PL401469A1 - Pochodna azabicykliczna, sposób jej wytwarzania, jej zastosowanie w medycynie oraz zawierajaca pochodna kompozycja - Google Patents
Pochodna azabicykliczna, sposób jej wytwarzania, jej zastosowanie w medycynie oraz zawierajaca pochodna kompozycjaInfo
- Publication number
- PL401469A1 PL401469A1 PL401469A PL40146901A PL401469A1 PL 401469 A1 PL401469 A1 PL 401469A1 PL 401469 A PL401469 A PL 401469A PL 40146901 A PL40146901 A PL 40146901A PL 401469 A1 PL401469 A1 PL 401469A1
- Authority
- PL
- Poland
- Prior art keywords
- derivative
- medicine
- production
- azabicyclic
- composition
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0010121A FR2812635B1 (fr) | 2000-08-01 | 2000-08-01 | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
FR00/10121 | 2000-08-01 | ||
PCT/FR2001/002418 WO2002010172A1 (fr) | 2000-08-01 | 2001-07-24 | Composes azabicycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
Publications (2)
Publication Number | Publication Date |
---|---|
PL401469A1 true PL401469A1 (pl) | 2013-02-04 |
PL234468B1 PL234468B1 (pl) | 2020-02-28 |
Family
ID=8853181
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL365162A PL216028B1 (pl) | 2000-08-01 | 2001-07-24 | Pochodna azabicykliczna, jej zastosowanie jako lek oraz zawierajaca ja kompozycja |
PL401469A PL234468B1 (pl) | 2000-08-01 | 2001-07-24 | Pochodna azabicykliczna, sposób jej wytwarzania, jej zastosowanie w medycynie oraz zawierająca tą pochodną kompozycja |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL365162A PL216028B1 (pl) | 2000-08-01 | 2001-07-24 | Pochodna azabicykliczna, jej zastosowanie jako lek oraz zawierajaca ja kompozycja |
Country Status (42)
Country | Link |
---|---|
US (5) | US7112592B2 (pl) |
EP (1) | EP1307457B1 (pl) |
JP (2) | JP4515704B2 (pl) |
KR (1) | KR100632906B1 (pl) |
CN (1) | CN1289500C (pl) |
AP (1) | AP1614A (pl) |
AR (1) | AR031716A1 (pl) |
AT (1) | ATE263768T1 (pl) |
AU (2) | AU7990501A (pl) |
BG (1) | BG66094B1 (pl) |
BR (1) | BRPI0112986B8 (pl) |
CA (1) | CA2417475C (pl) |
CR (1) | CR6895A (pl) |
CZ (1) | CZ294956B6 (pl) |
DE (1) | DE60102702T2 (pl) |
DK (1) | DK1307457T3 (pl) |
DZ (1) | DZ3397A1 (pl) |
EA (1) | EA004920B1 (pl) |
EC (1) | ECSP034460A (pl) |
EE (1) | EE05183B1 (pl) |
ES (1) | ES2220793T3 (pl) |
FR (1) | FR2812635B1 (pl) |
HK (1) | HK1060356A1 (pl) |
HR (1) | HRP20030034B1 (pl) |
HU (1) | HU226889B1 (pl) |
IL (2) | IL154187A0 (pl) |
MA (1) | MA26938A1 (pl) |
ME (2) | MEP17108A (pl) |
MX (1) | MXPA03000881A (pl) |
NO (1) | NO324940B1 (pl) |
NZ (1) | NZ523707A (pl) |
OA (1) | OA12347A (pl) |
PL (2) | PL216028B1 (pl) |
PT (1) | PT1307457E (pl) |
RS (1) | RS50214B (pl) |
SI (1) | SI1307457T1 (pl) |
SK (1) | SK287597B6 (pl) |
TR (1) | TR200400859T4 (pl) |
TW (1) | TWI292401B (pl) |
UA (1) | UA73791C2 (pl) |
WO (1) | WO2002010172A1 (pl) |
ZA (1) | ZA200300676B (pl) |
Families Citing this family (95)
Publication number | Priority date | Publication date | Assignee | Title |
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FR2812635B1 (fr) * | 2000-08-01 | 2002-10-11 | Aventis Pharma Sa | Nouveaux composes heterocycliques, preparation et utilisation comme medicaments notamment comme anti- bacteriens |
FR2835186B1 (fr) | 2002-01-28 | 2006-10-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, actifs comme inhibiteurs de beta-lactamases |
FR2844273B1 (fr) * | 2002-09-05 | 2008-04-04 | Aventis Pharma Sa | Nouveaux composes heterocycliques, procede et intermediaires de preparation et utilisation comme medicament, notamment comme inhibiteurs de beta-lactamases et anti-bacteriens. |
US7439253B2 (en) * | 2002-12-06 | 2008-10-21 | Novexel | Heterocyclic compounds, their preparation and their use as medicaments, in particular as antibacterials and beta-lactamase inhibitors |
FR2848210B1 (fr) * | 2002-12-06 | 2007-10-19 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens et inhibiteurs de beta-lactamases |
JP5180836B2 (ja) | 2005-12-07 | 2013-04-10 | バジリア ファルマスーチカ アーゲー | モノバクタム系抗生物質とβ−ラクタマーゼ系阻害剤との有用な組み合わせ |
AU2007272839B2 (en) | 2006-07-13 | 2012-05-24 | Achillion Pharmaceuticals, Inc. | 4-amino-4-oxobutanoyl peptides as inhibitors of viral replication |
EP2040698A4 (en) * | 2006-07-14 | 2011-08-10 | Shionogi & Co | OXIM CONNECTIONS AND ITS USE |
AU2007300531A1 (en) * | 2006-09-27 | 2008-04-03 | Merck Sharp & Dohme Corp. | Novel inhibitors of beta-lactamase |
MX2009004290A (es) * | 2006-10-23 | 2009-07-27 | Irm Llc | Inhibidores de proteasas de catepsina. |
US20100056497A1 (en) | 2007-01-31 | 2010-03-04 | Dainippon Sumitomo Pharma Co., Ltd | Amide derivative |
FR2914923B1 (fr) * | 2007-04-12 | 2013-06-14 | Novexel | Nouveaux composes heterocycliques azotes,leur preparation et leur utilisation comme medicaments antibacteriens. |
JP5323063B2 (ja) * | 2007-05-31 | 2013-10-23 | 塩野義製薬株式会社 | オキシイミノ化合物およびその使用 |
FR2921060B1 (fr) * | 2007-09-14 | 2012-06-15 | Novexel | Nouveau procede de preparation d'une piperidine disubsituee et nouveaux intermediaires |
CN101918407B (zh) * | 2008-01-18 | 2014-02-26 | 默沙东公司 | β-内酰胺酶抑制剂 |
ES2408159T3 (es) | 2008-06-11 | 2013-06-18 | Shionogi & Co., Ltd. | Compuestos de oxicarbamoilo y su utilización |
EP2135959A1 (en) | 2008-06-19 | 2009-12-23 | Novexel | Use of (1R,2S,5R) 1,6-Diazabicyclo [3,2,1]octane-2-carboxamide, 7-oxo-6-(sulfooxy)-, monosodium salt as a diagnostic reagent for detecting serine beta-lactamases |
FR2936798B1 (fr) | 2008-10-03 | 2012-09-28 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens. |
FR2937034B1 (fr) | 2008-10-10 | 2012-11-23 | Novexel | Nouveaux composes heterocycliques azotes, leur preparation et leur utilisation comme medicaments antibacteriens |
WO2010126820A2 (en) * | 2009-04-30 | 2010-11-04 | Merck Sharp & Dohme Corp. | Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids |
AU2010263641A1 (en) | 2009-06-24 | 2012-01-19 | Sumitomo Dainippon Pharma Co., Ltd. | N-substituted-cyclic amino derivative |
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US8772490B2 (en) | 2010-12-22 | 2014-07-08 | Meiji Seika Pharma Co., Ltd. | Optically active diazabicyclooctane derivatives and process for preparing the same |
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KR20140144254A (ko) | 2012-03-30 | 2014-12-18 | 큐비스트 파마슈티컬즈 인코포레이티드 | 1,3,4-옥사디아졸 및 1,3,4-티아디아졸 β-락타마제 억제제 |
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KR20210137159A (ko) | 2019-03-12 | 2021-11-17 | 아릭사 파마슈티컬스 인코포레이티드 | 아비박탐 유도체의 결정형 |
US11565999B2 (en) | 2019-04-25 | 2023-01-31 | Arixa Pharmaceuticals, Inc. | Methods of synthesizing aztreonam derivatives |
CN110078728B (zh) * | 2019-05-23 | 2020-10-23 | 江西富祥药业股份有限公司 | 一种阿维巴坦中间体、制备方法及其应用 |
WO2021106864A1 (en) * | 2019-11-25 | 2021-06-03 | Eisai R&D Management Co., Ltd. | Process for the preparation of producing pyrazolo[1,5-a] pyrimidine derivatives |
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JPS4939678B1 (pl) * | 1968-05-06 | 1974-10-28 | ||
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EP0260057A3 (en) * | 1986-09-02 | 1989-02-01 | The University Of Melbourne | 2-oxo-4-carboxy-pyrimidines |
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TW358097B (en) * | 1996-05-24 | 1999-05-11 | Hoffmann La Roche | Beta-lactams and their process and pharmaceutical compositions |
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DE69906059D1 (de) * | 1998-04-20 | 2003-04-24 | Fujisawa Pharmaceutical Co | Anthranilsäurederivate als inhibitoren der c-gmp-phosphodiesterase |
GB9817029D0 (en) * | 1998-08-05 | 1998-09-30 | Smithkline Beecham Plc | Novel compounds |
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