NO803868L - Fremgangsmaate ved fremstilling av nye kinazolinderivater - Google Patents

Fremgangsmaate ved fremstilling av nye kinazolinderivater

Info

Publication number
NO803868L
NO803868L NO803868A NO803868A NO803868L NO 803868 L NO803868 L NO 803868L NO 803868 A NO803868 A NO 803868A NO 803868 A NO803868 A NO 803868A NO 803868 L NO803868 L NO 803868L
Authority
NO
Norway
Prior art keywords
procedure
preparation
new
chinazoline derivatives
chinazoline
Prior art date
Application number
NO803868A
Other languages
English (en)
Other versions
NO154919B (no
NO154919C (no
Inventor
Terence Richard Jones
Kenneth Reginald Harrap
Alan Hilary Calvert
Original Assignee
Nat Res Dev
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nat Res Dev filed Critical Nat Res Dev
Publication of NO803868L publication Critical patent/NO803868L/no
Publication of NO154919B publication Critical patent/NO154919B/no
Publication of NO154919C publication Critical patent/NO154919C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D205/00Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/04Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO803868A 1979-12-19 1980-12-18 Analogifremgangsmaate ved fremstilling av nye kinazolinderivater. NO154919C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB7943715 1979-12-19
GB8006813 1980-02-28

Publications (3)

Publication Number Publication Date
NO803868L true NO803868L (no) 1981-06-22
NO154919B NO154919B (no) 1986-10-06
NO154919C NO154919C (no) 1987-01-14

Family

ID=26273917

Family Applications (1)

Application Number Title Priority Date Filing Date
NO803868A NO154919C (no) 1979-12-19 1980-12-18 Analogifremgangsmaate ved fremstilling av nye kinazolinderivater.

Country Status (17)

Country Link
US (2) US4447608A (no)
EP (1) EP0031237B1 (no)
AU (1) AU543237B2 (no)
CA (1) CA1184900A (no)
DE (1) DE3069468D1 (no)
DK (1) DK157019C (no)
ES (3) ES497884A0 (no)
FI (1) FI76791C (no)
GB (1) GB2065653B (no)
GR (1) GR72847B (no)
HU (1) HU193505B (no)
IE (1) IE51188B1 (no)
IL (1) IL61756A (no)
NO (1) NO154919C (no)
NZ (1) NZ195876A (no)
PT (1) PT72232B (no)
YU (1) YU321180A (no)

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US4818819A (en) * 1986-10-20 1989-04-04 The Trustees Of Princeton University Process for the preparation of fused pyridine compounds
US4902796A (en) * 1986-10-20 1990-02-20 The Trustees Of Princeton University 6-alkenyl and ethynyl derivatives of 2-amino-4-hydroxypyrido[2,3-d]pyrimidines
GB8707053D0 (en) * 1987-03-25 1987-04-29 Ici Plc Anti-tumour agents
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GB8727737D0 (en) * 1987-11-26 1987-12-31 Ici Plc Antitumour agents
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US4996206A (en) * 1989-12-11 1991-02-26 The Trustees Of Princeton University N-(pyrrolo[2,3-d]pyrimidin-3-ylacyl)-glutamic acid derivatives
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US5286726A (en) * 1990-04-12 1994-02-15 The Regents Of The University Of Michigan Difluoroglutamic acid conjugates with folates and anti-folates for the treatment of neoplastic diseases
ZA913730B (en) * 1990-05-30 1992-02-26 Ici Plc Anti-tumor compounds
US6762188B1 (en) 1990-06-19 2004-07-13 Smithkline Beecham Corporation Pharmaceutically active benzoquinazoline compounds
GB9013615D0 (en) * 1990-06-19 1990-08-08 Wellcome Found Pharmaceutical compounds
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US5145854A (en) * 1991-11-27 1992-09-08 Nair Madhavan G 1-formyl-5,8,10-trideazafolates
GB9205320D0 (en) * 1992-03-11 1992-04-22 Ici Plc Anti-tumour compounds
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US5430148A (en) * 1992-03-31 1995-07-04 Agouron Pharmaceuticals, Inc. Antiproliferative quinazolines
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GB9223352D0 (en) * 1992-11-06 1992-12-23 Ici Plc Tricyclic compounds
US5821231A (en) * 1993-12-06 1998-10-13 Cytel Corporation CS-1 peptidomimetics, compositions and methods of using same
CA2177840A1 (en) * 1993-12-06 1995-06-15 Thomas S. Arrhenius Cs-1 peptidomimetics, compositions and methods of using the same
WO1995015973A1 (en) * 1993-12-06 1995-06-15 Cytel Corporation Cs-1 peptidomimetics, compositions and methods of using the same
US5770573A (en) * 1993-12-06 1998-06-23 Cytel Corporation CS-1 peptidomimetics, compositions and methods of using the same
US5804396A (en) * 1994-10-12 1998-09-08 Sugen, Inc. Assay for agents active in proliferative disorders
US5837815A (en) * 1994-12-15 1998-11-17 Sugen, Inc. PYK2 related polypeptide products
US5837524A (en) * 1994-12-15 1998-11-17 Sugen, Inc. PYK2 related polynucleotide products
US5593999A (en) * 1995-06-07 1997-01-14 Nair; Madhavan G. Non-classical folate analogue inhibitors of glycinamide ribonucleotide formyltransferase (GARFT)
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US6716575B2 (en) 1995-12-18 2004-04-06 Sugen, Inc. Diagnosis and treatment of AUR1 and/or AUR2 related disorders
US7119174B2 (en) * 1995-12-18 2006-10-10 Sugen, Inc. Diagnosis and treatment of AUR1 and/or AUR2 related disorders
AU5596998A (en) * 1996-12-11 1998-07-03 New York University Medical Center Pyk2 related products and methods
US6818440B2 (en) * 1997-04-28 2004-11-16 Sugen, Inc. Diagnosis and treatment of alk-7 related disorders
US6228641B1 (en) 1997-05-20 2001-05-08 Sugen, Inc. Diagnosis and treatment of PTP04 related disorders
US7115710B2 (en) * 1997-06-11 2006-10-03 Sugen, Inc. Diagnosis and treatment of PTP related disorders
US6342593B1 (en) 1997-06-11 2002-01-29 Sugen, Inc. Diagnosis and treatment of ALP related disorders
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EP1049786A2 (en) 1998-01-21 2000-11-08 Sugen, Inc. Human orthologues of wart
JP2002522009A (ja) 1998-04-14 2002-07-23 スージェン・インコーポレーテッド Ste−20関連蛋白質キナーゼ
US6861442B1 (en) * 1998-12-30 2005-03-01 Sugen, Inc. PYK2 and inflammation
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US6521607B1 (en) 1999-09-23 2003-02-18 Pharmacia Corporation (R)-chiral halogenated substituted N-phenoxy N-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
US6476057B1 (en) 1999-09-23 2002-11-05 G.D. Searle & Co. Use of substituted N, N-disubstituted cycloalkyl aminoalcohol compounds for inhibiting cholesteryl ester transfer protein activity
US6677382B1 (en) 1999-09-23 2004-01-13 Pharmacia Corporation Substituted N,N-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity
US6835546B1 (en) 1999-10-22 2004-12-28 Pharmacia & Upjohn Company Drosophila G protein coupled receptors, nucleic acids, and methods related to the same
US7364866B2 (en) * 1999-10-22 2008-04-29 Pharmacia & Upjohn Company Drosophila G protein coupled receptors, nucleic acids, and methods related to the same
US20030162223A1 (en) * 1999-10-22 2003-08-28 Lowery David E. Drosophila G protein coupled receptors, nucleic acids, and methods related to the same
US20030082534A1 (en) * 1999-11-16 2003-05-01 Peter Lind Novel G protein-coupled receptors
CA2388865A1 (en) * 1999-11-16 2001-05-25 Pharmacia & Upjohn Company Novel g protein-coupled receptors
US6143776A (en) * 2000-02-02 2000-11-07 Sunesis Pharmaceuticals, Inc. Tosylproline analogs as thymidylate synthase inhibitors
US20030003451A1 (en) * 2000-02-23 2003-01-02 Gabriel Vogeli Novel G protein-coupled receptors
US20030027308A1 (en) * 2000-05-30 2003-02-06 Sugen Incorporated Novel human protein phosphatases identified from genomic sequencing
CA2321345A1 (fr) * 2000-10-02 2002-04-02 Abdelbast Guerfi Utilisation du graphite dans un composite pour reduire l'accumulation de glace
US20040157306A1 (en) * 2000-11-13 2004-08-12 Sugen Incorporated Mammalian protein phosphatases
US20050069976A1 (en) * 2001-02-14 2005-03-31 Peter Lind Protein-coupled receptor
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US3471498A (en) * 1967-08-11 1969-10-07 Parke Davis & Co Certain n-p-((2,4-diamino-6-quinazolinyl)-methyl)benzoylamino acids

Also Published As

Publication number Publication date
DK157019C (da) 1990-03-26
IE51188B1 (en) 1986-10-29
AU543237B2 (en) 1985-04-04
ES8300716A1 (es) 1982-11-01
DK540080A (da) 1981-06-20
EP0031237A1 (en) 1981-07-01
ES508454A0 (es) 1983-08-01
FI76791C (fi) 1988-12-12
GB2065653B (en) 1983-03-09
NO154919B (no) 1986-10-06
US4447608A (en) 1984-05-08
IL61756A0 (en) 1981-01-30
GR72847B (no) 1983-12-07
HU193505B (en) 1987-10-28
FI803957L (fi) 1981-06-20
NO154919C (no) 1987-01-14
PT72232B (en) 1981-11-02
ES497884A0 (es) 1982-11-01
ES8307762A1 (es) 1983-08-01
EP0031237B1 (en) 1984-10-17
US4564616A (en) 1986-01-14
ES8308314A1 (es) 1983-09-01
PT72232A (en) 1981-01-01
NZ195876A (en) 1983-11-18
AU6549580A (en) 1981-06-25
ES508453A0 (es) 1983-09-01
CA1184900A (en) 1985-04-02
GB2065653A (en) 1981-07-01
DE3069468D1 (en) 1984-11-22
IL61756A (en) 1987-02-27
FI76791B (fi) 1988-08-31
DK157019B (da) 1989-10-30
YU321180A (en) 1983-06-30
IE802672L (en) 1981-06-19

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