496A (pt)
MX (1) MX9604882A (pt)
PT (1) PT770615E (pt)
RU (1) RU2147584C1 (pt)
SG (1) SG55239A1 (pt)
SI (1) SI0770615T1 (pt)
SK (1) SK284071B6 (pt)
TR (1) TR199600792A2 (pt)
UA (1) UA48132C2 (pt)
ZA (1) ZA968957B (pt)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6117876A (en) 1997-04-14 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
BR9907863A (pt) * 1998-02-11 2000-10-24 American Cyanamid Co Composto, processo para a preparação do mesmo, composição fungicida, processo para combater fungo em um local, e, uso do composto ou da composição
US6117865A (en) * 1998-09-10 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
US6380202B1 (en) * 1998-09-25 2002-04-30 Basf Aktiengesellschaft Fungicidal fluoro-substituted 7-heterocyclyl-triazolopyrimidines
US6242451B1 (en) * 1998-09-25 2001-06-05 Klaus-Juergen Pees Fungicidal trihalophenyl-triazolopyrimidines
US6156925A (en) * 1998-09-25 2000-12-05 American Cyanamid Company Process for the preparation of halogenated phenylmaloates
US6559151B2 (en) 2000-05-08 2003-05-06 Basf Aktiengesellschaft 6-(2-trifluoromethyl-phenyl)-triazolopyrimidines
US6939873B2 (en) * 2000-07-26 2005-09-06 Taro Pharmaceuticals Industries Limited Non-sedating barbituric acid derivatives
US7683071B2 (en) * 2000-07-26 2010-03-23 Taro Pharmaceuticals Industries Ltd. Composition and method for improved bioavailability and enhanced brain delivery of 5,5-diphenyl barbituric acid
US6756379B2 (en) 2001-07-26 2004-06-29 Taro Pharmaceutical Industries Ltd. Non-sedating barbiturate compounds as neuroprotective agents
DE10063115A1 (de) * 2000-12-18 2002-06-27 Bayer Ag Triazolopyrimidine
JP2002249492A (ja) * 2000-12-22 2002-09-06 Nippon Bayer Agrochem Co Ltd トリアゾロピリミジン類
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
CA2452625A1 (en) 2001-07-05 2003-01-16 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, method for the production thereof and use thereof in controlling noxious fungi and agents containing said compounds
JP2005504743A (ja) 2001-07-18 2005-02-17 ビーエーエスエフ アクチェンゲゼルシャフト 殺菌薬としての置換された6−(2−メトキシ−フェニル)−トリアゾロピリミジン
UA76486C2 (en) 2001-07-26 2006-08-15 Basf Ag 7-amino triazolopyrimidines, a process of praparation, a fungicidal preparations based thereon and a method to control phytopathogenic fungi
DE60220296T2 (de) 2001-09-04 2008-01-17 Sumitomo Chemical Co., Ltd. IMIDAZO(1,2-a)PYRIMIDINE UND DIESE ENTHALTENDE FUNGIZIDZUSAMMENSETZUNGEN
CA2479766A1 (en) 2002-03-21 2003-10-02 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, methods for producing the same, use thereof for combating harmful fungi and agents containing said substances
ES2315569T3 (es) * 2002-12-11 2009-04-01 Taro Pharmaceutical Industries Ltd. Procedimiento de tratamiento de trastornos del movimiento usando derivados de acido barbiturico.
JP4695595B2 (ja) * 2003-09-24 2011-06-08 ワイス・ホールディングズ・コーポレイション 抗癌剤としての6−アリール−7−ハロ−イミダゾ[1,2−a]ピリミジン類
JP2007506744A (ja) * 2003-09-24 2007-03-22 ワイス・ホールディングズ・コーポレイション 抗癌剤としての6−[(置換)フェニル]トリアゾロピリミジン類
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
MY179926A (en) * 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
TW200533670A (en) * 2003-12-19 2005-10-16 Basf Ag 6-(aminocarbonylphenyl)triazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
DE102004007076A1 (de) * 2004-02-13 2005-08-25 Bayer Cropscience Ag Imidazolopyrimidine
ES2347664T3 (es) 2004-03-10 2010-11-03 Basf Se 5,6-dialquil-7-aminotriazolopirimidinas, el procedimiento para su obtencion y su utilizacion para combatir hongos perjudiciales, asi como los productos que las contienen.
US20070167463A1 (en) * 2004-03-10 2007-07-19 Basf Aktiengesellschaft 5,6-Dialkyl-7-aminotriazolopyrimidines, method for their production, their use for controlling pathogenic fungi, and agents containing said compounds
PE20060020A1 (es) * 2004-03-30 2006-03-10 Basf Ag 5-6-cicloalquil-7-amino-triazolopirimidinas para combatir hongos fitopatogenos y procedimientos para su obtencion
EP1781624A4 (en) * 2004-07-02 2010-06-23 Taro Pharma Ind PROCESS FOR THE PREPARATION OF 1-METHOXYMETHYL-5,5-DIPHENYLBARBITURIC ACID
WO2006092413A1 (de) * 2005-03-01 2006-09-08 Basf Aktiengesellschaft 5,6-dialkyl-7-amino-azolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
TW200640927A (en) * 2005-03-01 2006-12-01 Basf Ag 5,6-Dialkyl-7-aminoazolopyrimidines, their preparation and their use for controlling harmful fungi, and compositions comprising these compounds
US20080188493A1 (en) * 2005-03-01 2008-08-07 Basf Aktiengesellschaft 5,6-Dialkyl-7-Aminoazolopyrimidines, Their Preparation and Their Use For Controlling Harmful Fungi, and Compositions Comprising These Compounds
US20080139581A1 (en) * 2005-03-02 2008-06-12 Basf Aktiengesellschaft 2-Substituted 7-Aminoazolopyrimidines, Processes For Their Preparation And Their Use For Controlling Harmful Fungi, And Compositions Comprising These Compounds
US20080176744A1 (en) * 2005-03-10 2008-07-24 Basf Aktiengesellschaft Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
JP2008533099A (ja) * 2005-03-18 2008-08-21 ビーエーエスエフ ソシエタス・ヨーロピア 5−ハロ−2,4,6−トリフルオロイソフタル酸の製造方法
BRPI0612673A2 (pt) * 2005-06-27 2016-11-29 Basf Ag processo para preparar compostos, compostos, e, uso de compostos
BRPI0612676A2 (pt) * 2005-06-27 2016-11-29 Basf Ag processo para preparar compostos, compostos, e, uso de compostos
EP2081576A4 (en) * 2006-11-14 2010-06-30 Taro Pharmaceuticals North Ame METHOD FOR IMPROVING BIOAVAILABILITY FOR NON-EDMING BARBITURATES
CN101583613A (zh) * 2007-01-11 2009-11-18 巴斯夫欧洲公司 生产芳基取代的稠合嘧啶的方法
US8343977B2 (en) * 2009-12-30 2013-01-01 Arqule, Inc. Substituted triazolo-pyrimidine compounds

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3907799A (en) * 1971-08-16 1975-09-23 Icn Pharmaceuticals Xanthine oxidase inhibitors
JPS5962593A (ja) * 1982-09-30 1984-04-10 Ss Pharmaceut Co Ltd 3―置換―5,7―ジクロルトリアゾロピリミジン誘導体
DE3522463A1 (de) * 1985-06-22 1987-01-02 Bayer Ag Herbizide mittel
US4910306A (en) * 1987-11-09 1990-03-20 The Dow Chemical Company Preparation of substituted 1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US4892945A (en) * 1987-12-21 1990-01-09 Ciba-Geigy Corporation Isoindoline pigments containing at least one triazolopyrimidone radical
US5006656A (en) * 1990-02-26 1991-04-09 Dowelanco Preparation of 5,7-dihydroxy-1,2,4-triazolo[1,5-a]pyrimidine-2-sulfonanilides
US5177206A (en) * 1991-10-08 1993-01-05 Dowelanco Process for the preparation of substituted N-(aryl)-1,2,4-triazolopyrimidine-2-sulfonamides
TW224044B (pt) * 1991-12-30 1994-05-21 Shell Internat Res Schappej B V
IL108731A (en) * 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
CA2171003C (en) * 1993-10-18 2005-12-13 James W. Ringer Process for preparing n-(2,6-dichloro-3-methylphenyl)-5-7-dihalo[1,2,4]triazolo[1,5a]pyrimidine-2-sulfonamide by cyclization and halo-dehydroxylation

Also Published As

Publication number Publication date
UA48132C2 (uk) 2002-08-15
IL119496A0 (en) 1997-01-10
AR004122A1 (es) 1998-09-30
DE69628712T2 (de) 2004-04-29
TR199600792A2 (tr) 1997-05-21
EP0770615A1 (en) 1997-05-02
ZA968957B (en) 1998-04-24
SG55239A1 (en) 1998-12-21
DE69628712D1 (de) 2003-07-24
KR100443182B1 (ko) 2005-04-19
CA2188905A1 (en) 1997-04-28
JPH09124651A (ja) 1997-05-13
US5808066A (en) 1998-09-15
BR9605258A (pt) 1998-07-21
SK284071B6 (sk) 2004-09-08
HUP9602957A2 (en) 1997-06-30
DK0770615T3 (da) 2003-07-14
KR970021081A (ko) 1997-05-28
CA2188905C (en) 2005-12-06
SK137796A3 (en) 1997-05-07
IL119496A (en) 2001-07-24
JP4018182B2 (ja) 2007-12-05
HU9602957D0 (en) 1996-12-30
EP0770615B1 (en) 2003-06-18
HU217773B (hu) 2000-04-28
ES2202419T3 (es) 2004-04-01
MX9604882A (es) 1997-04-30
RU2147584C1 (ru) 2000-04-20
ATE243211T1 (de) 2003-07-15
HUP9602957A3 (en) 1998-01-28
SI0770615T1 (en) 2003-12-31

Similar Documents

Publication Publication Date Title
PT770615E (pt) Processo para a preparacao de di-haloazolopirimidinas
PT1256584E (pt) Processo para a preparacao de adefovir-dipivoxil
BR9710457A (pt) Processo para a prepara-Æo de ciclohexanodimetanol
BR9608471A (pt) Processo para a preparação de um composto
BR9606782A (pt) Processo para preparar ciclopilacetileno
BR9607301A (pt) Processo para a preparação de nootkatone ou nootkatol
BR9711201A (pt) Processo para a prepara-ao de um composto
BR9500668A (pt) Processo para a preparaçao de compostos polialquil-1-oxa- diazaspirodecano
PT824517E (pt) Processo para a preparacao de cloridrato de lercanidipina
BR9609533A (pt) Processo para preparação de 3-hidroxipirazóis n-substituídos
PT877738E (pt) Processo para a preparacao de derivados de fenil-imidazolidina
BR9708077A (pt) Processo para a preparação de um produto de alfa-olefina
BR9500613A (pt) Processo para a preparação contínua de mononitrotoluenos
BR9610887A (pt) Processo para a preparação de um composto
BR9609493A (pt) Processo para a preparação de um composto
BR9301399A (pt) Processo para a preparacao de um monoazocorante
BR9608904A (pt) Processo para a preparação de um composto
PT880498E (pt) Processo para a preparacao de compostos dicetonicos
BR9606199A (pt) Processo para produção de objetos
BR9610294A (pt) Processo para a preparação de um composto
BR9603223A (pt) Processo para a preparação de aminocarboniltriazolinonas substituídas
BR9611833A (pt) Processo para a preparação de dioxoazabiciclo-hexanos
PT1012152E (pt) Processo para a preparacao de oxazafosforina-2-aminas
BR9306316A (pt) Processo para a preparação de hexafluorclorobuteneno
BR9600086A (pt) Processo para a produção de hidroxialcoxibenzofenonas